Target Details
| UniProt AC | Q13535 |
|---|---|
| Gene Symbol | ATR |
| Protein Name | Serine/threonine-protein kinase ATR |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02259 (FAT) PF02260 (FATC) PF23593 (HEAT_ATR) PF25030 (M-HEAT_ATR) PF25032 (N-HEAT_ATR) PF00454 (PI3_PI4_kinase) PF08064 (UME) |
Summary
- Multi-target molecules 749
- Clinical molecules 0
- Avg pChEMBL 7.26
KEGG Pathways (7)
Associated Diseases (2)
Active Molecules (749)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LYTYLKIUCFTVLF
|
10.0 | IC50 | 2 | — | |
JZCWLJDSIRUGIN
|
9.7 | Ki | 16 | — | |
SSPHMGCXSJLCMP
|
9.7 | IC50 | 2 | — | |
BLHDWFGAYUVFER
|
9.6 | Ki | 2 | — | |
UFZMEAYSFGBIBJ
|
9.5 | IC50 | 4 | — | |
WJVYZVMUDBIEES
|
9.4 | IC50 | 2 | — | |
CHMDAOJBIGUHQC
|
9.3 | IC50 | 5 | — | |
UGAYOLUDSWRLMK
|
9.3 | IC50 | 2 | — | |
ZPRINXXEBIDTGA
|
9.3 | IC50 | 3 | — | |
DBWVYAZESBYVCG
|
9.1 | IC50 | 5 | — | |
IVXMCPRFCSMYPH
|
9.1 | IC50 | 5 | — | |
GEDMPLOWDYEDAT
|
9.0 | IC50 | 5 | — | |
IRPXBHAXMHTWAE
|
9.0 | IC50 | 2 | — | |
PTDUHCKFWWNGET
|
9.0 | Ki | 2 | — | |
RUBCMYKDFDSVRG
|
9.0 | IC50 | 2 | — | |
ZHIDPKVNWVGWNZ
|
9.0 | IC50 | 5 | — | |
HAFHNTJKCXCNQK
|
8.9 | IC50 | 2 | — | |
ILKWBAFOIJQVMU
|
8.8 | IC50 | 2 | — | |
IVXMCPRFCSMYPH
|
8.8 | IC50 | 5 | — | |
IJEDYDGSAXSVPY
|
8.8 | IC50 | 4 | — | |
SITYMNUOQUHVGI
|
8.8 | IC50 | 5 | — | |
USZDDOBUMPPACY
|
8.8 | IC50 | 3 | — | |
BRRNTTQYIGCNKV
|
8.7 | IC50 | 5 | — | |
CFWBGSAWHHCSAE
|
8.7 | IC50 | 5 | — | |
JOSOMFSRJONWIZ
|
8.7 | IC50 | 5 | — | |
KMZIUDOUGCQURL
|
8.7 | IC50 | 5 | — | |
SQYGYXGOJYZQEI
|
8.7 | IC50 | 2 | — | |
TUVIBSPKDKFDLJ
|
8.7 | IC50 | 5 | — | |
XTXRQWYMRAMWQP
|
8.7 | IC50 | 5 | — | |
YFNPMJYHBMGOCT
|
8.7 | IC50 | 5 | — | |
UTWDLQNUMKSECR
|
8.6 | IC50 | 2 | — | |
XKFALBVNCREIJB
|
8.6 | IC50 | 2 | — | |
HNEHJZKGHYOXGG
|
8.6 | IC50 | 5 | — | |
GTBPKBHPMAWGEF
|
8.5 | IC50 | 2 | — | |
HNEHJZKGHYOXGG
|
8.5 | IC50 | 5 | — | |
JSQQOGQSGLHJID
|
8.5 | IC50 | 5 | — | |
JXUKIPQXAFQFDU
|
8.5 | IC50 | 5 | — | |
LDMWKHKGTPOLDV
|
8.5 | IC50 | 5 | — | |
LITSZCPVOFHTLT
|
8.5 | IC50 | 5 | — | |
LKHMVKNMSWRHJH
|
8.5 | IC50 | 7 | — | |
NVZMSEJMRFYPED
|
8.5 | IC50 | 5 | — | |
PJPJLZRSSSFYEH
|
8.5 | IC50 | 5 | — | |
QEWWMCGBQGPTOB
|
8.5 | IC50 | 4 | — | |
QKGSJBBUUWELLN
|
8.5 | IC50 | 5 | — | |
QXPBQXCEIAUDEU
|
8.5 | IC50 | 5 | — | |
WQKHFVMPWAVYDL
|
8.5 | IC50 | 5 | — | |
WVPFDMOAIPTCRI
|
8.5 | IC50 | 5 | — | |
CUUVHIWAYRATBL
|
8.5 | IC50 | 2 | — | |
QXPBQXCEIAUDEU
|
8.5 | IC50 | 5 | — | |
GGGNYZCOIQPDJZ
|
8.4 | IC50 | 2 | — |