Target Details
| UniProt AC | Q13393 |
|---|---|
| Gene Symbol | PLD1 |
| Protein Name | Phospholipase D1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00169 (PH) PF00614 (PLDc) PF13091 (PLDc_2) PF00787 (PX) |
Summary
- Multi-target molecules 309
- Clinical molecules 1
- Avg pChEMBL 7.29
KEGG Pathways (16)
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Endocytosis
- Ether lipid metabolism
- Fc gamma R-mediated phagocytosis
- Glutamatergic synapse
- Glycerophospholipid metabolism
- GnRH signaling pathway
- Metabolic pathways
- Pancreatic cancer
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Phospholipase D signaling pathway
- Ras signaling pathway
- Sphingolipid signaling pathway
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DVYOUIBPYDWRAD
|
7.8 | IC50 | 2 | — | |
HDGZQALFFUBJMH
|
7.8 | IC50 | 2 | — | |
MCDNCMGVHBZICR
|
7.8 | IC50 | 2 | — | |
PKHUOIJRGIGZGB
|
7.8 | IC50 | 2 | — | |
SDFDDJALBRFAGL
|
7.8 | IC50 | 2 | — | |
VZIYKSOAERBDKN
|
7.8 | IC50 | 2 | — | |
COFPYVCKURUCND
|
7.7 | IC50 | 2 | — | |
PZXNWTCLLPQFLO
|
7.7 | IC50 | 2 | — | |
GHCNKPDLSIGADO
|
7.7 | IC50 | 2 | — | |
ASDFSRNMHPUURW
|
7.7 | IC50 | 2 | — | |
FKXBLUNBTQZMJI
|
7.7 | IC50 | 2 | — | |
NBROEJLBCWNSAV
|
7.7 | IC50 | 2 | — | |
OKVRCZNCIXFZRK
|
7.7 | IC50 | 2 | — | |
XUKRCEKSPDAOQE
|
7.7 | IC50 | 2 | — | |
FJUCIFYXMXZWOU
|
7.7 | IC50 | 2 | — | |
KCVCYFCTEPOPIX
|
7.7 | IC50 | 2 | — | |
MLJJFIFPBSIXMF
|
7.7 | IC50 | 2 | — | |
NBHPRWLFLUBAIE
|
7.7 | IC50 | 3 | — | |
UPDQTPSMDKPOCO
|
7.7 | IC50 | 2 | — | |
YPLWURRTGNQZTF
|
7.7 | IC50 | 2 | — | |
ZESQLHZOEOPFBM
|
7.7 | IC50 | 2 | — | |
ZLSKWSRGUOBONO
|
7.7 | IC50 | 2 | — | |
QLCFHHJOCOKGIV
|
7.7 | IC50 | 2 | — | |
GUXCVFKSLGMQOV
|
7.6 | IC50 | 2 | — | |
ONGBMNKFMKQBLC
|
7.6 | IC50 | 2 | — | |
RGXGHHOHYCFOPB
|
7.6 | IC50 | 2 | — | |
VBABLIIDDVFNQO
|
7.6 | IC50 | 2 | — | |
WOPSTAVQRUXOAA
|
7.6 | IC50 | 2 | — | |
WXVKMBZKSDYISN
|
7.6 | IC50 | 2 | — | |
ZEQAZSTXQGDDNQ
|
7.6 | IC50 | 2 | — | |
KUZKHNITNUUBGC
|
7.6 | IC50 | 2 | — | |
SUDHHKMBVPBXAQ
|
7.6 | IC50 | 2 | — | |
AMRVRQLHZXWMKB
|
7.6 | IC50 | 2 | — | |
KBMPJZSFOFZBQM
|
7.6 | IC50 | 2 | — | |
LZYJPIITZHZRLU
|
7.6 | IC50 | 2 | — | |
NWCJMCPTWFMEST
|
7.6 | IC50 | 2 | — | |
VALMDDHRZJXVOR
|
7.6 | IC50 | 2 | — | |
XISOZGLNHJHWPW
|
7.6 | IC50 | 2 | — | |
FDEPYPCYKHDPDF
|
7.6 | IC50 | 2 | — | |
GCVGWSQRPUQQJH
|
7.6 | IC50 | 2 | — | |
LAHOJMBICQHKHJ
|
7.6 | IC50 | 2 | — | |
PJNHTJBHQKTGOS
|
7.6 | IC50 | 2 | — | |
PXBKGMJWXHLVBN
|
7.6 | IC50 | 2 | — | |
QDYHNIGIBCJKIU
|
7.6 | IC50 | 2 | — | |
ZFKKKKMLLHXPBQ
|
7.6 | IC50 | 2 | — | |
ZGIZOXJDYPMVLA
|
7.6 | IC50 | 2 | — | |
IJGGHESNESJBMG
|
7.6 | IC50 | 2 | — | |
JYHPSYLWFWPJBU
|
7.6 | IC50 | 2 | — | |
LEUKGNOUEBECCA
|
7.6 | IC50 | 2 | — | |
LHSLMYPOSYZMQY
|
7.6 | IC50 | 2 | — |