Target Details
| UniProt AC | Q13557 |
|---|---|
| Gene Symbol | CAMK2D |
| Protein Name | Calcium/calmodulin-dependent protein kinase type II subunit delta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08332 (CaMKII_AD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 150
- Clinical molecules 34
- Avg pChEMBL 6.76
KEGG Pathways (34)
- Adrenergic signaling in cardiomyocytes
- Aldosterone synthesis and secretion
- Amphetamine addiction
- Axon guidance
- Calcium signaling pathway
- Cholinergic synapse
- Circadian entrainment
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Efferocytosis
- ErbB signaling pathway
- Gastric acid secretion
- Glioma
- Glucagon signaling pathway
- GnRH signaling pathway
- HIF-1 signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin secretion
- Lipid and atherosclerosis
- Long-term potentiation
- Melanogenesis
- Necroptosis
- Neurotrophin signaling pathway
- Olfactory transduction
- Oocyte meiosis
- Oxytocin signaling pathway
- Parkinson disease
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Proteoglycans in cancer
- Tuberculosis
- Wnt signaling pathway
- cAMP signaling pathway
Active Molecules (150)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SBFPHSVZEXSHTL
|
6.3 | Ki | 62 | — | |
UDFDIIVNIYWXDM
|
6.3 | Ki | 74 | — | |
UYGYYOIUVFMGKQ
|
6.3 | Ki | 30 | — | |
XSDJOIOVIMPMHD
|
6.3 | Ki | 44 | — | |
APPFRBZOALDJNI
|
6.3 | IC50 | 7 | Yes | |
PBCZSGKMGDDXIJ
|
6.3 | Kd | 68 | Yes | |
SZJYMJNAWBOTEU
|
6.3 | IC50 | 9 | Yes | |
QQWUGDVOUVUTOY
|
6.2 | Kd | 231 | Yes | |
JOOXLOJCABQBSG
|
6.2 | Kd | 139 | — | |
AHJRHEGDXFFMBM
|
6.2 | IC50 | 28 | — | |
ZHJGWYRLJUCMRT
|
6.2 | Kd | 18 | — | |
CHADTINFLWZSKR
|
6.2 | Ki | 26 | — | |
GCBJDOWIQHMCMR
|
6.2 | Ki | 84 | — | |
OWDRQHVEJIYVOI
|
6.2 | Ki | 47 | — | |
SKKRZILJUKYLJS
|
6.2 | Ki | 25 | — | |
SLKCVFPEQGHNSI
|
6.2 | Ki | 29 | — | |
TUJUZVJICDSNLY
|
6.2 | Ki | 19 | — | |
UUWNXFJBBYAMDT
|
6.2 | Ki | 46 | — | |
WUWDLXZGHZSWQZ
|
6.2 | Ki | 41 | — | |
RELJBNLDXPSLLS
|
6.2 | IC50 | 6 | — | |
FBTRDJIPJVBTHV
|
6.2 | IC50 | 6 | — | |
CSGQVNMSRKWUSH
|
6.2 | Kd | 21 | — | |
MGGBYMDAPCCKCT
|
6.2 | Kd | 23 | — | |
XCSNYNNJQSXDKR
|
6.1 | IC50 | 9 | Yes | |
CTNPALGJUAXMMC
|
6.1 | Kd | 151 | — | |
SFDFKLDQKSPRHB
|
6.1 | IC50 | 15 | Yes | |
DKSNLQYRZJKYOC
|
6.1 | Ki | 51 | — | |
DZGATJHVQUFYSK
|
6.1 | Ki | 12 | — | |
HSMUWLLZAZCLHF
|
6.1 | Ki | 25 | — | |
NZVDDFRUBIEKLV
|
6.1 | Ki | 20 | — | |
OWFLADWRSCINST
|
6.1 | Ki | 30 | — | |
RFBPWKMQWSIPEO
|
6.1 | Ki | 28 | — | |
UEIRKXUBXCSHJE
|
6.1 | Ki | 19 | — | |
UVZVWLFSZNPMBS
|
6.1 | Ki | 17 | — | |
XIOOJUQFJYPVLA
|
6.1 | Ki | 17 | — | |
ZGZVRPRSFXRGCF
|
6.1 | Ki | 76 | — | |
DYNHJHQFHQTFTP
|
6.1 | Kd | 38 | — | |
GMZCYCKIXQZORP
|
6.1 | IC50 | 6 | — | |
ADQKGRUFGPUORP
|
6.0 | IC50 | 9 | Yes | |
HTROFVQKJODSCL
|
6.0 | Ki | 11 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KRIUNPBAQZGFQA
|
6.0 | Ki | 76 | — | |
KTWBYGUSEYSRND
|
6.0 | Ki | 28 | — | |
LKUJDAHYLPICSE
|
6.0 | Ki | 24 | — | |
OLVBAUVSICCWEJ
|
6.0 | Ki | 39 | — | |
ORUUEFDGYYTXAF
|
6.0 | Ki | 26 | — | |
RZJKNYACYSIBFY
|
6.0 | IC50 | 4 | — | |
XNWKXXIGSPPPBH
|
6.0 | Ki | 31 | — | |
ZWVZORIKUNOTCS
|
6.0 | Ki | 69 | — | |
ZZSBPGIGIUFJRA
|
6.0 | Kd | 46 | — |