Target Details
| UniProt AC | Q13546 |
|---|---|
| Gene Symbol | RIPK1 |
| Protein Name | Receptor-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00531 (Death) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 315
- Clinical molecules 6
- Avg pChEMBL 8.13
KEGG Pathways (16)
- Alcoholic liver disease
- Apoptosis
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis C
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Necroptosis
- Pathogenic Escherichia coli infection
- RIG-I-like receptor signaling pathway
- Salmonella infection
- Shigellosis
- TNF signaling pathway
- Toll-like receptor signaling pathway
Associated Diseases (2)
Active Molecules (315)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OZMDCWDZDUUPCT
|
8.8 | IC50 | 2 | — | |
WHVHKBUPSUSYAL
|
8.8 | IC50 | 2 | — | |
FNRCSGQLGPGABP
|
8.7 | IC50 | 2 | — | |
IGCKQIYIOKUNKB
|
8.7 | IC50 | 2 | — | |
COCLXHBFUGZJBI
|
8.7 | IC50 | 2 | — | |
COCLXHBFUGZJBI
|
8.7 | IC50 | 2 | — | |
CRWZLQDCAINIKP
|
8.7 | IC50 | 2 | — | |
JCWYGDFYFWPQJD
|
8.7 | IC50 | 2 | — | |
NKNSMRWBHMCQTM
|
8.7 | IC50 | 2 | — | |
FDJIJMTZXHXLBI
|
8.7 | IC50 | 2 | — | |
ZJEITEDIBHPUSP
|
8.7 | IC50 | 2 | — | |
CLGXFAOGUWTIIO
|
8.7 | IC50 | 2 | — | |
GKXMLAZADXCTFY
|
8.7 | IC50 | 2 | — | |
XFLHXLODOOXMPE
|
8.7 | IC50 | 2 | — | |
ZUNSWLPTCRBOFX
|
8.7 | IC50 | 2 | — | |
QYIXADVHPFHXME
|
8.6 | IC50 | 2 | — | |
XUZTUIGKADFQTD
|
8.6 | IC50 | 2 | — | |
YMDRTFUXHKMYKK
|
8.6 | IC50 | 2 | — | |
ZJEITEDIBHPUSP
|
8.6 | IC50 | 2 | — | |
ITGRJBYMENVRNL
|
8.6 | IC50 | 2 | — | |
OOHWXVMNYAIFBU
|
8.6 | IC50 | 2 | — | |
PPSGHPXXRRIFGL
|
8.6 | IC50 | 2 | — | |
KCPIWHYTGKDOQZ
|
8.6 | IC50 | 2 | — | |
WKRKPIJCVMARCO
|
8.6 | IC50 | 2 | — | |
XPLCUEPEVWREIT
|
8.6 | IC50 | 2 | — | |
COCLXHBFUGZJBI
|
8.6 | IC50 | 2 | — | |
KCPIWHYTGKDOQZ
|
8.6 | IC50 | 2 | — | |
YMDRTFUXHKMYKK
|
8.6 | IC50 | 2 | — | |
ZJEITEDIBHPUSP
|
8.6 | IC50 | 2 | — | |
FDJIJMTZXHXLBI
|
8.6 | IC50 | 2 | — | |
FDJIJMTZXHXLBI
|
8.6 | IC50 | 2 | — | |
NXCZMDQVFMPBOI
|
8.6 | IC50 | 2 | — | |
KNIULYCUWOGHSI
|
8.6 | IC50 | 2 | — | |
MOYKEIUKAWAETD
|
8.6 | IC50 | 2 | — | |
SHJHUJPYBYTPPG
|
8.6 | IC50 | 2 | — | |
ALAZXNZFIANJMN
|
8.5 | IC50 | 2 | — | |
ATMWMZOSKFLIGS
|
8.5 | IC50 | 2 | — | |
MOYKEIUKAWAETD
|
8.5 | IC50 | 2 | — | |
UBLHPXNZDKOECN
|
8.5 | IC50 | 2 | — | |
FQTJUEYKGHZUES
|
8.5 | IC50 | 2 | — | |
ASFRLTODYTWPAU
|
8.5 | IC50 | 2 | — | |
IKYVVXPGERUFKR
|
8.5 | IC50 | 2 | — | |
NUYXPCXEOUUXIA
|
8.5 | IC50 | 2 | — | |
MVEBCLACXCZCEB
|
8.5 | IC50 | 2 | — | |
ZUNSWLPTCRBOFX
|
8.5 | IC50 | 2 | — | |
AVNYULWTERJTEY
|
8.4 | IC50 | 2 | — | |
FHMPYPIPCWQXEJ
|
8.4 | IC50 | 2 | — | |
ABECYZZLHDZIOZ
|
8.4 | IC50 | 2 | — | |
JBHRNPLTGWTGHX
|
8.4 | IC50 | 2 | — | |
XXYRQJUSJPPEAS
|
8.4 | IC50 | 2 | — |