Target Details
| UniProt AC | Q13546 |
|---|---|
| Gene Symbol | RIPK1 |
| Protein Name | Receptor-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00531 (Death) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 315
- Clinical molecules 6
- Avg pChEMBL 8.13
KEGG Pathways (16)
- Alcoholic liver disease
- Apoptosis
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis C
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Necroptosis
- Pathogenic Escherichia coli infection
- RIG-I-like receptor signaling pathway
- Salmonella infection
- Shigellosis
- TNF signaling pathway
- Toll-like receptor signaling pathway
Associated Diseases (2)
Active Molecules (315)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CZEXAUZTGDVUEV
|
7.2 | IC50 | 2 | — | |
ASFRLTODYTWPAU
|
7.2 | IC50 | 2 | — | |
SNRUTMWCDZHKKM
|
7.2 | Kd | 4 | — | |
YYLKKYCXAOBSRM
|
7.2 | Kd | 191 | — | |
INFXTIWUPWDDQY
|
7.2 | IC50 | 2 | — | |
PRWSIEBRGXYXAJ
|
7.2 | IC50 | 4 | — | |
QAEKSWBVYBVLNO
|
7.2 | IC50 | 5 | — | |
VYZYOJULVVGQRS
|
7.2 | IC50 | 2 | — | |
AIGWTZNVNIYEJA
|
7.2 | IC50 | 2 | — | |
WCZYJWNVPLJLFK
|
7.2 | IC50 | 2 | — | |
KMBAXSMUNQBQTG
|
7.1 | IC50 | 2 | — | |
BKDBTNDUTIFYHL
|
7.1 | IC50 | 2 | — | |
WCZYJWNVPLJLFK
|
7.1 | IC50 | 2 | — | |
JRUKWWHAQPEKAA
|
7.1 | IC50 | 2 | — | |
MVEBCLACXCZCEB
|
7.1 | IC50 | 2 | — | |
WGSZIBOZZBGNJW
|
7.0 | IC50 | 2 | — | |
ZQSZVECJMJELSV
|
7.0 | IC50 | 2 | — | |
MPVGZUGXCQEXTM
|
7.0 | IC50 | 61 | Yes | |
AVPUTQITOHDIOV
|
7.0 | Kd | 2 | — | |
SDSQERWTMKMZLA
|
7.0 | Kd | 2 | — | |
VLTNUYNTYZRWQD
|
7.0 | IC50 | 4 | — | |
DVBXOBNOQIIWQT
|
7.0 | IC50 | 2 | — | |
XIRIJHPESRRPNP
|
6.8 | IC50 | 2 | — | |
KDCYOEAWXNGQEB
|
6.8 | IC50 | 3 | — | |
LHCHFIVFJHGCNI
|
6.8 | IC50 | 2 | — | |
FXGOMJXGESCWPD
|
6.8 | IC50 | 2 | — | |
TXUWMXQFNYDOEZ
|
6.7 | IC50 | 2 | — | |
UFWJGUUHERHCOL
|
6.7 | IC50 | 3 | — | |
BXVRODNTVCIXSZ
|
6.7 | Kd | 2 | — | |
QMILKASSWHCTOF
|
6.7 | IC50 | 4 | — | |
RGPRFYTUFVLMEL
|
6.7 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
6.7 | Kd | 153 | — | |
NFUVBUNETZNUIB
|
6.7 | Kd | 2 | — | |
GUBJNPWVIUFSTR
|
6.6 | Kd | 103 | — | |
WFWVJTWOJNJWJW
|
6.6 | Kd | 2 | — | |
XZXHXSATPCNXJR
|
6.6 | Kd | 165 | Yes | |
CUIHSIWYWATEQL
|
6.6 | Kd | 61 | Yes | |
UFWXSGVSQZKZTR
|
6.5 | IC50 | 4 | — | |
FDRXUDVPGMWNHL
|
6.5 | IC50 | 2 | — | |
JNZKENWWCGIHDV
|
6.5 | IC50 | 3 | — | |
OJUQYRUOIGTYSD
|
6.5 | IC50 | 2 | — | |
PIQCTGMSNWUMAF
|
6.5 | Kd | 137 | Yes | |
VMXQAQDFSBPASA
|
6.5 | Kd | 2 | — | |
JTQDNMQENCMSFD
|
6.4 | IC50 | 2 | — | |
WINHZLLDWRZWRT
|
6.4 | Kd | 201 | Yes | |
NXCZMDQVFMPBOI
|
6.4 | IC50 | 2 | — | |
ASFRLTODYTWPAU
|
6.4 | IC50 | 2 | — | |
WANGYKOAXRTHJB
|
6.4 | Kd | 2 | — | |
OJFKUJDRGJSAQB
|
6.3 | Kd | 17 | — | |
WANGYKOAXRTHJB
|
6.3 | Kd | 2 | — |