Target Details
| UniProt AC | Q13541 |
|---|---|
| Gene Symbol | EIF4EBP1 |
| Protein Name | Eukaryotic translation initiation factor 4E-binding protein 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF05456 (eIF_4EBP) |
Summary
- Multi-target molecules 358
- Clinical molecules 0
- Avg pChEMBL 6.82
KEGG Pathways (15)
- AMPK signaling pathway
- Acute myeloid leukemia
- Cellular senescence
- Chemical carcinogenesis - receptor activation
- Choline metabolism in cancer
- EGFR tyrosine kinase inhibitor resistance
- ErbB signaling pathway
- HIF-1 signaling pathway
- Herpes simplex virus 1 infection
- Human cytomegalovirus infection
- Human papillomavirus infection
- Insulin signaling pathway
- Longevity regulating pathway
- PI3K-Akt signaling pathway
- mTOR signaling pathway
Active Molecules (358)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YFVARPBUZODTDL
|
8.5 | IC50 | 2 | — | |
KNZHZDWUGNKVCU
|
8.5 | IC50 | 2 | — | |
QVELPJBQWXPQJO
|
8.2 | IC50 | 2 | — | |
QPVXYFHYJBFCJN
|
8.1 | IC50 | 2 | — | |
IYPVCRHLVNPFHJ
|
8.1 | IC50 | 2 | — | |
XKWJHHAYVXZFEF
|
8.0 | IC50 | 2 | — | |
LWKKZQMIGMNFSQ
|
8.0 | IC50 | 2 | — | |
XGQVCYOBJAAXCY
|
8.0 | IC50 | 2 | — | |
QDOZHMYJWLOMAS
|
8.0 | IC50 | 2 | — | |
IRHZIZQNZWWCOP
|
7.9 | IC50 | 2 | — | |
IRHZIZQNZWWCOP
|
7.8 | IC50 | 2 | — | |
NWEQKJXRHPHOIG
|
7.8 | IC50 | 2 | — | |
PXLKGSDMUOWMFV
|
7.8 | IC50 | 2 | — | |
REWHONSUJOGBSP
|
7.8 | IC50 | 2 | — | |
BKLNVBNDWQJWOW
|
7.8 | IC50 | 2 | — | |
CJKHQVNBWXKDTR
|
7.8 | IC50 | 2 | — | |
JLRPXTBJBURBLI
|
7.8 | IC50 | 2 | — | |
QGBFIHKPDFHDTK
|
7.8 | IC50 | 2 | — | |
KYSMYUDUVPJVFP
|
7.7 | IC50 | 2 | — | |
OSZBAAQZFLOQIZ
|
7.7 | IC50 | 2 | — | |
RWIHQKQFGCEDMX
|
7.7 | IC50 | 2 | — | |
ZUBOOCCOALVOHE
|
7.7 | IC50 | 2 | — | |
LGJJFSHLUIESDI
|
7.7 | IC50 | 2 | — | |
RETSUKLFWSEHIK
|
7.6 | IC50 | 2 | — | |
LWCPSARTNBDWEF
|
7.6 | IC50 | 2 | — | |
WOTQDOAJRCJXMX
|
7.6 | IC50 | 2 | — | |
GQZURLKXQIWZOU
|
7.6 | IC50 | 2 | — | |
HOEORLXMBLMYQD
|
7.6 | IC50 | 2 | — | |
WEPNNXIAUNIUFX
|
7.6 | IC50 | 2 | — | |
GZZCERFOTCZFRM
|
7.5 | IC50 | 2 | — | |
IJLXLRYLWIBFNB
|
7.5 | IC50 | 2 | — | |
WLJJSIKKUZHWOH
|
7.5 | IC50 | 2 | — | |
KAVXXSSHPDJWOJ
|
7.5 | IC50 | 2 | — | |
PVMFBCHMZMAAJU
|
7.5 | IC50 | 2 | — | |
RWGAKXQRQXBVSB
|
7.5 | IC50 | 2 | — | |
PXLKGSDMUOWMFV
|
7.5 | IC50 | 2 | — | |
OXPBOTXWIBDJSR
|
7.5 | IC50 | 2 | — | |
MLGTXVZNEUGPAF
|
7.5 | IC50 | 2 | — | |
QNHIVCKLFHCFFL
|
7.5 | IC50 | 2 | — | |
WOQNMPVKPFWHGY
|
7.5 | IC50 | 2 | — | |
OQDAEOSEGGLQFE
|
7.5 | IC50 | 2 | — | |
XZHVESSSRWBYAX
|
7.5 | IC50 | 2 | — | |
HGNXTQDUTZQGAT
|
7.5 | IC50 | 2 | — | |
GJCSHJOVYLNJJW
|
7.5 | IC50 | 2 | — | |
PXPNZYBGNMWLJP
|
7.5 | IC50 | 2 | — | |
VSXZKELYMHCWQK
|
7.5 | IC50 | 2 | — | |
XYAALDPZFCIYBJ
|
7.5 | IC50 | 2 | — | |
YSOIMYNBQHTJBM
|
7.4 | IC50 | 2 | — | |
QZAIQPBWXIAOGQ
|
7.4 | IC50 | 2 | — | |
YHVOSMJSFVOFMQ
|
7.4 | IC50 | 2 | — |