Target Details
| UniProt AC | Q13470 |
|---|---|
| Gene Symbol | TNK1 |
| Protein Name | Non-receptor tyrosine-protein kinase TNK1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) PF22931 (SAM_TNK) |
Summary
- Multi-target molecules 150
- Clinical molecules 16
- Avg pChEMBL 7.53
Active Molecules (150)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QQWUGDVOUVUTOY
|
8.7 | Kd | 231 | Yes | |
HKSZLNNOFSGOKW
|
8.7 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
8.6 | Kd | 213 | — | |
XUFWBGKENCGHSD
|
8.6 | IC50 | 3 | — | |
ALKJNCZNEOTEMP
|
8.5 | Kd | 55 | — | |
JQJGYBASPJXNIJ
|
8.5 | IC50 | 3 | — | |
RSZFCUWJGDNCGK
|
8.5 | IC50 | 3 | — | |
DRPXVULWOOOZDV
|
8.4 | IC50 | 3 | — | |
RLKUZCOFKFUEHH
|
8.4 | IC50 | 3 | — | |
NXSJMRCTGYTSTK
|
8.4 | Kd | 200 | — | |
PZYRHYWULWFGBG
|
8.4 | IC50 | 3 | — | |
UWIOUEAALWYOMW
|
8.4 | IC50 | 3 | — | |
ONEIDYKHPRMDQO
|
8.4 | IC50 | 3 | — | |
CINNRILLZCDNOZ
|
8.3 | IC50 | 3 | — | |
OCLDJPYPPFDDNO
|
8.3 | IC50 | 3 | — | |
GRPXLKXGJAGYSD
|
8.3 | IC50 | 3 | — | |
DBLBOZLZPCJKAH
|
8.2 | IC50 | 3 | — | |
WQVZBZQCVBIXLT
|
8.2 | IC50 | 3 | — | |
IXNZYKNOAINDTN
|
8.2 | IC50 | 3 | — | |
QAJSMIVRRQDYBG
|
8.2 | IC50 | 3 | — | |
LCVIRAZGMYMNNT
|
8.2 | Kd | 20 | — | |
CBRIZHZYFLCPAP
|
8.2 | IC50 | 3 | — | |
OUERNEXEYTUWRZ
|
8.2 | IC50 | 3 | — | |
OTDIMNJLKVGGOB
|
8.1 | IC50 | 3 | — | |
RAPGQTWOPCNSEJ
|
8.1 | IC50 | 3 | — | |
FWZKUFCCKVNCSL
|
8.1 | IC50 | 2 | — | |
QWQRHMZFZSWUOD
|
8.1 | IC50 | 3 | — | |
UIARLYUEJFELEN
|
8.0 | Kd | 289 | Yes | |
CVLCVUYBIPUQBG
|
8.0 | IC50 | 3 | — | |
DVBFHLPDOMIKKR
|
8.0 | IC50 | 3 | — | |
CVTFVYCHNGODLR
|
8.0 | IC50 | 3 | — | |
CCWTWPIDXUGAKX
|
8.0 | IC50 | 3 | — | |
PITKHMJQSBHPED
|
8.0 | IC50 | 3 | — | |
SOASXIFPFLUWRH
|
8.0 | IC50 | 3 | — | |
VOQLJAINULFPEC
|
8.0 | IC50 | 2 | — | |
WPSFTNDXYZENJA
|
8.0 | IC50 | 3 | — | |
UOAHTPZUUUBPBK
|
8.0 | IC50 | 3 | — | |
XFINPBQKFDIRJH
|
8.0 | IC50 | 3 | — | |
MWLJLVHPVHBVDL
|
7.9 | IC50 | 3 | — | |
NRDDMPIVXPOIMZ
|
7.9 | IC50 | 2 | — | |
RZVRCAKYGAURIU
|
7.9 | IC50 | 2 | — | |
XULZRMKGTVQSFV
|
7.9 | IC50 | 2 | — | |
QSDUGBPLSHIMHQ
|
7.9 | IC50 | 3 | — | |
FJOFREJOLJFMNF
|
7.9 | IC50 | 3 | — | |
OLJYGSVADWZNIQ
|
7.9 | IC50 | 2 | — | |
NJQTWWNECKEAQJ
|
7.9 | IC50 | 3 | — | |
SOASXIFPFLUWRH
|
7.9 | IC50 | 2 | — | |
ICWAHMDHBIKSJI
|
7.9 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
7.9 | Kd | 170 | — | |
MGFDCSFBWGIIJD
|
7.9 | IC50 | 2 | — |