Target Details
| UniProt AC | Q13464 |
|---|---|
| Gene Symbol | ROCK1 |
| Protein Name | Rho-associated protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF25346 (PH_MRCK) PF00069 (Pkinase) PF08912 (Rho_Binding) |
Summary
- Multi-target molecules 1,614
- Clinical molecules 34
- Avg pChEMBL 7.13
KEGG Pathways (22)
- Adherens junction
- Axon guidance
- Cadherin signaling
- Chemokine signaling pathway
- Focal adhesion
- Human cytomegalovirus infection
- Leukocyte transendothelial migration
- MicroRNAs in cancer
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Platelet activation
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Sphingolipid signaling pathway
- TGF-beta signaling pathway
- Tight junction
- Vascular smooth muscle contraction
- Yersinia infection
- cAMP signaling pathway
- cGMP-PKG signaling pathway
Active Molecules (1,614)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MZBLKPUSLVWLBU
|
7.8 | IC50 | 2 | — | |
NMVQKQZIFRBWNR
|
7.8 | IC50 | 2 | — | |
WWFOLVBRNURGPW
|
7.8 | IC50 | 6 | — | |
XCUCJAJWXMJKLB
|
7.8 | IC50 | 2 | — | |
ZTFIBKWDXXXKRW
|
7.8 | IC50 | 2 | — | |
WPWSPITXILOZGO
|
7.8 | IC50 | 2 | — | |
ZTHAJPGZRABKDJ
|
7.8 | IC50 | 6 | — | |
CGXOKVWAHQLXGW
|
7.8 | IC50 | 2 | — | |
CLEGDJQQHUTCOW
|
7.8 | Ki | 43 | — | |
HWOQGLLRJCPMIZ
|
7.8 | IC50 | 2 | — | |
IFSJHRROANUFFS
|
7.8 | IC50 | 2 | — | |
JEZPZXAMLGEGDI
|
7.8 | IC50 | 2 | — | |
RFVBRKXQYUDGIO
|
7.8 | Ki | 23 | — | |
TVEREFRWBLRPPJ
|
7.8 | Ki | 15 | — | |
UCJIXVPTONWDEH
|
7.8 | IC50 | 3 | — | |
UHTJASDMENLSNM
|
7.8 | IC50 | 2 | — | |
ZCFDZMIXMIEOHC
|
7.8 | IC50 | 6 | — | |
ZDIVXJMVURCVPS
|
7.8 | IC50 | 2 | — | |
ZNDQOACBIHODQO
|
7.8 | IC50 | 3 | — | |
BLMKBLDBMAAGCC
|
7.8 | Ki | 3 | — | |
GLYMNXIYEPWMQN
|
7.8 | IC50 | 2 | — | |
HOKFQGROLDNJSI
|
7.8 | IC50 | 2 | — | |
KKFYJBLOJFXLCI
|
7.8 | IC50 | 2 | — | |
KSEWBEGMKXXEAT
|
7.8 | IC50 | 2 | — | |
LFBDSSPYPYYACO
|
7.8 | Ki | 2 | — | |
ABPSPQITFLVJSN
|
7.8 | IC50 | 2 | — | |
BIHSMCRXOPRSSF
|
7.8 | Ki | 2 | — | |
BSULSXCQOXQGND
|
7.8 | IC50 | 2 | — | |
CWKUJWGURSJFTK
|
7.8 | IC50 | 2 | — | |
GWBRWSIUAMTBNQ
|
7.8 | IC50 | 2 | — | |
JBAFISIOKGNSRP
|
7.8 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
7.8 | IC50 | 82 | — | |
MFBHZMTZVKYMTG
|
7.8 | IC50 | 2 | — | |
RBSPMMLWEZLNPN
|
7.8 | IC50 | 2 | — | |
HUXNQLSQBYWWAS
|
7.8 | IC50 | 2 | — | |
LXQGBVWOYPFPJU
|
7.8 | IC50 | 2 | — | |
PLIFSXNZAOLLSV
|
7.8 | IC50 | 2 | — | |
CICZGTVNSVVRFC
|
7.7 | IC50 | 2 | — | |
CVJDWPOZUNTTIU
|
7.7 | IC50 | 2 | — | |
GZVUGIYFFYQNCJ
|
7.7 | Ki | 4 | — | |
JSBFPPNKJVBJKX
|
7.7 | IC50 | 2 | — | |
LGAOSGWGEUZJCW
|
7.7 | IC50 | 6 | — | |
PBRPSSPCDCQDDX
|
7.7 | IC50 | 2 | — | |
PUDPIQFNZNNYGT
|
7.7 | IC50 | 3 | — | |
RSSVYLIGOHSPNV
|
7.7 | IC50 | 2 | — | |
SLODBPIAZZPOFN
|
7.7 | IC50 | 7 | — | |
ZTXPZKBYVPEULR
|
7.7 | Ki | 3 | — | |
BMMXFLCCJJRAMC
|
7.7 | Ki | 4 | — | |
KXPTUMLQPMMHGT
|
7.7 | IC50 | 4 | — | |
YAGRGEPEYURZTE
|
7.7 | IC50 | 2 | — |