Target Details
| UniProt AC | Q13443 |
|---|---|
| Gene Symbol | ADAM9 |
| Protein Name | Disintegrin and metalloproteinase domain-containing protein 9 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF08516 (ADAM_CR) PF00200 (Disintegrin) PF01562 (Pep_M12B_propep) PF01421 (Reprolysin) |
Summary
- Multi-target molecules 25
- Clinical molecules 20
- Avg pChEMBL 6.59
KEGG Pathways (1)
Associated Diseases (1)
Active Molecules (25)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NITYDPDXAAFEIT
|
8.1 | IC50 | 20 | Yes | |
FAXGPCHRFPCXOO
|
7.2 | IC50 | 14 | — | |
RTKNMWBYPISZDZ
|
7.2 | IC50 | 7 | Yes | |
SQYRXZTYDRVAMZ
|
7.2 | IC50 | 5 | Yes | |
MAVDNGWEBZTACC
|
7.1 | IC50 | 9 | Yes | |
MAVDNGWEBZTACC
|
7.1 | IC50 | 6 | — | |
BQDVTMRZPWSYOT
|
7.0 | IC50 | 7 | — | |
TZNUGSCRBFBAFR
|
6.7 | IC50 | 7 | Yes | |
DPQCHTZYBRQXQC
|
6.7 | IC50 | 7 | Yes | |
RBLCSCFFNCADJO
|
6.6 | IC50 | 7 | Yes | |
QSFJZGINKPYVRC
|
6.6 | IC50 | 7 | Yes | |
NQYWUYPYYFALAI
|
6.5 | IC50 | 6 | Yes | |
MXGYLPKHTGTZKG
|
6.4 | IC50 | 7 | Yes | |
LXKHXLQQHKRMFP
|
6.4 | IC50 | 7 | Yes | |
LZUHYMGQNXWOHQ
|
6.3 | IC50 | 6 | — | |
GMNFREWQYNXZAF
|
6.3 | IC50 | 7 | Yes | |
CDUNTBSHRUTDFM
|
6.3 | IC50 | 7 | Yes | |
JFMSSTVXWKCAJH
|
6.2 | IC50 | 7 | Yes | |
IBUXWZOBVVWCHD
|
6.2 | IC50 | 7 | Yes | |
XRIFBRFEZLXEFP
|
6.2 | IC50 | 5 | — | |
DWFUVVZGNJNHKO
|
6.2 | IC50 | 7 | Yes | |
LICJLIVFDQFASY
|
6.1 | IC50 | 6 | Yes | |
KADFIIKJGHEHDF
|
6.1 | IC50 | 7 | Yes | |
HFCXLBPJFPHTAN
|
6.0 | IC50 | 7 | Yes | |
IAZFWEJODMHVIO
|
6.0 | IC50 | 7 | Yes |