Target Details
| UniProt AC | Q13555 |
|---|---|
| Gene Symbol | CAMK2G |
| Protein Name | Calcium/calmodulin-dependent protein kinase type II subunit gamma |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08332 (CaMKII_AD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 123
- Clinical molecules 36
- Avg pChEMBL 6.78
KEGG Pathways (34)
- Adrenergic signaling in cardiomyocytes
- Aldosterone synthesis and secretion
- Amphetamine addiction
- Axon guidance
- Calcium signaling pathway
- Cholinergic synapse
- Circadian entrainment
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Efferocytosis
- ErbB signaling pathway
- Gastric acid secretion
- Glioma
- Glucagon signaling pathway
- GnRH signaling pathway
- HIF-1 signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin secretion
- Lipid and atherosclerosis
- Long-term potentiation
- Melanogenesis
- Necroptosis
- Neurotrophin signaling pathway
- Olfactory transduction
- Oocyte meiosis
- Oxytocin signaling pathway
- Parkinson disease
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Proteoglycans in cancer
- Tuberculosis
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (123)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MEXUTNIFSHFQRG
|
6.7 | IC50 | 21 | Yes | |
UBPYILGKFZZVDX
|
6.7 | IC50 | 130 | Yes | |
DFMCXVONDDGQIY
|
6.7 | Ki | 66 | — | |
GCYXEGSPUDSZJY
|
6.7 | Ki | 82 | — | |
PSCJSWRVCKUMSL
|
6.7 | Ki | 35 | — | |
XQVVPGYIWAGRNI
|
6.7 | Ki | 19 | — | |
SDUWPCYMTHMQAZ
|
6.7 | IC50 | 8 | Yes | |
RPSCADUVKLRNEB
|
6.6 | IC50 | 8 | Yes | |
RHXHGRAEPCAFML
|
6.6 | Kd | 9 | — | |
XUZMWHLSFXCVMG
|
6.6 | Kd | 24 | — | |
MIKAKZKNMYZLDX
|
6.6 | Ki | 42 | — | |
RYYNGWLOYLRZLK
|
6.6 | Ki | 104 | — | |
YUOWJICKAJQZLS
|
6.6 | Ki | 35 | — | |
ZHBAGBACXDDSPH
|
6.6 | IC50 | 9 | Yes | |
AYCPARAPKDAOEN
|
6.6 | Kd | 73 | — | |
GGUSTVFLQLGLJX
|
6.5 | IC50 | 7 | Yes | |
AIQDZMUPVYDVLB
|
6.5 | Ki | 48 | — | |
NLUPJKQOKWBWFC
|
6.5 | Ki | 69 | — | |
OADRBDVURCEKRP
|
6.5 | Ki | 44 | — | |
UDFDIIVNIYWXDM
|
6.5 | Ki | 74 | — | |
WUBHCQHBUVGGRX
|
6.5 | Ki | 11 | — | |
ZGZVRPRSFXRGCF
|
6.5 | Ki | 76 | — | |
ATHMTZOFUCSRPV
|
6.4 | IC50 | 7 | Yes | |
JZTOUVBEZONDKA
|
6.4 | Ki | 80 | — | |
ZYTFPHRVOZXPGZ
|
6.4 | Ki | 30 | — | |
NZXJTWVLQGCJJH
|
6.4 | IC50 | 7 | Yes | |
CLEGDJQQHUTCOW
|
6.3 | Ki | 43 | — | |
DBXGGXLBTWZXBB
|
6.3 | Ki | 39 | — | |
DKSNLQYRZJKYOC
|
6.3 | Ki | 51 | — | |
LRZYYIZFBXFSJB
|
6.3 | Ki | 69 | — | |
NWAUBAGBGOPJLF
|
6.3 | Ki | 51 | Yes | |
SBFPHSVZEXSHTL
|
6.3 | Ki | 62 | — | |
UUWNXFJBBYAMDT
|
6.3 | Ki | 46 | — | |
APPFRBZOALDJNI
|
6.3 | IC50 | 7 | Yes | |
SZJYMJNAWBOTEU
|
6.3 | IC50 | 9 | Yes | |
JOOXLOJCABQBSG
|
6.3 | Kd | 139 | — | |
ARYNBWZQYLWGFJ
|
6.3 | IC50 | 2 | — | |
BNGOYHGMLMEWGU
|
6.3 | IC50 | 2 | — | |
DRCZFJISSIKTPA
|
6.3 | IC50 | 2 | — | |
PQNWNVWJXPSZFR
|
6.2 | Ki | 21 | — | |
UVZVWLFSZNPMBS
|
6.2 | Ki | 17 | — | |
YMIJUBCSOKSFRU
|
6.2 | Ki | 87 | — | |
WINHZLLDWRZWRT
|
6.2 | Kd | 201 | Yes | |
CSGQVNMSRKWUSH
|
6.1 | Kd | 21 | — | |
XCSNYNNJQSXDKR
|
6.1 | IC50 | 9 | Yes | |
DYNHJHQFHQTFTP
|
6.1 | Kd | 38 | — | |
QQWUGDVOUVUTOY
|
6.1 | Kd | 231 | Yes | |
SFDFKLDQKSPRHB
|
6.1 | IC50 | 15 | Yes | |
DJLORVJVWIBDME
|
6.1 | Ki | 24 | — | |
KAKFXRYHYUPXSU
|
6.1 | Ki | 16 | — |