Target Details
| UniProt AC | Q13393 |
|---|---|
| Gene Symbol | PLD1 |
| Protein Name | Phospholipase D1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00169 (PH) PF00614 (PLDc) PF13091 (PLDc_2) PF00787 (PX) |
Summary
- Multi-target molecules 309
- Clinical molecules 1
- Avg pChEMBL 7.29
KEGG Pathways (16)
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Endocytosis
- Ether lipid metabolism
- Fc gamma R-mediated phagocytosis
- Glutamatergic synapse
- Glycerophospholipid metabolism
- GnRH signaling pathway
- Metabolic pathways
- Pancreatic cancer
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Phospholipase D signaling pathway
- Ras signaling pathway
- Sphingolipid signaling pathway
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XZUPOSGJWHSFAX
|
6.7 | IC50 | 2 | — | |
QUYIDBQRQADSRU
|
6.7 | IC50 | 2 | — | |
LPAULIXUZNIAQB
|
6.7 | IC50 | 2 | — | |
NZXHDXCFOVXCIS
|
6.7 | IC50 | 2 | — | |
ZUYRHZPMTJHLLP
|
6.7 | IC50 | 2 | — | |
QETCCDKOGJYGPE
|
6.7 | IC50 | 2 | — | |
GJXAHJGBUHLBIJ
|
6.6 | IC50 | 2 | — | |
KIEQYIJZGSJRCI
|
6.6 | IC50 | 2 | — | |
IVABHIBSCUZIJC
|
6.6 | IC50 | 2 | — | |
PBMPEXWMZJDNKQ
|
6.6 | IC50 | 2 | — | |
JMFZDOZFSCZKIL
|
6.6 | IC50 | 2 | — | |
YIVATKPBWYSRKM
|
6.6 | IC50 | 2 | — | |
HRCANAIPZZVDRQ
|
6.6 | IC50 | 2 | — | |
NQEKNLBAZBZRST
|
6.6 | IC50 | 2 | — | |
ULRNQBZYHZFNNJ
|
6.6 | IC50 | 2 | — | |
UOKGZPYGRJDACN
|
6.6 | IC50 | 7 | Yes | |
ZRRZCDIHCHFDRR
|
6.6 | IC50 | 2 | — | |
WUECGPBROZUDNQ
|
6.6 | IC50 | 2 | — | |
YOERETJHCLVSKU
|
6.6 | IC50 | 2 | — | |
INMSGESUKZJUQI
|
6.6 | IC50 | 2 | — | |
IYRBYYVLBSVPMQ
|
6.6 | IC50 | 2 | — | |
MSZARNKUTLCEOK
|
6.6 | IC50 | 2 | — | |
ARUKIZSLQFCUHJ
|
6.5 | IC50 | 2 | — | |
JGBPEBXXYSKYMT
|
6.5 | IC50 | 2 | — | |
YTFQTLDICXXHOV
|
6.5 | IC50 | 2 | — | |
MLJJFIFPBSIXMF
|
6.5 | IC50 | 2 | — | |
XDFGIRYIOADGQC
|
6.5 | IC50 | 2 | — | |
KVWIBTWIQNUDAW
|
6.5 | IC50 | 2 | — | |
WGDTUWQZIICPGE
|
6.5 | IC50 | 2 | — | |
BJSNIBQSXKKSGB
|
6.5 | IC50 | 2 | — | |
ZKRQAIRGNZQYEW
|
6.5 | IC50 | 2 | — | |
HTFKMKKLSFEKLE
|
6.5 | IC50 | 2 | — | |
JMYDKZPDDRCJDG
|
6.5 | IC50 | 2 | — | |
SMUNQTVQGIWCLD
|
6.5 | IC50 | 2 | — | |
VINUTNSITPWXDD
|
6.4 | IC50 | 2 | — | |
ZXKPXFGTJBBJGQ
|
6.4 | IC50 | 2 | — | |
ULBMHPWYZIPTRZ
|
6.4 | IC50 | 2 | — | |
MOWZHOSXFCAOCS
|
6.4 | IC50 | 2 | — | |
NOUXCUCVFQMAIM
|
6.4 | IC50 | 2 | — | |
XSHQBIXMLULFEV
|
6.4 | IC50 | 13 | — | |
VQQVPNPRBMXNPM
|
6.4 | IC50 | 2 | — | |
BAHMBPJZGYBLIO
|
6.3 | IC50 | 2 | — | |
VQDSYSHRRXTEOA
|
6.3 | IC50 | 2 | — | |
ILKDWZKZLIHMFM
|
6.3 | IC50 | 8 | — | |
SRJOPLMFGKVXMP
|
6.3 | IC50 | 2 | — | |
MVIHEGXCXLFEMC
|
6.3 | IC50 | 4 | — | |
QHLQNXZTJUCDDL
|
6.2 | IC50 | 2 | — | |
HPUGSXICKYRBKG
|
6.2 | IC50 | 2 | — | |
UVAWLRVDFFZJLV
|
6.2 | IC50 | 2 | — | |
YYNKKHDPIFRJSN
|
6.1 | IC50 | 2 | — |