Target Details
| UniProt AC | Q13557 |
|---|---|
| Gene Symbol | CAMK2D |
| Protein Name | Calcium/calmodulin-dependent protein kinase type II subunit delta |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08332 (CaMKII_AD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 150
- Clinical molecules 34
- Avg pChEMBL 6.76
KEGG Pathways (34)
- Adrenergic signaling in cardiomyocytes
- Aldosterone synthesis and secretion
- Amphetamine addiction
- Axon guidance
- Calcium signaling pathway
- Cholinergic synapse
- Circadian entrainment
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Efferocytosis
- ErbB signaling pathway
- Gastric acid secretion
- Glioma
- Glucagon signaling pathway
- GnRH signaling pathway
- HIF-1 signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin secretion
- Lipid and atherosclerosis
- Long-term potentiation
- Melanogenesis
- Necroptosis
- Neurotrophin signaling pathway
- Olfactory transduction
- Oocyte meiosis
- Oxytocin signaling pathway
- Parkinson disease
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Proteoglycans in cancer
- Tuberculosis
- Wnt signaling pathway
- cAMP signaling pathway
Active Molecules (150)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DRCZFJISSIKTPA
|
6.8 | IC50 | 2 | — | |
LPILBMJJRGTKOQ
|
6.8 | Ki | 27 | — | |
LRZYYIZFBXFSJB
|
6.8 | Ki | 69 | — | |
XQVVPGYIWAGRNI
|
6.8 | Ki | 19 | — | |
YUOWJICKAJQZLS
|
6.8 | Ki | 35 | — | |
ZYTFPHRVOZXPGZ
|
6.8 | Ki | 30 | — | |
DJKBFCHOHWZUOH
|
6.8 | IC50 | 7 | Yes | |
SFQZZXBCKCLFFC
|
6.8 | IC50 | 6 | — | |
BDOCJJUGIOCUKN
|
6.8 | IC50 | 7 | Yes | |
MEXUTNIFSHFQRG
|
6.7 | IC50 | 21 | Yes | |
KOZFSFOOLUUIGY
|
6.7 | Kd | 88 | Yes | |
GLMWKEAUVZDGKE
|
6.7 | Ki | 23 | — | |
KWRXWPRFIUJQBP
|
6.7 | Ki | 25 | — | |
RYYNGWLOYLRZLK
|
6.7 | Ki | 104 | — | |
VNGYQBMDQMDALH
|
6.7 | Ki | 25 | — | |
YEHCNYAQEBQCCS
|
6.7 | Ki | 74 | — | |
SDUWPCYMTHMQAZ
|
6.7 | IC50 | 8 | Yes | |
RPSCADUVKLRNEB
|
6.6 | IC50 | 8 | Yes | |
MIKAKZKNMYZLDX
|
6.6 | Ki | 42 | — | |
PLHUMPJXRHMFFR
|
6.6 | Ki | 28 | — | |
SRONQUHCRFZABC
|
6.6 | Ki | 28 | — | |
WDARYLSSWBWVCU
|
6.6 | Ki | 49 | — | |
YMIJUBCSOKSFRU
|
6.6 | Ki | 87 | — | |
ZHBAGBACXDDSPH
|
6.6 | IC50 | 9 | Yes | |
BPNUQXPIQBZCMR
|
6.6 | Kd | 83 | Yes | |
RHXHGRAEPCAFML
|
6.5 | Kd | 9 | — | |
GGUSTVFLQLGLJX
|
6.5 | IC50 | 7 | Yes | |
UQHKJRCFSLMWIA
|
6.5 | IC50 | 3 | — | |
XUZMWHLSFXCVMG
|
6.5 | Kd | 24 | — | |
HOYRWTWZUFFACV
|
6.5 | Ki | 28 | — | |
LSLPDHNUWRDOGC
|
6.5 | Ki | 25 | — | |
OADRBDVURCEKRP
|
6.5 | Ki | 44 | — | |
PIQCTGMSNWUMAF
|
6.5 | Ki | 137 | Yes | |
UYJNQQDJUOUFQJ
|
6.5 | Ki | 68 | — | |
AYCPARAPKDAOEN
|
6.5 | Kd | 73 | — | |
APYXQTXFRIDSGE
|
6.4 | IC50 | 4 | — | |
ATHMTZOFUCSRPV
|
6.4 | IC50 | 7 | Yes | |
RJVLFQBBRSMWHX
|
6.4 | IC50 | 2 | — | |
BGYVWFZMYBWCNY
|
6.4 | Ki | 30 | — | |
CNQGNADBGYCKKV
|
6.4 | Ki | 25 | — | |
DBXGGXLBTWZXBB
|
6.4 | Ki | 39 | — | |
DPEXRCOBPACFOO
|
6.4 | Ki | 36 | — | |
JZTOUVBEZONDKA
|
6.4 | Ki | 80 | — | |
LCHCSKHPVCDXAU
|
6.4 | Ki | 30 | — | |
XXSPHNFKLDJDAK
|
6.4 | Ki | 26 | — | |
NZXJTWVLQGCJJH
|
6.4 | IC50 | 7 | Yes | |
WINHZLLDWRZWRT
|
6.4 | Kd | 201 | Yes | |
AIQDZMUPVYDVLB
|
6.3 | Ki | 48 | — | |
LRINYHMQZRENCY
|
6.3 | Ki | 29 | — | |
NLUPJKQOKWBWFC
|
6.3 | Ki | 69 | — |