Target Details
| UniProt AC | Q13464 |
|---|---|
| Gene Symbol | ROCK1 |
| Protein Name | Rho-associated protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF25346 (PH_MRCK) PF00069 (Pkinase) PF08912 (Rho_Binding) |
Summary
- Multi-target molecules 1,614
- Clinical molecules 34
- Avg pChEMBL 7.13
KEGG Pathways (22)
- Adherens junction
- Axon guidance
- Cadherin signaling
- Chemokine signaling pathway
- Focal adhesion
- Human cytomegalovirus infection
- Leukocyte transendothelial migration
- MicroRNAs in cancer
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Platelet activation
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Sphingolipid signaling pathway
- TGF-beta signaling pathway
- Tight junction
- Vascular smooth muscle contraction
- Yersinia infection
- cAMP signaling pathway
- cGMP-PKG signaling pathway
Active Molecules (1,614)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZANIGAVBLOXUNT
|
7.3 | IC50 | 2 | — | |
ZZRYLKQMDUISGY
|
7.3 | IC50 | 2 | — | |
GUIBMJRAVIMUQK
|
7.3 | IC50 | 2 | — | |
OQDKYJBFAREBIO
|
7.3 | IC50 | 2 | — | |
CELVWXWADDJEMH
|
7.3 | IC50 | 3 | — | |
JPIZMTCZKMZLDC
|
7.3 | IC50 | 2 | — | |
LFPUNHMXMCZMLZ
|
7.3 | IC50 | 3 | — | |
LKVWXTDYMZEGFK
|
7.3 | IC50 | 2 | — | |
ONZAMBWLADUDER
|
7.3 | IC50 | 2 | — | |
VTSLKIKDRBEGHX
|
7.3 | Ki | 3 | — | |
XEXJRQIFMJLDKP
|
7.3 | IC50 | 2 | — | |
AWBKTMLYSSBTLA
|
7.3 | IC50 | 2 | — | |
OTRYRVUEBNQHDC
|
7.3 | IC50 | 2 | — | |
PPJJUYYHDQPMBM
|
7.3 | IC50 | 2 | — | |
BXVVJBRCXPFGAH
|
7.3 | IC50 | 2 | — | |
HNXJWWRRSGDVIW
|
7.3 | Ki | 13 | — | |
NKEUPUJTVALZIK
|
7.3 | Ki | 28 | — | |
PQGVJYYWZHMBEY
|
7.3 | IC50 | 2 | — | |
QBWKZDBFMHLSHV
|
7.3 | IC50 | 2 | — | |
QEWSTOOMTBAUAG
|
7.3 | Ki | 17 | — | |
RQJNDHYSIAYHOI
|
7.3 | IC50 | 2 | — | |
SODGZPDNROVASD
|
7.3 | Ki | 7 | — | |
VGSYMGCEDYSPMI
|
7.3 | IC50 | 2 | — | |
ZSRGQQNNHDFZKU
|
7.3 | IC50 | 2 | — | |
ZYTFPHRVOZXPGZ
|
7.3 | Ki | 30 | — | |
JQXGSDPBFXEDBN
|
7.3 | IC50 | 4 | — | |
LVAMWHFZQXITMS
|
7.3 | IC50 | 2 | — | |
QSKQVZWVLOIIEV
|
7.3 | IC50 | 4 | — | |
RVLBWZZSHLQKAN
|
7.3 | IC50 | 2 | — | |
KRPHFYXXDKDNKY
|
7.3 | IC50 | 3 | — | |
LYLJYIZTSPUCNP
|
7.3 | IC50 | 2 | — | |
NENOOZASAODLIG
|
7.3 | IC50 | 2 | — | |
PCKDJQQSQGGVGF
|
7.3 | IC50 | 3 | — | |
SYAFKJOXGPOOAP
|
7.3 | IC50 | 2 | — | |
UIWCYNRIHYQWRJ
|
7.3 | IC50 | 2 | — | |
ISRFXEQOQGZVMK
|
7.3 | IC50 | 2 | — | |
JILSPXHZRNLZHV
|
7.3 | IC50 | 2 | — | |
QQUHYDVWIHRQBS
|
7.3 | IC50 | 5 | — | |
UTXFYQOYXIBPAU
|
7.3 | IC50 | 2 | — | |
XVWAHNBWATXACB
|
7.3 | IC50 | 2 | — | |
BPNUQXPIQBZCMR
|
7.3 | IC50 | 83 | Yes | |
DYGYVRRCXQMZJC
|
7.3 | IC50 | 2 | — | |
KMIKGPNXOFBRHM
|
7.3 | IC50 | 2 | — | |
NHCZWHGCNNIQHP
|
7.3 | IC50 | 2 | — | |
PCGOLHRVCCFRNK
|
7.3 | IC50 | 2 | — | |
RJMZRJDWOXEUNY
|
7.3 | IC50 | 2 | — | |
WFKLCCZTEPHYPI
|
7.3 | IC50 | 2 | — | |
WNFAWYDESPZZIJ
|
7.3 | IC50 | 2 | — | |
ZFBYIIFQXUFBCC
|
7.3 | IC50 | 2 | — | |
DZSWYUCCPNQWOQ
|
7.2 | Ki | 4 | — |