Target Details
| UniProt AC | Q13546 |
|---|---|
| Gene Symbol | RIPK1 |
| Protein Name | Receptor-interacting serine/threonine-protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00531 (Death) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 315
- Clinical molecules 6
- Avg pChEMBL 8.13
KEGG Pathways (16)
- Alcoholic liver disease
- Apoptosis
- Cytosolic DNA-sensing pathway
- Epstein-Barr virus infection
- Hepatitis C
- Human cytomegalovirus infection
- Human immunodeficiency virus 1 infection
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Necroptosis
- Pathogenic Escherichia coli infection
- RIG-I-like receptor signaling pathway
- Salmonella infection
- Shigellosis
- TNF signaling pathway
- Toll-like receptor signaling pathway
Associated Diseases (2)
Active Molecules (315)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GQVHRJHJTSLMII
|
9.0 | IC50 | 2 | — | |
GQVHRJHJTSLMII
|
9.0 | IC50 | 2 | — | |
MIUSSYJRPWRECR
|
9.0 | IC50 | 2 | — | |
MRYPBXQDXGBARZ
|
9.0 | IC50 | 2 | — | |
MRYPBXQDXGBARZ
|
9.0 | IC50 | 2 | — | |
PENDQBTWOLHSKH
|
9.0 | IC50 | 2 | — | |
UBLHPXNZDKOECN
|
9.0 | IC50 | 2 | — | |
UGQKUBUQYPHWQD
|
9.0 | IC50 | 2 | — | |
XCTMAPWBKRRVPM
|
9.0 | IC50 | 2 | — | |
YSBWBLIHHMJTAY
|
9.0 | IC50 | 2 | — | |
CNYNPLQCTPSHJT
|
9.0 | IC50 | 2 | — | |
RVGCSKSAZFLLMP
|
9.0 | IC50 | 2 | — | |
CNYNPLQCTPSHJT
|
9.0 | IC50 | 2 | — | |
DPXSEFVBHQPHJW
|
9.0 | IC50 | 2 | — | |
RBBVTNBEGNSCQJ
|
9.0 | IC50 | 2 | — | |
SNACPLHRWSDHBB
|
9.0 | IC50 | 2 | — | |
UGQKUBUQYPHWQD
|
9.0 | IC50 | 2 | — | |
YTBVDZYESXPMNS
|
9.0 | IC50 | 2 | — | |
AGYFORVGFVMPGZ
|
8.9 | IC50 | 2 | — | |
FQTJUEYKGHZUES
|
8.9 | IC50 | 2 | — | |
ITGRJBYMENVRNL
|
8.9 | IC50 | 2 | — | |
VDFIPIOXCKVOHD
|
8.9 | IC50 | 2 | — | |
WHVHKBUPSUSYAL
|
8.9 | IC50 | 2 | — | |
WKRKPIJCVMARCO
|
8.9 | IC50 | 2 | — | |
XCTMAPWBKRRVPM
|
8.9 | IC50 | 2 | — | |
GPXNCTKGLKXRLY
|
8.9 | IC50 | 2 | — | |
DXPDLSPXAQNOCK
|
8.9 | IC50 | 2 | — | |
LVGZUKBSCYYWMC
|
8.9 | IC50 | 2 | — | |
NUYXPCXEOUUXIA
|
8.9 | IC50 | 2 | — | |
OKTKFTUTVQYYFJ
|
8.9 | IC50 | 2 | — | |
WKRKPIJCVMARCO
|
8.9 | IC50 | 2 | — | |
GVKUVROQJDFDPO
|
8.8 | IC50 | 2 | — | |
GVNGLGMOHLFLJG
|
8.8 | IC50 | 2 | — | |
KNJIEFIBWDIOPD
|
8.8 | IC50 | 2 | — | |
LWGOFWWGJAJUKJ
|
8.8 | IC50 | 2 | — | |
NOSHXUYWLDKLQJ
|
8.8 | IC50 | 2 | — | |
PKHQKYDPPNNWGZ
|
8.8 | IC50 | 2 | — | |
XIPVJEOSHKSCNE
|
8.8 | IC50 | 2 | — | |
XYVQOYARHKRTFN
|
8.8 | IC50 | 2 | — | |
DQKRPRPKEWJOMT
|
8.8 | IC50 | 2 | — | |
IKYVVXPGERUFKR
|
8.8 | IC50 | 2 | — | |
QXDDBMBCCRLQMR
|
8.8 | IC50 | 2 | — | |
SHJHUJPYBYTPPG
|
8.8 | IC50 | 2 | — | |
ZJUJVFQXYFFLSK
|
8.8 | IC50 | 2 | — | |
ZJUJVFQXYFFLSK
|
8.8 | IC50 | 2 | — | |
IUSXFQNTDSJZSX
|
8.8 | IC50 | 2 | — | |
GRNPQAUIFHUTSP
|
8.8 | IC50 | 2 | — | |
RVGCSKSAZFLLMP
|
8.8 | IC50 | 2 | — | |
MIUSSYJRPWRECR
|
8.8 | IC50 | 2 | — | |
NIQNYGCQGCERBQ
|
8.8 | IC50 | 2 | — |