Target Details
| UniProt AC | Q13546 |
|---|---|
| Gene Symbol | RIPK1 |
| Protein Name | Receptor-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00531 (Death) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 315
- Clinical molecules 6
- Avg pChEMBL 8.13
KEGG Pathways (16)
- Alcoholic liver disease
- Apoptosis
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis C
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Necroptosis
- Pathogenic Escherichia coli infection
- RIG-I-like receptor signaling pathway
- Salmonella infection
- Shigellosis
- TNF signaling pathway
- Toll-like receptor signaling pathway
Associated Diseases (2)
Active Molecules (315)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CLGXFAOGUWTIIO
|
8.4 | IC50 | 2 | — | |
MAHFVAHPQSLLJF
|
8.4 | Ki | 288 | — | |
XUZTUIGKADFQTD
|
8.4 | IC50 | 2 | — | |
AIGWTZNVNIYEJA
|
8.4 | IC50 | 2 | — | |
JRUKWWHAQPEKAA
|
8.4 | IC50 | 2 | — | |
RGPRFYTUFVLMEL
|
8.4 | IC50 | 2 | — | |
ILYGNYJWIRLLTD
|
8.4 | IC50 | 2 | — | |
GKXMLAZADXCTFY
|
8.4 | IC50 | 2 | — | |
YSBWBLIHHMJTAY
|
8.4 | IC50 | 2 | — | |
ZDFKAHHMHOYWBF
|
8.3 | IC50 | 2 | — | |
MVFLEIABXLOCKI
|
8.3 | IC50 | 2 | — | |
DNWHHGJZSGNIPU
|
8.3 | IC50 | 2 | — | |
JBHRNPLTGWTGHX
|
8.3 | IC50 | 2 | — | |
XUZTUIGKADFQTD
|
8.3 | IC50 | 2 | — | |
RGPRFYTUFVLMEL
|
8.3 | IC50 | 2 | — | |
FDJIJMTZXHXLBI
|
8.3 | IC50 | 2 | — | |
WNBHLRSJGCOCPC
|
8.3 | IC50 | 2 | — | |
VLBBPJJXSYYNQP
|
8.2 | IC50 | 2 | — | |
XXNLYFOKFFASDY
|
8.2 | IC50 | 2 | — | |
JLIIFVXHGLWALL
|
8.2 | IC50 | 2 | — | |
KDKJFCOXFFFARW
|
8.2 | IC50 | 2 | — | |
OQLPCBATCBGXCA
|
8.2 | IC50 | 2 | — | |
NXCZMDQVFMPBOI
|
8.2 | IC50 | 2 | — | |
DNWHHGJZSGNIPU
|
8.2 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
8.2 | IC50 | 92 | — | |
XZBGRGYKTKCJDO
|
8.2 | IC50 | 2 | — | |
XOSHQHWNDZFWKX
|
8.2 | IC50 | 2 | — | |
APPXQUDJLJXULP
|
8.2 | IC50 | 47 | — | |
BPKSNNJTKPIZKR
|
8.1 | IC50 | 2 | — | |
KCPIWHYTGKDOQZ
|
8.1 | IC50 | 2 | — | |
MLULYTTTYREQGB
|
8.1 | IC50 | 2 | — | |
FHMPYPIPCWQXEJ
|
8.1 | IC50 | 2 | — | |
KNJIEFIBWDIOPD
|
8.1 | IC50 | 2 | — | |
SHJHUJPYBYTPPG
|
8.1 | IC50 | 2 | — | |
WNBHLRSJGCOCPC
|
8.1 | IC50 | 2 | — | |
IUSXFQNTDSJZSX
|
8.1 | IC50 | 2 | — | |
LZEJBUBDGUVITP
|
8.1 | IC50 | 2 | — | |
GKXMLAZADXCTFY
|
8.1 | IC50 | 2 | — | |
KDKXJCPRPAGSRR
|
8.1 | IC50 | 2 | — | |
KMBAXSMUNQBQTG
|
8.1 | IC50 | 2 | — | |
AYEGXXOXIOWXCD
|
8.1 | IC50 | 2 | — | |
QOMIPWZFCYOBMP
|
8.1 | IC50 | 2 | — | |
INFXTIWUPWDDQY
|
8.0 | IC50 | 2 | — | |
JLIIFVXHGLWALL
|
8.0 | IC50 | 2 | — | |
MVFLEIABXLOCKI
|
8.0 | IC50 | 2 | — | |
NOSHXUYWLDKLQJ
|
8.0 | IC50 | 2 | — | |
NQNSGMASKOVWNF
|
8.0 | IC50 | 2 | — | |
WGLQAYNJIFOANO
|
8.0 | IC50 | 2 | — | |
IGCKQIYIOKUNKB
|
8.0 | IC50 | 2 | — | |
ZCSNBHBTCQUAPF
|
8.0 | IC50 | 2 | — |