Target Details
| UniProt AC | Q13541 |
|---|---|
| Gene Symbol | EIF4EBP1 |
| Protein Name | Eukaryotic translation initiation factor 4E-binding protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05456 (eIF_4EBP) |
Summary
- Multi-target molecules 358
- Clinical molecules 0
- Avg pChEMBL 6.82
KEGG Pathways (15)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cellular senescence
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- ErbB signaling pathway
- HIF-1 signaling pathway
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- Longevity regulating pathway
- PI3K-Akt signaling pathway
- mTOR signaling pathway
Active Molecules (358)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FRDABAGCZROUAQ
|
7.1 | IC50 | 2 | — | |
QCDHLPHOYLKMTM
|
7.1 | IC50 | 2 | — | |
VHTVUPUAIGVZSV
|
7.1 | IC50 | 2 | — | |
XFBHLCKHGYCSBE
|
7.1 | IC50 | 2 | — | |
NIICOGRNEQTQIR
|
7.1 | IC50 | 2 | — | |
NJSJSWLFDFRFTE
|
7.1 | IC50 | 2 | — | |
JYJHGZINGZGSNW
|
7.1 | IC50 | 2 | — | |
UFMSYLHFOHJGCA
|
7.1 | IC50 | 2 | — | |
FONXCRIWQVSSMY
|
7.1 | IC50 | 2 | — | |
LYDYVTHVNXVDII
|
7.1 | IC50 | 2 | — | |
MVUIDPBVBKMPMO
|
7.1 | IC50 | 2 | — | |
QJBMWGZRUUEZHG
|
7.1 | IC50 | 2 | — | |
UWHJOJFSLYJIJP
|
7.1 | IC50 | 2 | — | |
JHKXOLFIJJMDNJ
|
7.1 | IC50 | 2 | — | |
ACYYKSBFJRQCIP
|
7.0 | IC50 | 2 | — | |
NIXRXQKDQGSXJP
|
7.0 | IC50 | 2 | — | |
SDXSWTUMDYCRGM
|
7.0 | IC50 | 2 | — | |
SSRXIEXJJQECJW
|
7.0 | IC50 | 2 | — | |
AKORDSRNMHCEGR
|
7.0 | IC50 | 2 | — | |
TVPDFYOLAMKSBS
|
7.0 | IC50 | 2 | — | |
WAGGFGZFYGBCCS
|
7.0 | IC50 | 2 | — | |
COMZQGZNVCZCRG
|
7.0 | IC50 | 2 | — | |
HEEHFNCDPGEWFO
|
7.0 | IC50 | 2 | — | |
WFCDKASIYRHWNV
|
7.0 | IC50 | 2 | — | |
IDXJXNORFKDAJG
|
7.0 | IC50 | 2 | — | |
MVUIDPBVBKMPMO
|
7.0 | IC50 | 2 | — | |
NHANZHHEBNMTLH
|
7.0 | IC50 | 2 | — | |
VYTGIYXPWUXYOK
|
7.0 | IC50 | 2 | — | |
MUJZPGJHMHTNNP
|
7.0 | IC50 | 2 | — | |
QHUHWHHMXRIFPD
|
7.0 | IC50 | 2 | — | |
WPDVFZRSYJNWPR
|
7.0 | IC50 | 2 | — | |
CCDAMXZGPBFFJA
|
7.0 | IC50 | 2 | — | |
ADQDEDWKTWBPRE
|
7.0 | IC50 | 2 | — | |
FTYNGPOXJWSFOU
|
7.0 | IC50 | 2 | — | |
DHRBLTKJQMOWJP
|
7.0 | IC50 | 2 | — | |
LIQUWRNMKAPUML
|
7.0 | IC50 | 2 | — | |
QWUAXKYGKQVBII
|
7.0 | IC50 | 2 | — | |
FBZPWWQIICDRCM
|
7.0 | IC50 | 2 | — | |
FUTBNXOGIIEFAJ
|
7.0 | IC50 | 2 | — | |
HOYQJXSPBVEPKQ
|
7.0 | IC50 | 2 | — | |
HNYPHJYMMJPWPA
|
6.9 | IC50 | 2 | — | |
YNPVGOBHTWGSRF
|
6.9 | IC50 | 2 | — | |
GEWKLKKHXXAEBK
|
6.9 | IC50 | 2 | — | |
KAEBLGCBBNJALL
|
6.9 | IC50 | 2 | — | |
ZNXMLFCQOGVKKP
|
6.9 | IC50 | 2 | — | |
FHMBJQUMBGPPMR
|
6.9 | IC50 | 2 | — | |
PBAUKBUFZJRMKW
|
6.9 | IC50 | 2 | — | |
QTBWMULTLYFJLH
|
6.9 | IC50 | 2 | — | |
ZBKJIOFGFMYADW
|
6.9 | IC50 | 2 | — | |
ZGKAPTCEJSSYAH
|
6.9 | IC50 | 2 | — |