Target Details
| UniProt AC | Q13523 |
|---|---|
| Gene Symbol | PRP4K |
| Protein Name | Serine/threonine-protein kinase PRP4 homolog |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 9
- Clinical molecules 5
- Avg pChEMBL 6.86
Active Molecules (9)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XZXHXSATPCNXJR
|
8.1 | Kd | 165 | Yes | |
SKAFXNGFXPGQIG
|
7.8 | IC50 | 3 | — | |
BMGQWWVMWDBQGC
|
7.3 | Kd | 147 | Yes | |
HKSZLNNOFSGOKW
|
6.7 | Kd | 408 | — | |
YYLKKYCXAOBSRM
|
6.6 | Kd | 191 | — | |
JOOXLOJCABQBSG
|
6.4 | Kd | 139 | — | |
WINHZLLDWRZWRT
|
6.4 | Kd | 201 | Yes | |
UIARLYUEJFELEN
|
6.3 | Kd | 289 | Yes | |
PIQCTGMSNWUMAF
|
6.2 | Kd | 137 | Yes |