Target Details
| UniProt AC | Q13555 |
|---|---|
| Gene Symbol | CAMK2G |
| Protein Name | Calcium/calmodulin-dependent protein kinase type II subunit gamma |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08332 (CaMKII_AD) PF00069 (Pkinase) |
Summary
- Multi-target molecules 123
- Clinical molecules 36
- Avg pChEMBL 6.78
KEGG Pathways (34)
- Adrenergic signaling in cardiomyocytes
- Aldosterone synthesis and secretion
- Amphetamine addiction
- Axon guidance
- Calcium signaling pathway
- Cholinergic synapse
- Circadian entrainment
- Cushing syndrome
- Diabetic cardiomyopathy
- Dopaminergic synapse
- Efferocytosis
- ErbB signaling pathway
- Gastric acid secretion
- Glioma
- Glucagon signaling pathway
- GnRH signaling pathway
- HIF-1 signaling pathway
- Inflammatory mediator regulation of TRP channels
- Insulin secretion
- Lipid and atherosclerosis
- Long-term potentiation
- Melanogenesis
- Necroptosis
- Neurotrophin signaling pathway
- Olfactory transduction
- Oocyte meiosis
- Oxytocin signaling pathway
- Parkinson disease
- Pathways in cancer
- Pathways of neurodegeneration - multiple diseases
- Proteoglycans in cancer
- Tuberculosis
- Wnt signaling pathway
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (123)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HKSZLNNOFSGOKW
|
9.3 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
9.3 | Kd | 213 | — | |
YISMQBFJYDFMAL
|
9.2 | IC50 | 46 | — | |
MSEGDVOYFLNBPZ
|
9.1 | IC50 | 2 | — | |
ADMFLILDQJSEIK
|
8.4 | Ki | 72 | — | |
NJPWCTYVEJIQBM
|
8.4 | Ki | 72 | — | |
NXSJMRCTGYTSTK
|
8.1 | Kd | 200 | — | |
OSVUGUHRKMMBSE
|
8.1 | Kd | 170 | — | |
UMTWTCVTRDYHQQ
|
8.0 | Ki | 56 | — | |
MWKSRKSEWLRPBL
|
8.0 | Kd | 1075 | — | |
YWTBGJGMTBHQTM
|
7.9 | Ki | 65 | — | |
CHTMRWQLNNRRFJ
|
7.8 | Ki | 70 | — | |
BPNUQXPIQBZCMR
|
7.6 | Ki | 60 | — | |
BSFNGHCTZDCQBF
|
7.6 | Ki | 93 | — | |
KAJXOWFGKYKMMZ
|
7.6 | IC50 | 26 | Yes | |
LEJHMQJABOLACY
|
7.6 | IC50 | 9 | Yes | |
UIARLYUEJFELEN
|
7.6 | Kd | 289 | Yes | |
UZWDCWONPYILKI
|
7.5 | IC50 | 47 | — | |
FUMCKNCUEAQHCV
|
7.5 | Ki | 103 | — | |
KSILWADEZRASEE
|
7.5 | IC50 | 4 | — | |
NOVLXWHGKLXEJS
|
7.4 | IC50 | 4 | — | |
ZCCPLJOKGAACRT
|
7.4 | Kd | 599 | — | |
OWRXHGAFWZFFCW
|
7.4 | Ki | 113 | — | |
WINHZLLDWRZWRT
|
7.4 | Ki | 66 | — | |
APALQVMWCDGRJB
|
7.3 | IC50 | 9 | Yes | |
AILRADAXUVEEIR
|
7.3 | IC50 | 75 | — | |
ZNEQEOGXKINPPR
|
7.3 | IC50 | 9 | Yes | |
GDYZFFBMSBDTAA
|
7.3 | Ki | 60 | — | |
PCQMERRARZKTPW
|
7.3 | Ki | 68 | — | |
VXYDJXMHISGSDA
|
7.3 | Ki | 59 | — | |
LAMWYYXJYIQOQL
|
7.2 | IC50 | 16 | Yes | |
GPNZOTCLQNMQIC
|
7.2 | IC50 | 7 | Yes | |
MVJMMLFMPWITEJ
|
7.2 | Ki | 110 | — | |
OAVGBZOFDPFGPJ
|
7.1 | Ki | 42 | Yes | |
XPHWIERLJBFPFV
|
7.1 | Ki | 69 | — | |
XOFQJBDORDALAH
|
7.1 | IC50 | 9 | Yes | |
ZPEBZVFGLUUCDX
|
7.1 | IC50 | 6 | — | |
WMUGNCAVDUVWIE
|
7.0 | IC50 | 9 | Yes | |
CHOKPCNUYFDUDO
|
7.0 | IC50 | 9 | Yes | |
BRGYPSBHCUNPNP
|
7.0 | IC50 | 9 | Yes | |
HFNKQEVNSGCOJV
|
7.0 | Kd | 65 | — | |
XFWUTMHVDGPWLH
|
7.0 | Ki | 75 | — | |
YEHCNYAQEBQCCS
|
6.9 | Ki | 74 | — | |
BMGQWWVMWDBQGC
|
6.8 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.8 | Kd | 91 | Yes | |
GLMWKEAUVZDGKE
|
6.8 | Ki | 23 | — | |
DJKBFCHOHWZUOH
|
6.8 | IC50 | 7 | Yes | |
KOZFSFOOLUUIGY
|
6.8 | Kd | 88 | Yes | |
SFQZZXBCKCLFFC
|
6.8 | IC50 | 6 | — | |
BDOCJJUGIOCUKN
|
6.8 | IC50 | 7 | Yes |