Target Details
| UniProt AC | Q13393 |
|---|---|
| Gene Symbol | PLD1 |
| Protein Name | Phospholipase D1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00169 (PH) PF00614 (PLDc) PF13091 (PLDc_2) PF00787 (PX) |
Summary
- Multi-target molecules 309
- Clinical molecules 1
- Avg pChEMBL 7.29
KEGG Pathways (16)
- Chemical carcinogenesis - reactive oxygen species
- Choline metabolism in cancer
- Endocytosis
- Ether lipid metabolism
- Fc gamma R-mediated phagocytosis
- Glutamatergic synapse
- Glycerophospholipid metabolism
- GnRH signaling pathway
- Metabolic pathways
- Pancreatic cancer
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Phospholipase D signaling pathway
- Ras signaling pathway
- Sphingolipid signaling pathway
- cAMP signaling pathway
Associated Diseases (1)
Active Molecules (309)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CUBHHKRMIJNNFB
|
9.0 | IC50 | 2 | — | |
HIMZKRKANIVDNR
|
9.0 | IC50 | 2 | — | |
MSSVPLXKRPFKDV
|
9.0 | IC50 | 2 | — | |
MDMOJYODKZQMGP
|
8.7 | IC50 | 2 | — | |
MSUMQFORLFESPA
|
8.7 | IC50 | 2 | — | |
MWKBJPMDIRQKGV
|
8.7 | IC50 | 2 | — | |
REVZYRDPYGXHCC
|
8.7 | IC50 | 2 | — | |
ZNFHTAUUBDJHTE
|
8.7 | IC50 | 2 | — | |
GMZVJMYMLXBFRA
|
8.5 | IC50 | 2 | — | |
HUUWWQMWJIZOTF
|
8.5 | IC50 | 2 | — | |
LPIPUHBDLDDLRV
|
8.5 | IC50 | 2 | — | |
HBVVABXIVRGPET
|
8.5 | IC50 | 2 | — | |
ZNFHTAUUBDJHTE
|
8.4 | IC50 | 2 | — | |
AVJLSXGOQNVYRT
|
8.4 | IC50 | 2 | — | |
BSGGZEUVJPHPOY
|
8.4 | IC50 | 2 | — | |
CRHUKUIICKDJBR
|
8.4 | IC50 | 2 | — | |
QYLRVQUJNPPZPM
|
8.4 | IC50 | 2 | — | |
WCCRPCLBWZNRNV
|
8.4 | IC50 | 2 | — | |
XYFYPTXOUKXAET
|
8.4 | IC50 | 2 | — | |
PBLTYRBFXNGWNE
|
8.4 | IC50 | 2 | — | |
FOKWDPRXQQGFID
|
8.3 | IC50 | 2 | — | |
HPTPLUVUBNHEQY
|
8.3 | IC50 | 2 | — | |
HWHBSTPKWDIKIG
|
8.3 | IC50 | 2 | — | |
LWPPJHFDFCBNHR
|
8.3 | IC50 | 2 | — | |
YJQWRAAPDSTDOW
|
8.2 | IC50 | 2 | — | |
RFKXAYJUFUZBMA
|
8.2 | IC50 | 2 | — | |
AREIGOLWYGBISF
|
8.2 | IC50 | 2 | — | |
LPNLGPZYTTUDSO
|
8.2 | IC50 | 2 | — | |
QRQOZMAZJKRVIF
|
8.2 | IC50 | 2 | — | |
HXMOFRYLDQHGOC
|
8.1 | IC50 | 2 | — | |
JPNXEMBKUUKKCS
|
8.1 | IC50 | 2 | — | |
QYXQSMNQBJSTTJ
|
8.1 | IC50 | 2 | — | |
HGYSAUZNGFRJIG
|
8.1 | IC50 | 2 | — | |
SZYKHOATMDIEMC
|
8.1 | IC50 | 2 | — | |
IISXBFMJBUQZEA
|
8.0 | IC50 | 2 | — | |
MNKBFXBSNSUUTP
|
8.0 | IC50 | 2 | — | |
OPIZCRLQYOQSKJ
|
8.0 | IC50 | 2 | — | |
QMXFZMPBYFJYLO
|
7.9 | IC50 | 2 | — | |
XOHZLGSSMQKYGN
|
7.9 | IC50 | 2 | — | |
ZAAQLYAZEYYWIE
|
7.9 | IC50 | 2 | — | |
LHABRXRGDLASIH
|
7.9 | IC50 | 2 | — | |
GHCJQOQUTCHJQB
|
7.8 | IC50 | 2 | — | |
SHEQGRPLNRDRQC
|
7.8 | IC50 | 2 | — | |
UDJCBYWCKABSOL
|
7.8 | IC50 | 2 | — | |
UYRJZCTXPMSAAL
|
7.8 | IC50 | 2 | — | |
YNXITEIAXSVMJI
|
7.8 | IC50 | 2 | — | |
BLGZUAXJXQZYJK
|
7.8 | IC50 | 2 | — | |
CUBHHKRMIJNNFB
|
7.8 | IC50 | 2 | — | |
GXCLXNQTXLNGOA
|
7.8 | IC50 | 2 | — | |
SFJGIYVIEAZRDO
|
7.8 | IC50 | 2 | — |