Target Details
| UniProt AC | Q13535 |
|---|---|
| Gene Symbol | ATR |
| Protein Name | Serine/threonine-protein kinase ATR |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02259 (FAT) PF02260 (FATC) PF23593 (HEAT_ATR) PF25030 (M-HEAT_ATR) PF25032 (N-HEAT_ATR) PF00454 (PI3_PI4_kinase) PF08064 (UME) |
Summary
- Multi-target molecules 749
- Clinical molecules 0
- Avg pChEMBL 7.26
KEGG Pathways (7)
Associated Diseases (2)
Active Molecules (749)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ADGHHBMQUXGGFP
|
8.4 | IC50 | 5 | — | |
CHMDAOJBIGUHQC
|
8.4 | IC50 | 5 | — | |
DTDLHHWBDQLEOL
|
8.4 | IC50 | 2 | — | |
GVOLNWLXBNDZFA
|
8.4 | IC50 | 5 | — | |
KEBPTIFOURCVEJ
|
8.4 | IC50 | 3 | — | |
MFKMYMWETJVOSR
|
8.4 | IC50 | 5 | — | |
NXOLIFWGYRQEFT
|
8.4 | IC50 | 5 | — | |
QOCIHCAHGWGNEB
|
8.4 | IC50 | 5 | — | |
ZVOIZFFFPDDJHJ
|
8.4 | IC50 | 2 | — | |
RLJWVWNWUMCCKR
|
8.4 | IC50 | 2 | — | |
YXHFWCWUIZMGMT
|
8.4 | IC50 | 2 | — | |
UAFDJFMWWRFFDD
|
8.4 | IC50 | 2 | — | |
ISJIRABUEDACFO
|
8.3 | IC50 | 2 | — | |
VTCHWSGDIXAKIE
|
8.3 | IC50 | 2 | — | |
RIAAGYPMCVIWMN
|
8.3 | IC50 | 2 | — | |
ICQWHVDPJXWVOU
|
8.3 | IC50 | 5 | — | |
MDWOMVXILMHLAO
|
8.3 | IC50 | 5 | — | |
MFZAHAAVYSHLCP
|
8.3 | IC50 | 7 | — | |
PCENXOZMURIZBY
|
8.3 | IC50 | 2 | — | |
SCGCBAAYLFTIJU
|
8.3 | IC50 | 3 | — | |
USVCWSAJUAARAL
|
8.3 | Kd | 8 | — | |
XMBTYCKMMPGSCG
|
8.3 | IC50 | 5 | — | |
ZFQAKLNTCBPIMT
|
8.3 | Ki | 2 | — | |
RPEQRNIMAGWHDH
|
8.3 | IC50 | 2 | — | |
JVVIZDTUQUHDNK
|
8.3 | IC50 | 2 | — | |
LLQPSNXUTNHFGL
|
8.3 | IC50 | 2 | — | |
MFKMYMWETJVOSR
|
8.3 | IC50 | 5 | — | |
JZCTVPONNMDAHV
|
8.3 | IC50 | 2 | — | |
TVMCTGPFPZTNOB
|
8.3 | IC50 | 2 | — | |
RWXSXPWXWPADRF
|
8.2 | IC50 | 2 | — | |
DXPMEKJAAORXIP
|
8.2 | IC50 | 2 | — | |
XRHJGQDNJQEZCK
|
8.2 | IC50 | 2 | — | |
OJVBRFYQEXGWAZ
|
8.2 | IC50 | 5 | — | |
QPYMNQFGNMMOFD
|
8.2 | IC50 | 2 | — | |
WUPAWUQYUGWFGP
|
8.2 | IC50 | 2 | — | |
VCGTXINEJSPRPB
|
8.2 | IC50 | 2 | — | |
FLASJXOUDJHRKI
|
8.2 | IC50 | 2 | — | |
JESNSKPPMWEWAT
|
8.2 | IC50 | 2 | — | |
MKRQUXZNVWJMND
|
8.2 | IC50 | 2 | — | |
GZIKIPGWBKBSLB
|
8.2 | IC50 | 2 | — | |
QWRCTZZUCIJJMB
|
8.2 | IC50 | 2 | — | |
ANNKLDNOHGGDCC
|
8.2 | IC50 | 2 | — | |
KERWPTUPMVZLOH
|
8.2 | IC50 | 2 | — | |
OZOPDYQAHKCSAR
|
8.2 | IC50 | 5 | — | |
URFFOIICYKCKOA
|
8.2 | IC50 | 5 | — | |
YBXRSCXGRPSTMW
|
8.2 | IC50 | 6 | — | |
OQPWFOOQCMOSRA
|
8.1 | IC50 | 2 | — | |
ZITUZZUKNOLFQJ
|
8.1 | IC50 | 2 | — | |
DQMZENNBQZZXEV
|
8.1 | IC50 | 2 | — | |
GRPUEGHDFGOXTK
|
8.1 | IC50 | 2 | — |