Target Details
| UniProt AC | Q13541 |
|---|---|
| Gene Symbol | EIF4EBP1 |
| Protein Name | Eukaryotic translation initiation factor 4E-binding protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05456 (eIF_4EBP) |
Summary
- Multi-target molecules 358
- Clinical molecules 0
- Avg pChEMBL 6.82
KEGG Pathways (15)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cellular senescence
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- ErbB signaling pathway
- HIF-1 signaling pathway
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- Longevity regulating pathway
- PI3K-Akt signaling pathway
- mTOR signaling pathway
Active Molecules (358)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GGYDQJOIDXXNAD
|
6.7 | IC50 | 2 | — | |
NESWARBIGUFKHF
|
6.7 | IC50 | 2 | — | |
QECSLTSUPKPCOK
|
6.7 | IC50 | 2 | — | |
RGEHFHLXCNKTKG
|
6.7 | IC50 | 2 | — | |
YBHPXJIMTWMEJT
|
6.7 | IC50 | 2 | — | |
AXPGIAWEDLKSJN
|
6.7 | IC50 | 2 | — | |
MQGRZGUCHDKHNR
|
6.7 | IC50 | 2 | — | |
XJNNUINBYKQHBT
|
6.7 | IC50 | 2 | — | |
XQZNBIAOAZZLSL
|
6.7 | IC50 | 2 | — | |
DUXSJWIIUXEQQE
|
6.7 | IC50 | 2 | — | |
OFGNLXBZBTYXBG
|
6.7 | IC50 | 2 | — | |
BXPHNMPXKAJHHY
|
6.7 | IC50 | 2 | — | |
RCFBNHQDAJWNCA
|
6.7 | IC50 | 2 | — | |
UADVXORRMJPTDS
|
6.6 | IC50 | 2 | — | |
VZDBDEYISQDTBM
|
6.6 | IC50 | 2 | — | |
DKUZBXNXNHWZKA
|
6.6 | IC50 | 2 | — | |
FNBKWJVELNIWLT
|
6.6 | IC50 | 2 | — | |
HZOJZTFEDPTFSO
|
6.6 | IC50 | 2 | — | |
LKSCUIYYIYTNTE
|
6.6 | IC50 | 2 | — | |
CLLWUPCFDBDWON
|
6.6 | IC50 | 2 | — | |
JLBJJIDIWBSTIA
|
6.6 | IC50 | 2 | — | |
SVPOWBUEBDEALD
|
6.6 | IC50 | 2 | — | |
HWKXZBQFLIMONN
|
6.6 | IC50 | 2 | — | |
YCVYHOCIKNJWRL
|
6.6 | IC50 | 2 | — | |
FPOCBLRVVDFIOQ
|
6.6 | IC50 | 2 | — | |
RZUCBMAANBDFJB
|
6.6 | IC50 | 2 | — | |
NOKMYNQVCCHVIR
|
6.6 | IC50 | 2 | — | |
FNLSJKPQJLPUGU
|
6.6 | IC50 | 2 | — | |
IFIYBCBXLAZUDH
|
6.6 | IC50 | 2 | — | |
BGGOSKLBAUHBDA
|
6.6 | IC50 | 2 | — | |
CVGGBQOMIMFPPO
|
6.6 | IC50 | 2 | — | |
DQSCMYJOJSQDON
|
6.6 | IC50 | 2 | — | |
JBFJLZSRJTYSON
|
6.6 | IC50 | 2 | — | |
LMFWUHGJVXWUSA
|
6.6 | IC50 | 2 | — | |
NGJOYTHCGJOPSB
|
6.6 | IC50 | 2 | — | |
RINLRGAXKQYLIS
|
6.5 | IC50 | 2 | — | |
CELAWHXBDAYIJN
|
6.5 | IC50 | 2 | — | |
YVQRQYJXSJQAQQ
|
6.5 | IC50 | 2 | — | |
HDFFYDVYQRNIRG
|
6.5 | IC50 | 2 | — | |
XKKSAFGGYRQHRP
|
6.5 | IC50 | 2 | — | |
XSFPZWZGEDLCKA
|
6.5 | IC50 | 2 | — | |
DKUZBXNXNHWZKA
|
6.5 | IC50 | 2 | — | |
PYKOTVUQLKQSBL
|
6.5 | IC50 | 2 | — | |
FHPHKMHCGAXDJN
|
6.5 | IC50 | 2 | — | |
NDSXIYRSQWELFU
|
6.5 | IC50 | 2 | — | |
OTHYFALQZBNKFZ
|
6.5 | IC50 | 2 | — | |
XZFRDVYLKDGXDJ
|
6.5 | IC50 | 2 | — | |
LBWPISKIJQPZBG
|
6.5 | IC50 | 2 | — | |
MOZHYIOMDQDQSC
|
6.5 | IC50 | 2 | — | |
OSVXRFQNFDFQOR
|
6.5 | IC50 | 2 | — |