Target Details
| UniProt AC | Q13563 |
|---|---|
| Gene Symbol | PKD2 |
| Protein Name | Polycystin-2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18109 (Fer4_24) PF08016 (PKD_channel) PF20519 (Polycystin_dom) |
Summary
- Multi-target molecules 29
- Clinical molecules 0
- Avg pChEMBL 7.41
Associated Diseases (1)
Active Molecules (29)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IHAKCSKGCPKKPZ
|
9.0 | IC50 | 2 | — | |
MTXHXAFTVABHOY
|
9.0 | IC50 | 3 | — | |
VWVQWSIGDZWPIL
|
8.7 | IC50 | 2 | — | |
ZYRFDYUCAPSAAJ
|
8.7 | IC50 | 2 | — | |
HCMOZLPTNMKKAS
|
8.2 | IC50 | 3 | — | |
KKMZQQWZVBKDFC
|
8.1 | IC50 | 3 | — | |
VDRJYOAEHZMFEB
|
8.1 | IC50 | 3 | — | |
XNWDRALEEPGBHB
|
8.1 | IC50 | 3 | — | |
YKWMQNUCOUUHQO
|
8.1 | IC50 | 3 | — | |
WXGCJNLWHYWDFU
|
7.7 | IC50 | 3 | — | |
VBWZGQKYVCFADL
|
7.5 | IC50 | 3 | — | |
HXYGELZVZAPWID
|
7.5 | IC50 | 3 | — | |
FTCSRLCKGZJDCK
|
7.3 | IC50 | 3 | — | |
LRYNHRWGDADZKP
|
7.2 | IC50 | 3 | — | |
SFSGIDJMRRLJFG
|
7.2 | IC50 | 3 | — | |
ZIATUPKJNZVSLT
|
7.2 | IC50 | 3 | — | |
ZVKJUDYDWABBFR
|
7.2 | IC50 | 3 | — | |
VAVGLCQDZFLPHS
|
7.1 | IC50 | 3 | — | |
SFSGIDJMRRLJFG
|
7.1 | IC50 | 3 | — | |
CNLCKMDXRXVYMV
|
7.0 | IC50 | 3 | — | |
VJHWVSYYFZRUEK
|
6.9 | IC50 | 3 | — | |
WMFOYAZROOMVDL
|
6.8 | IC50 | 3 | — | |
NDIUYMHNCUTVGE
|
6.8 | Ki | 25 | — | |
PNZJIQBIMCZAKU
|
6.7 | IC50 | 3 | — | |
NVHXHWFKRHCFCI
|
6.6 | IC50 | 3 | — | |
AACFPJSJOWQNBN
|
6.5 | IC50 | 4 | — | |
LTWPQYSXDJCNBR
|
6.4 | IC50 | 3 | — | |
WXGCJNLWHYWDFU
|
6.3 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
6.0 | IC50 | 408 | — |