Target Details
| UniProt AC | Q13464 |
|---|---|
| Gene Symbol | ROCK1 |
| Protein Name | Rho-associated protein kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF25346 (PH_MRCK) PF00069 (Pkinase) PF08912 (Rho_Binding) |
Summary
- Multi-target molecules 1,614
- Clinical molecules 34
- Avg pChEMBL 7.13
KEGG Pathways (22)
- Adherens junction
- Axon guidance
- Cadherin signaling
- Chemokine signaling pathway
- Focal adhesion
- Human cytomegalovirus infection
- Leukocyte transendothelial migration
- MicroRNAs in cancer
- Oxytocin signaling pathway
- Pathogenic Escherichia coli infection
- Pathways in cancer
- Platelet activation
- Proteoglycans in cancer
- Regulation of actin cytoskeleton
- Shigellosis
- Sphingolipid signaling pathway
- TGF-beta signaling pathway
- Tight junction
- Vascular smooth muscle contraction
- Yersinia infection
- cAMP signaling pathway
- cGMP-PKG signaling pathway
Active Molecules (1,614)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NSQJYQIGGJGUKK
|
7.6 | IC50 | 2 | — | |
OSVUGUHRKMMBSE
|
7.6 | Kd | 170 | — | |
SOEYUSIWHOBEMJ
|
7.6 | IC50 | 2 | — | |
URYCVJWDQPAEFD
|
7.6 | IC50 | 2 | — | |
AEVCWYWUPQHFFI
|
7.6 | IC50 | 2 | — | |
BDCUKYUIVYKXCQ
|
7.6 | IC50 | 2 | — | |
IFYDROJSRZHNOS
|
7.6 | IC50 | 7 | — | |
IIRWNGPLJQXWFJ
|
7.6 | Kd | 21 | — | |
SIYJLMVIVBKINW
|
7.6 | IC50 | 2 | — | |
DYMMJEIVULXUAB
|
7.5 | IC50 | 2 | — | |
FFJWOJIKTPHFRY
|
7.5 | IC50 | 2 | — | |
GWHBGZBCJKQNCZ
|
7.5 | IC50 | 4 | — | |
VKORCHLUUJGKEE
|
7.5 | Ki | 3 | — | |
WSXKSMSBOLIXMK
|
7.5 | IC50 | 2 | — | |
JIKVGTFJHKLPJM
|
7.5 | IC50 | 2 | — | |
JTVBXQAYBIJXRP
|
7.5 | IC50 | 20 | — | |
NZTPJNIILSLMRH
|
7.5 | IC50 | 7 | — | |
PATAJJRKSXHPFR
|
7.5 | IC50 | 2 | — | |
SCCMLQDEEDXQCZ
|
7.5 | Ki | 3 | — | |
ZNGHRZYYUDIWDX
|
7.5 | IC50 | 2 | — | |
CWFBWCJRVBRKPQ
|
7.5 | Ki | 2 | — | |
DWTNLZZEPSCAIH
|
7.5 | IC50 | 2 | — | |
GMKAERKZQVDXFL
|
7.5 | IC50 | 2 | — | |
MHOIPADYLYCBEO
|
7.5 | IC50 | 2 | — | |
OBRQLJITIRIMLQ
|
7.5 | IC50 | 11 | — | |
OPSKOBJDDUDMAW
|
7.5 | IC50 | 2 | — | |
OQORIVHBMBWOAH
|
7.5 | IC50 | 2 | — | |
PZUHTMLHMMXBQW
|
7.5 | IC50 | 2 | — | |
SWQDUVOIJJCWIG
|
7.5 | Ki | 4 | — | |
VUKPYAYVXNDTIK
|
7.5 | IC50 | 2 | — | |
ZPQGWIWZWZNROO
|
7.5 | IC50 | 6 | — | |
NVVLAIWWHAUHCF
|
7.5 | Ki | 4 | — | |
OATPNKANSMGAAO
|
7.5 | IC50 | 2 | — | |
PNMGTDVFGLZVQH
|
7.5 | IC50 | 3 | — | |
UTPDQPQSXIPZQG
|
7.5 | IC50 | 2 | — | |
BSFNGHCTZDCQBF
|
7.5 | Ki | 93 | — | |
DPAPGNJIIHRZFH
|
7.5 | IC50 | 2 | — | |
LUPCHAFIKZSOOK
|
7.5 | Ki | 15 | — | |
LWBSSNRDDDFHSH
|
7.5 | Ki | 9 | — | |
OUJZYQBEFNDJQN
|
7.5 | Ki | 71 | — | |
PTOPXBFSXASLNA
|
7.5 | IC50 | 6 | — | |
SHENEEFOURUIBP
|
7.5 | Ki | 29 | — | |
VVEGARMQKNYDID
|
7.5 | Ki | 24 | — | |
XNWKXXIGSPPPBH
|
7.5 | Ki | 31 | — | |
XNOBXYSDKGIVFG
|
7.5 | IC50 | 2 | — | |
AMBHUZIJUSXSQJ
|
7.5 | IC50 | 2 | — | |
BKCNFBWOOAHROL
|
7.5 | IC50 | 3 | — | |
BPKLWGGNPZJROD
|
7.5 | IC50 | 2 | — | |
DFEBLGYTZYBLCJ
|
7.5 | IC50 | 2 | — | |
JHZPLXPNLZAPIG
|
7.5 | IC50 | 3 | — |