Target Details
| UniProt AC | Q13541 |
|---|---|
| Gene Symbol | EIF4EBP1 |
| Protein Name | Eukaryotic translation initiation factor 4E-binding protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05456 (eIF_4EBP) |
Summary
- Multi-target molecules 358
- Clinical molecules 0
- Avg pChEMBL 6.82
KEGG Pathways (15)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cellular senescence
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- ErbB signaling pathway
- HIF-1 signaling pathway
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- Longevity regulating pathway
- PI3K-Akt signaling pathway
- mTOR signaling pathway
Active Molecules (358)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZAAJUKAVVSLHLS
|
7.4 | IC50 | 2 | — | |
CYPIPAWOVNZEIW
|
7.4 | IC50 | 2 | — | |
XOAIPYGZUPIDQG
|
7.4 | IC50 | 2 | — | |
FQWALNMWAZFEIZ
|
7.4 | IC50 | 2 | — | |
ONDBCZKTKORVJM
|
7.4 | IC50 | 2 | — | |
FCMGDNPJWSBTBA
|
7.4 | IC50 | 2 | — | |
QYHVTAWDQUJTLQ
|
7.4 | IC50 | 2 | — | |
CBJSJPHQJZZZBJ
|
7.4 | IC50 | 2 | — | |
DPDKXRXCVGMVEM
|
7.4 | IC50 | 2 | — | |
IGQIUZMLIZEOQJ
|
7.4 | IC50 | 2 | — | |
JHYSJUKQCDHYGF
|
7.3 | IC50 | 2 | — | |
APXACZNSDJVBSQ
|
7.3 | IC50 | 2 | — | |
RWKKVHPRIRQYRI
|
7.3 | IC50 | 2 | — | |
YHVOSMJSFVOFMQ
|
7.3 | IC50 | 2 | — | |
SHQQUJAKINJZNK
|
7.3 | IC50 | 2 | — | |
UYQQKLAVLNUUHG
|
7.3 | IC50 | 2 | — | |
KLPNFMUYMCNKEH
|
7.3 | IC50 | 2 | — | |
BHGLEQQCJLBHBN
|
7.3 | IC50 | 2 | — | |
KDGGQHGWEXXQMX
|
7.3 | IC50 | 2 | — | |
LQBOHPIFHZAHIW
|
7.3 | IC50 | 2 | — | |
VWKBLWNCMYPXNT
|
7.3 | IC50 | 2 | — | |
MHYSMEKJTZKCOY
|
7.3 | IC50 | 2 | — | |
OAWASDLQTXZOGB
|
7.3 | IC50 | 2 | — | |
RWKKVHPRIRQYRI
|
7.3 | IC50 | 2 | — | |
WECYZHCCVIBACH
|
7.3 | IC50 | 2 | — | |
NHVXZKPKHCFZNZ
|
7.3 | IC50 | 2 | — | |
NNDCZVVJUNTIFC
|
7.3 | IC50 | 2 | — | |
OBIGDDPHTXVOJZ
|
7.3 | IC50 | 2 | — | |
QCWNJJVJHYUHDA
|
7.2 | IC50 | 2 | — | |
SRZPPPLVIWOXKV
|
7.2 | IC50 | 2 | — | |
OCFDWLYZPXUNDH
|
7.2 | IC50 | 2 | — | |
VCEWVFDKQWQGRN
|
7.2 | IC50 | 2 | — | |
ZFHZFVWDHGSTDZ
|
7.2 | IC50 | 2 | — | |
BRUWHQQTGREOMP
|
7.2 | IC50 | 2 | — | |
NIIUWQZAJDHQLS
|
7.2 | IC50 | 2 | — | |
YRIVXOLOXTUIBC
|
7.2 | IC50 | 2 | — | |
DVIIUTBOLKCXRG
|
7.2 | IC50 | 2 | — | |
FWCSMTRMWRLHPK
|
7.2 | IC50 | 2 | — | |
PBHGZSPFSJSBLB
|
7.2 | IC50 | 2 | — | |
WDKUVFOQBLPPGF
|
7.2 | IC50 | 2 | — | |
CYJWXNOPHVYBKD
|
7.2 | IC50 | 2 | — | |
FGUDFCKQOZFVKP
|
7.2 | IC50 | 2 | — | |
FXCVSCBHVMQRPG
|
7.2 | IC50 | 2 | — | |
LRONEBCMCIAYJY
|
7.2 | IC50 | 2 | — | |
TZQFJVKLBOSVRQ
|
7.2 | IC50 | 2 | — | |
JVVLREAUZPIBNO
|
7.2 | IC50 | 2 | — | |
KPPRNNNLUVSXFC
|
7.2 | IC50 | 2 | — | |
PPSMGSQSDNLTNZ
|
7.2 | IC50 | 2 | — | |
XDAQWJJXEGGVBI
|
7.2 | IC50 | 2 | — | |
PLUNAYMYYPXSQP
|
7.1 | IC50 | 2 | — |