Target Details
| UniProt AC | Q13393 |
|---|---|
| Gene Symbol | PLD1 |
| Protein Name | Phospholipase D1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00169 (PH) PF00614 (PLDc) PF13091 (PLDc_2) PF00787 (PX) |
Summary
- Multi-target molecules 309
- Clinical molecules 1
- Avg pChEMBL 7.29
KEGG Pathways (16)
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Endocytosis
- Ether lipid metabolism
- Fc gamma R-mediated phagocytosis
- Glutamatergic synapse
- Glycerophospholipid metabolism
- GnRH signaling pathway
- Metabolic pathways
- Pancreatic cancer
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Phospholipase D signaling pathway
- Ras signaling pathway
- Sphingolipid signaling pathway
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NUXXESNUMKLEHZ
|
6.1 | IC50 | 2 | — | |
LMGGKAGUODAECN
|
6.1 | IC50 | 2 | — | |
XTLUPAALUSVNDV
|
6.1 | IC50 | 2 | — | |
HQYFYGHOHBPKMU
|
6.1 | IC50 | 2 | — | |
MVKMHBXENCIAGV
|
6.1 | IC50 | 2 | — | |
WBQNNMYOSBMSBZ
|
6.1 | IC50 | 2 | — | |
NUJRIFUQIQAKOJ
|
6.0 | IC50 | 2 | — | |
XWZHLCVDFJHMTB
|
6.0 | IC50 | 2 | — | |
FAIFAFUXFFWVNQ
|
6.0 | IC50 | 2 | — |