Target Details
| UniProt AC | Q13470 |
|---|---|
| Gene Symbol | TNK1 |
| Protein Name | Non-receptor tyrosine-protein kinase TNK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF22931 (SAM_TNK) |
Summary
- Multi-target molecules 150
- Clinical molecules 16
- Avg pChEMBL 7.53
Active Molecules (150)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WEKCQPVMVKJTQD
|
7.5 | IC50 | 2 | — | |
AFWLAWBSENRTOI
|
7.4 | IC50 | 2 | — | |
HGJVONCBQFKWRI
|
7.4 | IC50 | 2 | — | |
NPOFZKXRQDDDDY
|
7.4 | IC50 | 2 | — | |
BPWNUTSKZNJOAK
|
7.4 | IC50 | 2 | — | |
PVIVFFQABAVRDM
|
7.4 | IC50 | 2 | — | |
ASUGUQWIHMTFJL
|
7.3 | Kd | 18 | — | |
BRHAGWRGTMVKQA
|
7.3 | IC50 | 2 | — | |
FHQJOMRJKRMAOH
|
7.3 | IC50 | 2 | — | |
XKFTZKGMDDZMJI
|
7.3 | Kd | 64 | Yes | |
FBGYDRBIQYAULP
|
7.3 | IC50 | 2 | — | |
WVXNSAVVKYZVOE
|
7.3 | Kd | 92 | — | |
HPNPGKDJVPSETA
|
7.2 | IC50 | 2 | — | |
LRRAZXKYVVVMLY
|
7.2 | IC50 | 2 | — | |
ODPGGGTTYSGTGO
|
7.2 | Kd | 153 | — | |
BFSMGDJOXZAERB
|
7.2 | Kd | 33 | — | |
BMGQWWVMWDBQGC
|
7.1 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
7.1 | Kd | 91 | Yes | |
GCIKSSRWRFVXBI
|
7.1 | Kd | 109 | Yes | |
PHXJVRSECIGDHY
|
7.1 | Kd | 59 | — | |
KOMGSVVWXUEBNT
|
7.0 | IC50 | 3 | — | |
MLCFDNDRFBGJAZ
|
7.0 | IC50 | 2 | — | |
ZGMGCVMYDSXGAA
|
7.0 | IC50 | 2 | — | |
RRTBNWLSPAIIKM
|
6.9 | IC50 | 2 | — | |
LQVXSNNAFNGRAH
|
6.8 | Kd | 33 | Yes | |
GKDRMWXFWHEQQT
|
6.8 | Kd | 7 | — | |
RITAVMQDGBJQJZ
|
6.8 | Kd | 43 | — | |
UEVFMGJBRLJVKO
|
6.8 | IC50 | 3 | — | |
XZXHXSATPCNXJR
|
6.7 | Kd | 165 | Yes | |
HUFOZJXAKZVRNJ
|
6.5 | Kd | 10 | — | |
KOZFSFOOLUUIGY
|
6.5 | Kd | 88 | Yes | |
KTEIFNKAUNYNJU
|
6.5 | Kd | 114 | — | |
JOOXLOJCABQBSG
|
6.4 | Kd | 139 | — | |
VAARYSWULJUGST
|
6.4 | Kd | 119 | Yes | |
RYYNGWLOYLRZLK
|
6.4 | Kd | 45 | — | |
QTBWCSQGBMPECM
|
6.3 | Kd | 21 | Yes | |
WKDACQVEJIVHMZ
|
6.2 | Kd | 46 | — | |
YYLKKYCXAOBSRM
|
6.2 | Kd | 191 | — | |
ZZSBPGIGIUFJRA
|
6.2 | Kd | 46 | — | |
XUZMWHLSFXCVMG
|
6.2 | Kd | 24 | — | |
AAKJLRGGTJKAMG
|
6.2 | Kd | 50 | Yes | |
UJLAWZDWDVHWOW
|
6.2 | Kd | 16 | — | |
WINHZLLDWRZWRT
|
6.2 | Kd | 201 | Yes | |
ZBNZXTGUTAYRHI
|
6.2 | Kd | 102 | Yes | |
HWXVIOGONBBTBY
|
6.0 | Kd | 27 | — | |
CUIHSIWYWATEQL
|
6.0 | Kd | 61 | Yes | |
KDKUVYLMPJIGKA
|
6.0 | Kd | 91 | Yes | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — |