Target Details
| UniProt AC | Q13546 |
|---|---|
| Gene Symbol | RIPK1 |
| Protein Name | Receptor-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00531 (Death) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 315
- Clinical molecules 6
- Avg pChEMBL 8.13
KEGG Pathways (16)
- Alcoholic liver disease
- Apoptosis
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis C
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Necroptosis
- Pathogenic Escherichia coli infection
- RIG-I-like receptor signaling pathway
- Salmonella infection
- Shigellosis
- TNF signaling pathway
- Toll-like receptor signaling pathway
Associated Diseases (2)
Active Molecules (315)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PHXJVRSECIGDHY
|
7.9 | IC50 | 59 | — | |
VRQMAABPASPXMW
|
7.9 | IC50 | 8 | — | |
FEDLMIZRTVANRW
|
7.9 | IC50 | 2 | — | |
ARUQRSCNTGVZST
|
7.9 | IC50 | 2 | — | |
KNDPXYAMINMLED
|
7.9 | IC50 | 11 | — | |
YMDRTFUXHKMYKK
|
7.9 | IC50 | 2 | — | |
FEDLMIZRTVANRW
|
7.9 | IC50 | 2 | — | |
QWVQHMXZDUMKQL
|
7.9 | IC50 | 2 | — | |
RLKXEZDLONNHDZ
|
7.8 | IC50 | 2 | — | |
AGYFORVGFVMPGZ
|
7.8 | IC50 | 2 | — | |
BSHFVIJHRDSZBW
|
7.8 | IC50 | 2 | — | |
JGKVEIHLYOIAKC
|
7.8 | IC50 | 2 | — | |
QWVQHMXZDUMKQL
|
7.8 | IC50 | 2 | — | |
VCATZNOHJNXWNN
|
7.8 | IC50 | 2 | — | |
PPJWJOYOOLVOPL
|
7.7 | IC50 | 2 | — | |
SIXVRXARNAVBTC
|
7.7 | IC50 | 12 | — | |
HKDBKENBVSIISE
|
7.7 | IC50 | 2 | — | |
HKDBKENBVSIISE
|
7.7 | IC50 | 2 | — | |
PPTQWMQTXBVAHT
|
7.7 | Kd | 2 | — | |
SZNYUUZOQHNEKB
|
7.7 | IC50 | 7 | — | |
DUHJQNPBNDWRPM
|
7.7 | IC50 | 2 | — | |
GCIKSSRWRFVXBI
|
7.7 | Kd | 109 | Yes | |
LSVIBAPJYUUVJJ
|
7.7 | IC50 | 4 | — | |
BBCKARALJWASLJ
|
7.7 | IC50 | 2 | — | |
DUHJQNPBNDWRPM
|
7.7 | IC50 | 2 | — | |
KDKXJCPRPAGSRR
|
7.7 | IC50 | 2 | — | |
XXYRQJUSJPPEAS
|
7.7 | IC50 | 2 | — | |
CRWZLQDCAINIKP
|
7.6 | IC50 | 2 | — | |
KZCPUGTZKJUVSG
|
7.6 | IC50 | 2 | — | |
BSHFVIJHRDSZBW
|
7.6 | IC50 | 2 | — | |
HKDBKENBVSIISE
|
7.6 | IC50 | 2 | — | |
JLIIFVXHGLWALL
|
7.6 | IC50 | 2 | — | |
XXXNLTQQWQAHRA
|
7.6 | IC50 | 2 | — | |
RBBVTNBEGNSCQJ
|
7.5 | IC50 | 2 | — | |
ZLIMBNIXPSWXRS
|
7.5 | IC50 | 2 | — | |
IBZKREARIHWPAX
|
7.4 | IC50 | 2 | — | |
IUSXFQNTDSJZSX
|
7.4 | IC50 | 2 | — | |
VCATZNOHJNXWNN
|
7.4 | IC50 | 2 | — | |
BSHFVIJHRDSZBW
|
7.4 | IC50 | 2 | — | |
LHCHFIVFJHGCNI
|
7.4 | IC50 | 2 | — | |
QGNBGHSJBKSEAE
|
7.4 | IC50 | 2 | — | |
WXNOXFAWDUEBAQ
|
7.4 | IC50 | 2 | — | |
NXCZMDQVFMPBOI
|
7.4 | IC50 | 2 | — | |
MBZJKJGRSPJARC
|
7.3 | IC50 | 2 | — | |
FUARSVCNRXAGKF
|
7.3 | IC50 | 2 | — | |
LMJOMRYRQJWXNS
|
7.3 | IC50 | 2 | — | |
MBZJKJGRSPJARC
|
7.3 | IC50 | 2 | — | |
LZTBBNONIGEIKH
|
7.3 | Kd | 2 | — | |
PZBUOCXBGCVSAF
|
7.3 | Kd | 2 | — | |
MXJOJOBEDQVCNB
|
7.2 | IC50 | 2 | — |