Target Details
| UniProt AC | Q13393 |
|---|---|
| Gene Symbol | PLD1 |
| Protein Name | Phospholipase D1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00169 (PH) PF00614 (PLDc) PF13091 (PLDc_2) PF00787 (PX) |
Summary
- Multi-target molecules 309
- Clinical molecules 1
- Avg pChEMBL 7.29
KEGG Pathways (16)
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Endocytosis
- Ether lipid metabolism
- Fc gamma R-mediated phagocytosis
- Glutamatergic synapse
- Glycerophospholipid metabolism
- GnRH signaling pathway
- Metabolic pathways
- Pancreatic cancer
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Phospholipase D signaling pathway
- Ras signaling pathway
- Sphingolipid signaling pathway
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NDSWYRYHESOGHB
|
7.6 | IC50 | 2 | — | |
QIDIOVNYYFENPN
|
7.6 | IC50 | 2 | — | |
UBRSEWJZIORIJP
|
7.6 | IC50 | 2 | — | |
UDTGVCDGNVXVTB
|
7.6 | IC50 | 2 | — | |
XJCZYPYMNVFQCU
|
7.6 | IC50 | 2 | — | |
DBEKQTQXJPKLML
|
7.5 | IC50 | 2 | — | |
UXRNIIRMQLYYFA
|
7.5 | IC50 | 2 | — | |
JHUHHBBYJSRVJQ
|
7.5 | IC50 | 2 | — | |
KIIXLQWDXRMANC
|
7.5 | IC50 | 2 | — | |
OHQVPJLSLKNZKZ
|
7.5 | IC50 | 2 | — | |
OTPWKFYADLFEEO
|
7.5 | IC50 | 2 | — | |
RXOYNWHWLALWQL
|
7.5 | IC50 | 2 | — | |
DLUPXNMRCKJWAL
|
7.5 | IC50 | 2 | — | |
FKTRMPQBGCZBRZ
|
7.5 | IC50 | 2 | — | |
FOVKVWCJRIQJSJ
|
7.5 | IC50 | 2 | — | |
GCNASPCPGQAUQY
|
7.5 | IC50 | 2 | — | |
JLJOIYYJDOJZDM
|
7.5 | IC50 | 2 | — | |
OLBVSDIHGLJWOC
|
7.5 | IC50 | 2 | — | |
WAJCYNWNVYRAPB
|
7.5 | IC50 | 2 | — | |
HYCGYICLLKSQMN
|
7.5 | IC50 | 2 | — | |
KPNDMXHPGLZXCL
|
7.5 | IC50 | 2 | — | |
XFPLPNQDZHMCDM
|
7.5 | IC50 | 2 | — | |
ARMZNEAMIDUKRJ
|
7.5 | IC50 | 2 | — | |
BBNKAFWTEFUAQZ
|
7.5 | IC50 | 2 | — | |
BFRGUJCFIYTJDR
|
7.5 | IC50 | 2 | — | |
HYUQKTOSTOPFRH
|
7.5 | IC50 | 2 | — | |
DRXXUPYAYMSQSQ
|
7.5 | IC50 | 2 | — | |
FJLQWJXTAWKZRU
|
7.5 | IC50 | 2 | — | |
FCHRUZHGMJRVTC
|
7.5 | IC50 | 2 | — | |
RPNWIDZCXVGQPT
|
7.5 | IC50 | 2 | — | |
UQEMLZKHAQPVOU
|
7.5 | IC50 | 2 | — | |
YWBSXKSUAXYZFW
|
7.5 | IC50 | 2 | — | |
ASSCTZAOZGZFBS
|
7.4 | IC50 | 2 | — | |
LNBKAIMWXSJEPK
|
7.4 | IC50 | 2 | — | |
XGCOKDOXUPKYDC
|
7.4 | IC50 | 2 | — | |
JUVRFAVSTPVCNE
|
7.4 | IC50 | 2 | — | |
NZLJVMMLHOTFAG
|
7.4 | IC50 | 2 | — | |
VOGNGPBBHABISW
|
7.4 | IC50 | 2 | — | |
AIEXUFPTTDMPRC
|
7.4 | IC50 | 2 | — | |
BUMZOIBPBJTWIL
|
7.4 | IC50 | 2 | — | |
SARPSSFXUSFCDB
|
7.4 | IC50 | 2 | — | |
IZWYURUKGNFWMK
|
7.4 | IC50 | 2 | — | |
LWPPVRZWNRKLJH
|
7.4 | IC50 | 2 | — | |
MDIQXYIDELVTLG
|
7.4 | IC50 | 2 | — | |
ZCPAKJKFPGVKMN
|
7.4 | IC50 | 2 | — | |
BTZFCQGLCLGZJB
|
7.4 | IC50 | 2 | — | |
UKFTYRWQERGPME
|
7.4 | IC50 | 2 | — | |
DTKIOTNZOCNINZ
|
7.4 | IC50 | 2 | — | |
QZTNMIITKLUEOG
|
7.4 | IC50 | 2 | — | |
ROILKBDWDUQTQU
|
7.4 | IC50 | 2 | — |