Target Details
| UniProt AC | Q13535 |
|---|---|
| Gene Symbol | ATR |
| Protein Name | Serine/threonine-protein kinase ATR |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02259 (FAT) PF02260 (FATC) PF23593 (HEAT_ATR) PF25030 (M-HEAT_ATR) PF25032 (N-HEAT_ATR) PF00454 (PI3_PI4_kinase) PF08064 (UME) |
Summary
- Multi-target molecules 749
- Clinical molecules 0
- Avg pChEMBL 7.26
KEGG Pathways (7)
Associated Diseases (2)
Active Molecules (749)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HDEFPSLBSGSNJP
|
8.1 | IC50 | 2 | — | |
AAOWFOJFVUVELU
|
8.1 | IC50 | 5 | — | |
DCVVQEGQUHXZHH
|
8.1 | IC50 | 2 | — | |
UCURUMIOUNMOIW
|
8.1 | IC50 | 5 | — | |
IBZFTEIXMCWYFZ
|
8.1 | IC50 | 2 | — | |
XICUSQBAQPGQPR
|
8.1 | IC50 | 2 | — | |
BCPQAFMDNKIZDR
|
8.1 | IC50 | 2 | — | |
BRGUQOISTYVOBM
|
8.1 | IC50 | 2 | — | |
BTSQQLQBVZAAPN
|
8.1 | IC50 | 2 | — | |
GFPADOXPUVWONC
|
8.1 | IC50 | 2 | — | |
LGCYSSLIKLXLGP
|
8.1 | IC50 | 2 | — | |
XMRWLWQHRURMCJ
|
8.1 | IC50 | 2 | — | |
XPSOVSGFOFAMHM
|
8.1 | IC50 | 2 | — | |
VQRIKGUNZDKECM
|
8.0 | IC50 | 2 | — | |
ZOONXTMYZJYHGZ
|
8.0 | IC50 | 2 | — | |
PUKGKZKXDAYXGE
|
8.0 | IC50 | 2 | — | |
QVHPJUVSFRPYAB
|
8.0 | IC50 | 2 | — | |
XDWMVLMBPVLMJU
|
8.0 | IC50 | 2 | — | |
DVPUUPYVTPQLKN
|
8.0 | IC50 | 2 | — | |
FBNBXXUPCZPXHZ
|
8.0 | IC50 | 5 | — | |
IGVKRFFAXWAUKB
|
8.0 | IC50 | 2 | — | |
IRAFDUYEUVGWMA
|
8.0 | IC50 | 2 | — | |
OHOFYMYNIHAJOB
|
8.0 | IC50 | 2 | — | |
OIYSXDOSZSGSBD
|
8.0 | IC50 | 2 | — | |
PAEFRKXGUAROEW
|
8.0 | IC50 | 2 | — | |
VOVKUEBSMPEEHC
|
8.0 | IC50 | 2 | — | |
WEYDDJKJZQNJEX
|
8.0 | IC50 | 2 | — | |
ZJKUSJSSUAQWIZ
|
8.0 | IC50 | 2 | — | |
ZKNAKMCADIOISC
|
8.0 | IC50 | 5 | — | |
MWKSRKSEWLRPBL
|
8.0 | Kd | 1075 | — | |
VELJXSNFROECOU
|
8.0 | IC50 | 2 | — | |
JPJAHPRMACPWEW
|
8.0 | IC50 | 2 | — | |
TXEQGTLUSHXVQT
|
8.0 | IC50 | 2 | — | |
XTVCYRIFUFASTE
|
8.0 | IC50 | 2 | — | |
BSPZDIRDBAUPEG
|
8.0 | IC50 | 2 | — | |
JLZXCKXHOJJPOR
|
8.0 | IC50 | 2 | — | |
ROPCSAYESHEAEI
|
8.0 | IC50 | 2 | — | |
DWPDDGARZOCDAG
|
7.9 | IC50 | 2 | — | |
KNDFCORKVNCDSE
|
7.9 | IC50 | 2 | — | |
VCUIFULJTLGNAV
|
7.9 | IC50 | 2 | — | |
CFIWMFHGZXJCCO
|
7.9 | IC50 | 2 | — | |
GNEFGLFGNKFHAR
|
7.9 | IC50 | 2 | — | |
JFASXZPYFCTYNF
|
7.9 | IC50 | 2 | — | |
PQZRQQJFBGSJAY
|
7.9 | IC50 | 2 | — | |
SKPPEINHCIBGKD
|
7.9 | IC50 | 2 | — | |
XCTGUZFTYAWGDL
|
7.9 | IC50 | 2 | — | |
LNMBSFNTFNLWGE
|
7.9 | IC50 | 2 | — | |
MSULNMGXCWJIOP
|
7.9 | IC50 | 2 | — | |
VGCZMUWEPHMXQH
|
7.9 | IC50 | 2 | — | |
WLVBJQUVPORFNZ
|
7.9 | IC50 | 2 | — |