Target Details
| UniProt AC | Q13541 |
|---|---|
| Gene Symbol | EIF4EBP1 |
| Protein Name | Eukaryotic translation initiation factor 4E-binding protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05456 (eIF_4EBP) |
Summary
- Multi-target molecules 358
- Clinical molecules 0
- Avg pChEMBL 6.82
KEGG Pathways (15)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cellular senescence
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- ErbB signaling pathway
- HIF-1 signaling pathway
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- Longevity regulating pathway
- PI3K-Akt signaling pathway
- mTOR signaling pathway
Active Molecules (358)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RSLLZOSASJVFBJ
|
6.0 | IC50 | 2 | — | |
UCTNDDUDPRBCJE
|
6.0 | IC50 | 2 | — | |
VPTYLIGDGTUUET
|
6.0 | IC50 | 2 | — | |
YPWCSDHWZJKCPB
|
6.0 | IC50 | 2 | — | |
HPWSGFGIKNOPOQ
|
6.0 | IC50 | 2 | — | |
NZPUGYRDIMWBAR
|
6.0 | IC50 | 2 | — | |
KLRDTUBOFCWLPG
|
6.0 | IC50 | 2 | — | |
DWPYAYCRPGWLPV
|
6.0 | IC50 | 2 | — |