Target Details
| UniProt AC | Q13490 |
|---|---|
| Gene Symbol | BIRC2 |
| Protein Name | Baculoviral IAP repeat-containing protein 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00653 (BIR) PF00619 (CARD) PF21290 (UBA_BIRC2-3) PF13920 (zf-C3HC4_3) |
Summary
- Multi-target molecules 876
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (16)
- Apoptosis
- Apoptosis - multiple species
- Focal adhesion
- Herpes simplex virus 1 infection
- Hippo signaling pathway
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Necroptosis
- Pathways in cancer
- Platinum drug resistance
- Salmonella infection
- Small cell lung cancer
- TNF signaling pathway
- Toxoplasmosis
- Transcriptional misregulation in cancer
- Ubiquitin mediated proteolysis
Active Molecules (876)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OXPBXFHQSIRUSU
|
8.8 | IC50 | 3 | — | |
RAFMZBCYVHJCOA
|
8.8 | IC50 | 2 | — | |
TYXHMZBEDPKUQY
|
8.8 | IC50 | 2 | — | |
FGDXYJJKIYGYHI
|
8.8 | IC50 | 2 | — | |
KPERLEZLNFSKGP
|
8.8 | IC50 | 2 | — | |
YBYZHVZWINISJO
|
8.8 | Ki | 4 | — | |
GGSBCIHJHQMJEB
|
8.8 | IC50 | 2 | — | |
QCYGMXHLGJJCRO
|
8.8 | Ki | 3 | — | |
SLDGGQPUIMOVMN
|
8.8 | IC50 | 3 | — | |
LPWZUSXPNBYNES
|
8.8 | IC50 | 2 | — | |
TYXHMZBEDPKUQY
|
8.8 | IC50 | 2 | — | |
XQDCNKGNHWZJNL
|
8.8 | IC50 | 2 | — | |
YJQFWHYMLWMKJK
|
8.7 | IC50 | 2 | — | |
BJHUHNWTABFPGG
|
8.7 | IC50 | 2 | — | |
JVVKFFPQWDMFOA
|
8.7 | IC50 | 3 | — | |
KKAHHENNYGUCJF
|
8.7 | IC50 | 2 | — | |
KNODPLACRRUGBI
|
8.7 | IC50 | 2 | — | |
KUALBBKNPXFGDB
|
8.7 | IC50 | 2 | — | |
MGNFGDSTJAIDEC
|
8.7 | IC50 | 2 | — | |
OOIACXVWWQFCNE
|
8.7 | IC50 | 2 | — | |
PWGNJALKXKCHCQ
|
8.7 | IC50 | 2 | — | |
QMYOVGLYSKKPJK
|
8.7 | IC50 | 3 | — | |
VYZMHQWZWYAOIA
|
8.7 | IC50 | 3 | — | |
YBZIUCCRKJMKFE
|
8.7 | IC50 | 2 | — | |
YGGSGHUSONEQIX
|
8.7 | IC50 | 2 | — | |
GIAUJOMDUOPYLU
|
8.7 | IC50 | 3 | — | |
NMLATCDGFYOQGB
|
8.7 | IC50 | 3 | — | |
AQTZITKPGZRNPV
|
8.7 | IC50 | 3 | — | |
GIAUJOMDUOPYLU
|
8.7 | IC50 | 2 | — | |
HLCXKAQSMLQHSZ
|
8.7 | IC50 | 2 | — | |
MVQVBQBVVYPBCQ
|
8.6 | IC50 | 2 | — | |
GUYDSOLIABCZFM
|
8.6 | IC50 | 3 | — | |
ZJOWQMMGXYFDHJ
|
8.6 | IC50 | 2 | — | |
BOOCCBUATVVXCL
|
8.6 | IC50 | 3 | — | |
UGUURTYDXRGYRM
|
8.6 | IC50 | 2 | — | |
VMPRMTGUXGJSDU
|
8.6 | IC50 | 3 | — | |
VMZLJSJMQIJQNE
|
8.6 | IC50 | 2 | — | |
BAODQHPEQZHMBP
|
8.6 | IC50 | 3 | — | |
FIXMENDEDQBFFM
|
8.6 | IC50 | 2 | — | |
OYFPDRMHCIQNHZ
|
8.6 | IC50 | 3 | — | |
XDBOAVJEQWZFNY
|
8.6 | Kd | 2 | — | |
HJBKSCJHQJDSAS
|
8.5 | IC50 | 3 | — | |
MNFHOUJRTFUIQJ
|
8.5 | IC50 | 2 | — | |
PTJLGMSXZVHPLT
|
8.5 | IC50 | 3 | — | |
AVAOWCBMADPQBJ
|
8.5 | IC50 | 3 | — | |
CNHIJRXXUZNFIO
|
8.5 | IC50 | 2 | — | |
DKSXMHRSKSOZAT
|
8.5 | Ki | 3 | — | |
HFZARJHWLBCIML
|
8.5 | IC50 | 3 | — | |
HJDQNNIRKWGQGL
|
8.5 | IC50 | 4 | — | |
LDCYOQDORMHQPW
|
8.5 | IC50 | 3 | — |