Target Details
| UniProt AC | Q13490 |
|---|---|
| Gene Symbol | BIRC2 |
| Protein Name | Baculoviral IAP repeat-containing protein 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00653 (BIR) PF00619 (CARD) PF21290 (UBA_BIRC2-3) PF13920 (zf-C3HC4_3) |
Summary
- Multi-target molecules 876
- Clinical molecules 0
- Avg pChEMBL 7.55
KEGG Pathways (16)
- Apoptosis
- Apoptosis - multiple species
- Focal adhesion
- Herpes simplex virus 1 infection
- Hippo signaling pathway
- NF-kappa B signaling pathway
- NOD-like receptor signaling pathway
- Necroptosis
- Pathways in cancer
- Platinum drug resistance
- Salmonella infection
- Small cell lung cancer
- TNF signaling pathway
- Toxoplasmosis
- Transcriptional misregulation in cancer
- Ubiquitin mediated proteolysis
Active Molecules (876)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MKBRPDBPQLDLIT
|
9.0 | IC50 | 2 | — | |
MPWIGZHHNCNVOO
|
9.0 | IC50 | 2 | — | |
NICRIMMNOCVZDK
|
9.0 | IC50 | 2 | — | |
NJZSVYYBBZWHGJ
|
9.0 | IC50 | 2 | — | |
NSFLHGPXAPXKSS
|
9.0 | IC50 | 3 | — | |
OHXWQHZHQZPUCS
|
9.0 | IC50 | 3 | — | |
OJRHRPFWEXAEQA
|
9.0 | IC50 | 2 | — | |
OOOHUPBTSUEVGE
|
9.0 | IC50 | 2 | — | |
ORQDPDLQZJORFE
|
9.0 | IC50 | 2 | — | |
PGUWLFVOCFDUHZ
|
9.0 | IC50 | 3 | — | |
PUKQEAYHOGMUGF
|
9.0 | IC50 | 3 | — | |
QGGDHYLQLDPUCF
|
9.0 | IC50 | 2 | — | |
ROMCJEPRVBSBEK
|
9.0 | IC50 | 2 | — | |
RVXKLPGEBCDTMK
|
9.0 | IC50 | 2 | — | |
SOZXCUHRCMBRSI
|
9.0 | IC50 | 3 | — | |
VKHIIHCOKPKPJZ
|
9.0 | IC50 | 2 | — | |
VKKPWLVOASHEOF
|
9.0 | IC50 | 2 | — | |
WCEKPSGXNVKDPR
|
9.0 | IC50 | 2 | — | |
WELBXKPSYNELDG
|
9.0 | IC50 | 2 | — | |
XIVQNOQUXQCLEI
|
9.0 | IC50 | 2 | — | |
XPQTUUJPXMXNET
|
9.0 | IC50 | 2 | — | |
YSWMEDPQKFWVOU
|
9.0 | IC50 | 2 | — | |
ZHJDTJNSIZPBCQ
|
9.0 | IC50 | 2 | — | |
BGCVKEKYZIOAGX
|
9.0 | IC50 | 2 | — | |
MBKNBOLIPVRUSC
|
9.0 | IC50 | 3 | — | |
XDBOAVJEQWZFNY
|
9.0 | IC50 | 2 | — | |
YEVVNGCYGSNANK
|
9.0 | IC50 | 2 | — | |
YKDUDNBQXZHFLC
|
9.0 | Ki | 3 | — | |
GVAUTEQHOXIAJI
|
8.9 | Ki | 3 | — | |
KMHMGJITTBRABL
|
8.9 | Ki | 2 | — | |
MNGUBMKVFGTZKL
|
8.9 | Ki | 3 | — | |
MPXBKLQSQUXEDB
|
8.9 | IC50 | 2 | — | |
NOVQMSAXBZDRHD
|
8.9 | IC50 | 3 | — | |
SBCXEQHIGXRICU
|
8.9 | Ki | 3 | — | |
XRNWGSINTQPCAV
|
8.9 | Ki | 3 | — | |
AATYEYGQEXDYIH
|
8.9 | Ki | 3 | — | |
FLOFERYEJWPXFA
|
8.9 | Ki | 3 | — | |
IYOZNYWYRADTNN
|
8.9 | Ki | 4 | — | |
MIWHOUGMEANWCH
|
8.9 | Ki | 3 | — | |
POABUJYLADOSRL
|
8.9 | IC50 | 3 | — | |
QTPJJORUJRBSTP
|
8.9 | IC50 | 3 | — | |
UKNQPDHAXSCGKL
|
8.9 | Ki | 3 | — | |
WQLHYSFOEZZZDD
|
8.9 | Kd | 2 | — | |
XYDGOXJJDFKAAT
|
8.9 | IC50 | 2 | — | |
YSDXUKHVYYZKGA
|
8.9 | Ki | 3 | — | |
UJONUJWQMPOLGZ
|
8.9 | IC50 | 3 | — | |
BOHYEMVPKFXRSG
|
8.8 | IC50 | 3 | — | |
FDGOQDOYZLIFKI
|
8.8 | IC50 | 2 | — | |
GSYCIPSRQKSJPJ
|
8.8 | Ki | 3 | — | |
KSALHYXGSMEPIV
|
8.8 | IC50 | 2 | — |