Target Details
| UniProt AC | Q13541 |
|---|---|
| Gene Symbol | EIF4EBP1 |
| Protein Name | Eukaryotic translation initiation factor 4E-binding protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05456 (eIF_4EBP) |
Summary
- Multi-target molecules 358
- Clinical molecules 0
- Avg pChEMBL 6.82
KEGG Pathways (15)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cellular senescence
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- ErbB signaling pathway
- HIF-1 signaling pathway
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- Longevity regulating pathway
- PI3K-Akt signaling pathway
- mTOR signaling pathway
Active Molecules (358)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BVJMFJYEYXOKIR
|
6.9 | IC50 | 2 | — | |
IYPKDTLBOJKBLA
|
6.9 | IC50 | 2 | — | |
NQJSLIMBLRMYFC
|
6.9 | IC50 | 2 | — | |
OMODKRMMOUGEIV
|
6.9 | IC50 | 2 | — | |
CLLFCBFCIOEDIY
|
6.9 | IC50 | 2 | — | |
FNJYGWXOHJRMBU
|
6.9 | IC50 | 2 | — | |
LYZLGXPMHYYYFT
|
6.9 | IC50 | 2 | — | |
CMWFYQDSBGBXTD
|
6.9 | IC50 | 2 | — | |
GGYDQJOIDXXNAD
|
6.9 | IC50 | 2 | — | |
AHJYPGQPZSIWTJ
|
6.9 | IC50 | 2 | — | |
AKORDSRNMHCEGR
|
6.9 | IC50 | 2 | — | |
MWZDMGXGOPCHIL
|
6.9 | IC50 | 2 | — | |
SUAYPYXLCIZIKW
|
6.9 | IC50 | 2 | — | |
VFSUHKOBBKTMEB
|
6.9 | IC50 | 2 | — | |
LVWAWJDFZBIZLL
|
6.9 | IC50 | 2 | — | |
SIWYGZQLUWEPFI
|
6.9 | IC50 | 2 | — | |
UNOQCUYQBYKAKH
|
6.9 | IC50 | 2 | — | |
ZENIUFRGSIDYDD
|
6.9 | IC50 | 2 | — | |
BCANLOWELFOMRO
|
6.9 | IC50 | 2 | — | |
JDNVKUHTVLWBAH
|
6.9 | IC50 | 2 | — | |
MQVFFOPWPVDQCQ
|
6.9 | IC50 | 2 | — | |
YAWYOCPEWTUYCH
|
6.9 | IC50 | 2 | — | |
IBFVXHTUIMMYLU
|
6.8 | IC50 | 2 | — | |
KTCRMYZFFGNMPG
|
6.8 | IC50 | 2 | — | |
UTIVDLSAKSYZOG
|
6.8 | IC50 | 2 | — | |
AOTOIICCFQTTEQ
|
6.8 | IC50 | 2 | — | |
FUTBNXOGIIEFAJ
|
6.8 | IC50 | 2 | — | |
JJLMNZPGWQJXGI
|
6.8 | IC50 | 2 | — | |
OSBIPPWRAXAMBO
|
6.8 | IC50 | 2 | — | |
BHDYLHVNHVDDKS
|
6.8 | IC50 | 2 | — | |
JOSDAYWFWADPST
|
6.8 | IC50 | 2 | — | |
RGIMIYIDJJUSFN
|
6.8 | IC50 | 2 | — | |
SAVAYDMRDFIIQZ
|
6.8 | IC50 | 2 | — | |
YUCZZMOTXCKDJU
|
6.8 | IC50 | 2 | — | |
NVIQRXPGZDMBQA
|
6.8 | IC50 | 2 | — | |
NFYQQSYXVKUCCT
|
6.8 | IC50 | 2 | — | |
CRZPODWMHZOFNR
|
6.8 | IC50 | 2 | — | |
UDBICAGHRVNBMK
|
6.8 | IC50 | 2 | — | |
ATLBSXNUGRIZMX
|
6.8 | IC50 | 2 | — | |
KOKKZTUCYCIGLZ
|
6.8 | IC50 | 2 | — | |
SRBDAAHEZZEWGL
|
6.8 | IC50 | 2 | — | |
XJNNUINBYKQHBT
|
6.8 | IC50 | 2 | — | |
FIFQOOFOISFGPG
|
6.7 | IC50 | 2 | — | |
DECXTCNNSOQVGW
|
6.7 | IC50 | 2 | — | |
OEXCDEUJESZFMP
|
6.7 | IC50 | 2 | — | |
YNSQFVJJPOAFKI
|
6.7 | IC50 | 2 | — | |
IIMUGTCVSMQHBT
|
6.7 | IC50 | 2 | — | |
OFMDSONOVVHNML
|
6.7 | IC50 | 2 | — | |
WNTUAMVHPLRERV
|
6.7 | IC50 | 2 | — | |
CBDGAYOSNQGGCK
|
6.7 | IC50 | 2 | — |