Target Details
| UniProt AC | Q13470 |
|---|---|
| Gene Symbol | TNK1 |
| Protein Name | Non-receptor tyrosine-protein kinase TNK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF22931 (SAM_TNK) |
Summary
- Multi-target molecules 150
- Clinical molecules 16
- Avg pChEMBL 7.53
Active Molecules (150)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CDELRUCHGDJWNM
|
7.9 | IC50 | 3 | — | |
VAOQBNBDBKHNQY
|
7.9 | IC50 | 3 | — | |
DBTLGWQFPVIXTJ
|
7.8 | IC50 | 2 | — | |
INRRUWSEBDJLPW
|
7.8 | IC50 | 3 | — | |
MFPOWTKEAYCCGQ
|
7.8 | IC50 | 2 | — | |
OOMBFNDWQIGHEK
|
7.8 | Kd | 22 | — | |
ORSBXGBOZDSEJT
|
7.8 | IC50 | 3 | — | |
AURCLDMUVVKGCY
|
7.8 | IC50 | 3 | — | |
FBIGNDFZRCUSDQ
|
7.8 | IC50 | 3 | — | |
SMSCYHHVBZIUMV
|
7.8 | IC50 | 2 | — | |
CEGOEVTXZXXUSN
|
7.8 | IC50 | 2 | — | |
JKCHNICKXRIXAL
|
7.8 | IC50 | 2 | — | |
NZDMYHLPDHCLGC
|
7.8 | IC50 | 3 | — | |
TWZQEBQCXWLACN
|
7.8 | IC50 | 3 | — | |
IZKKJBVPFFOLOL
|
7.8 | IC50 | 2 | — | |
WEFPHDYTHUNVAM
|
7.8 | IC50 | 3 | — | |
DPKCTDXZHPAPLS
|
7.8 | IC50 | 3 | — | |
FSFKDNPHPFINJD
|
7.8 | IC50 | 3 | — | |
SCONNUWWGIRXAF
|
7.8 | IC50 | 2 | — | |
WPTNASIDXWQCDG
|
7.7 | IC50 | 3 | — | |
SOASXIFPFLUWRH
|
7.7 | IC50 | 2 | — | |
WOBDQRLNYWLLJQ
|
7.7 | IC50 | 2 | — | |
SVYQAPDHJLXDGC
|
7.7 | IC50 | 3 | — | |
CXQHYVUVSFXTMY
|
7.7 | Kd | 154 | — | |
SEJGTFPOEJWEGG
|
7.7 | Kd | 149 | — | |
LZKGLICEGUTSDW
|
7.7 | IC50 | 3 | — | |
XGFMLKJENFANEN
|
7.6 | IC50 | 2 | — | |
SLEWGGZPOQNVSU
|
7.6 | Kd | 22 | — | |
MWLJLVHPVHBVDL
|
7.6 | IC50 | 2 | — | |
NHHQJBCNYHBUSI
|
7.6 | Kd | 220 | — | |
OXULFDKDMPHAFP
|
7.6 | IC50 | 3 | — | |
GBEWXEQDDXPZJQ
|
7.6 | IC50 | 2 | — | |
AXAVOVXYAFPCSL
|
7.6 | IC50 | 2 | — | |
IWIRGSJMTCVGQQ
|
7.6 | IC50 | 2 | — | |
VERWOWGGCGHDQE
|
7.6 | Kd | 23 | — | |
FADNVFGOLBDUSB
|
7.6 | IC50 | 2 | — | |
MWKSRKSEWLRPBL
|
7.6 | Kd | 1075 | — | |
DDTPGANIPBKTNU
|
7.5 | Kd | 8 | — | |
GXXRJPKTTBCLNF
|
7.5 | IC50 | 2 | — | |
QBLCDAXXROYNNC
|
7.5 | IC50 | 2 | — | |
MGGBYMDAPCCKCT
|
7.5 | IC50 | 23 | — | |
UCQAPUVIUAYEGE
|
7.5 | IC50 | 3 | — | |
AMWNTQXPBJQZET
|
7.5 | IC50 | 3 | — | |
DILZMEVBCHRKIZ
|
7.5 | IC50 | 3 | — | |
GXLCEYYXBWDRJO
|
7.5 | IC50 | 3 | — | |
KHGMRXFPRSSDPX
|
7.5 | IC50 | 2 | — | |
GYUCFGYTWSIWKA
|
7.5 | IC50 | 2 | — | |
ZMRSDMLCFJDLKR
|
7.5 | IC50 | 3 | — | |
IRVJFMHHDJQNGA
|
7.5 | IC50 | 2 | — | |
SJYGJUQORXZRIJ
|
7.5 | IC50 | 3 | — |