Target Details
| UniProt AC | Q13393 |
|---|---|
| Gene Symbol | PLD1 |
| Protein Name | Phospholipase D1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00169 (PH) PF00614 (PLDc) PF13091 (PLDc_2) PF00787 (PX) |
Summary
- Multi-target molecules 309
- Clinical molecules 1
- Avg pChEMBL 7.29
KEGG Pathways (16)
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Endocytosis
- Ether lipid metabolism
- Fc gamma R-mediated phagocytosis
- Glutamatergic synapse
- Glycerophospholipid metabolism
- GnRH signaling pathway
- Metabolic pathways
- Pancreatic cancer
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Phospholipase D signaling pathway
- Ras signaling pathway
- Sphingolipid signaling pathway
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IUVMBCWHRADVCG
|
7.4 | IC50 | 2 | — | |
LEGHNVWKVYNKKN
|
7.4 | IC50 | 2 | — | |
OYCZAQWPOJRNFX
|
7.4 | IC50 | 2 | — | |
UIOJSVXCECGAEL
|
7.4 | IC50 | 2 | — | |
LWPPVRZWNRKLJH
|
7.4 | IC50 | 2 | — | |
MJEJRCOVVQBCRU
|
7.4 | IC50 | 2 | — | |
AOQBWSMWTCRNGX
|
7.3 | IC50 | 2 | — | |
PBVNVWVUHATERF
|
7.3 | IC50 | 2 | — | |
YCJSIBLGQJIWDH
|
7.3 | IC50 | 2 | — | |
YNXITEIAXSVMJI
|
7.3 | IC50 | 2 | — | |
CRHGZNNSBJNMPL
|
7.3 | IC50 | 2 | — | |
DRIMIUYGTDAQOX
|
7.3 | IC50 | 2 | — | |
IXGWLWZIGFRGDR
|
7.3 | IC50 | 2 | — | |
KHFXETJCUMUPHB
|
7.3 | IC50 | 2 | — | |
VSVQUDYXUOHKEV
|
7.3 | IC50 | 2 | — | |
DRLLWYJGUKYYKT
|
7.3 | IC50 | 2 | — | |
AMDSHJQDFLEAPT
|
7.3 | IC50 | 2 | — | |
NLUMBNOKEOCUQG
|
7.3 | IC50 | 2 | — | |
SEPMEKJITYIWGF
|
7.3 | IC50 | 2 | — | |
YEDRZAMDJSGXSJ
|
7.3 | IC50 | 2 | — | |
APJRFCWYQFJHGB
|
7.2 | IC50 | 2 | — | |
KTAATQUDEMNBHO
|
7.2 | IC50 | 2 | — | |
WKZPHFNFYXVPCM
|
7.2 | IC50 | 2 | — | |
BPUCGNUARDSAOI
|
7.2 | IC50 | 2 | — | |
LIYOXSHYNMNNMX
|
7.2 | IC50 | 2 | — | |
MVZPDWNZEYMGQG
|
7.2 | IC50 | 2 | — | |
WNYCYGCNORZQPH
|
7.2 | IC50 | 2 | — | |
SNSUBJOGYOJHHN
|
7.2 | IC50 | 2 | — | |
COOIOSTYBGGMTL
|
7.2 | IC50 | 2 | — | |
KTAATQUDEMNBHO
|
7.2 | IC50 | 2 | — | |
CLLNHRCVIIUYSP
|
7.2 | IC50 | 2 | — | |
FTIMUWXHUSLHKZ
|
7.2 | IC50 | 2 | — | |
HHOJOWSNAJQLGJ
|
7.2 | IC50 | 2 | — | |
TYGKALZYXWTOJQ
|
7.2 | IC50 | 2 | — | |
TYNAPBDIKCLKGO
|
7.2 | IC50 | 2 | — | |
FWQNFTIWJZDHLW
|
7.2 | IC50 | 2 | — | |
AQBINFRWIVSTNH
|
7.2 | IC50 | 2 | — | |
JRLJLDRKZKLXKK
|
7.2 | IC50 | 2 | — | |
SAYDLSNHEFBCSP
|
7.2 | IC50 | 2 | — | |
XKLWCFAKYSNXEQ
|
7.2 | IC50 | 2 | — | |
FIQSXKOIBQFWLX
|
7.1 | IC50 | 2 | — | |
ZWWQYHMQQPNGJJ
|
7.1 | IC50 | 2 | — | |
AWGOXNPIJXMUOD
|
7.1 | IC50 | 2 | — | |
RFKXAYJUFUZBMA
|
7.1 | IC50 | 2 | — | |
FQFFYVYBFUVPGG
|
7.1 | IC50 | 2 | — | |
IXLLRNNFUYEADZ
|
7.1 | IC50 | 2 | — | |
GYXOIULGUSTJEH
|
7.1 | IC50 | 2 | — | |
FXCPNMVRVXUAGZ
|
7.1 | IC50 | 2 | — | |
SLNRIYGPRGCBAK
|
7.1 | IC50 | 2 | — | |
JFFLYDRHDDWALA
|
7.1 | IC50 | 2 | — |