Target Details
| UniProt AC | Q13464 |
|---|---|
| Gene Symbol | ROCK1 |
| Protein Name | Rho-associated protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF25346 (PH_MRCK) PF00069 (Pkinase) PF08912 (Rho_Binding) |
Summary
- Multi-target molecules 1,614
- Clinical molecules 34
- Avg pChEMBL 7.13
KEGG Pathways (22)
- Adherens junction
- Axon guidance
- Cadherin signaling
- Chemokine signaling pathway
- Focal adhesion
- Human cytomegalovirus infection
- Leukocyte transendothelial migration
- MicroRNAs in cancer
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Platelet activation
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Sphingolipid signaling pathway
- TGF-beta signaling pathway
- Tight junction
- Vascular smooth muscle contraction
- Yersinia infection
- cAMP signaling pathway
- cGMP-PKG signaling pathway
Active Molecules (1,614)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JAWPAUHQCGKVGI
|
8.2 | IC50 | 2 | — | |
KACIGJBSABVNRF
|
8.2 | IC50 | 2 | — | |
KWQRIWDMNAKJAF
|
8.2 | Ki | 3 | — | |
KZYAHEIPPAPADQ
|
8.2 | IC50 | 3 | — | |
MQHAUPTVCAFIJM
|
8.2 | IC50 | 2 | — | |
NGOKTEXAUPRBFP
|
8.2 | IC50 | 2 | — | |
QPDAFPVNIOVXCG
|
8.2 | IC50 | 2 | — | |
YYQWLNWVYQGLHK
|
8.2 | IC50 | 2 | — | |
GHPFQRTVUDXWCC
|
8.2 | Ki | 35 | — | |
MLGGUGPIWDHBAI
|
8.2 | IC50 | 10 | — | |
PUYIXDDMOUMMRR
|
8.2 | Ki | 27 | — | |
XZVLUQDUOAWQMB
|
8.2 | Ki | 4 | — | |
BWJHMGCCCMRFBU
|
8.2 | IC50 | 2 | — | |
CYJWEDGBZCTVAV
|
8.2 | IC50 | 2 | — | |
KQDDDWVLLDDHOF
|
8.2 | IC50 | 2 | — | |
MURRHZDIBOUBHB
|
8.2 | IC50 | 7 | — | |
PDWFMHXAWIQAEE
|
8.2 | IC50 | 2 | — | |
QFHANDBITKFWTC
|
8.2 | IC50 | 7 | — | |
GCKIJVYMPZVOFI
|
8.2 | IC50 | 2 | — | |
IKBDBMJIRDOTCY
|
8.2 | IC50 | 2 | — | |
OEYSQZKVMVAGLO
|
8.2 | IC50 | 2 | — | |
RBUCEYWKPHIQNJ
|
8.2 | IC50 | 2 | — | |
DUUFTCDTPYSKCS
|
8.2 | IC50 | 2 | — | |
ICQSNTDFCNRKLY
|
8.2 | IC50 | 2 | — | |
IZBXLPNFYAKSMH
|
8.2 | Ki | 2 | — | |
PXLAOJRRWUJJHK
|
8.2 | IC50 | 2 | — | |
RVYJKUWZLONOCK
|
8.2 | IC50 | 2 | — | |
YKJXZODWOQJHCQ
|
8.2 | IC50 | 2 | — | |
HSCQYWDDHGGJSS
|
8.1 | IC50 | 2 | — | |
JBXUKWIGBDQLCO
|
8.1 | IC50 | 7 | — | |
ONZAMBWLADUDER
|
8.1 | IC50 | 2 | — | |
DWWGQXYDCWJWKM
|
8.1 | IC50 | 2 | — | |
NUSTUPPCTIUXFR
|
8.1 | IC50 | 2 | — | |
YCNNWSRSIAKLGS
|
8.1 | IC50 | 2 | — | |
BGMFLWUQWMTTSW
|
8.1 | IC50 | 8 | — | |
DFXUOVUWCCNNPV
|
8.1 | IC50 | 2 | — | |
FPNYVINXEGJSCQ
|
8.1 | IC50 | 2 | — | |
PHRUWSDSXOMMTK
|
8.1 | IC50 | 2 | — | |
BGZVXNSBCSLMND
|
8.1 | IC50 | 5 | — | |
BSULSXCQOXQGND
|
8.1 | IC50 | 2 | — | |
FCDBVNCRKMBDIO
|
8.1 | IC50 | 2 | — | |
FUMCKNCUEAQHCV
|
8.1 | Ki | 103 | — | |
GVOJSDSHNFLVIW
|
8.1 | IC50 | 2 | — | |
OYNBTBJATZVIGH
|
8.1 | IC50 | 3 | — | |
RHTXWIKPNGROHZ
|
8.1 | IC50 | 3 | — | |
UMTWTCVTRDYHQQ
|
8.1 | Ki | 56 | — | |
UYQVTFFVWVLMAA
|
8.1 | IC50 | 2 | — | |
VGNKOJURPOHWJF
|
8.1 | Ki | 21 | — | |
XSRHBCYNCKAFKS
|
8.1 | Ki | 45 | — | |
YFZKQJYONASWFW
|
8.1 | IC50 | 7 | — |