Target Details
| UniProt AC | Q13324 |
|---|---|
| Gene Symbol | CRHR2 |
| Protein Name | Corticotropin-releasing factor receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00002 (7tm_2) PF02793 (HRM) |
Summary
- Multi-target molecules 42
- Clinical molecules 0
- Avg pChEMBL 7.7
KEGG Pathways (4)
Active Molecules (42)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BIIOOWPFSOAZSO
|
9.9 | IC50 | 2 | — | |
QBZAHNFIFYKUAQ
|
9.4 | IC50 | 2 | — | |
UPVFHCQGPPALAB
|
9.3 | IC50 | 2 | — | |
BBNGUKKQYPAMTB
|
9.2 | IC50 | 2 | — | |
BPJKLNRBFUIHRZ
|
9.2 | IC50 | 2 | — | |
VHTUCYOJWFRPJN
|
9.2 | IC50 | 2 | — | |
HPYIIXJJVYSMCV
|
9.2 | IC50 | 2 | — | |
ZXQWGXPBQWFYKG
|
9.2 | IC50 | 2 | — | |
KBXXQHLYNYCQAE
|
9.1 | IC50 | 2 | — | |
BXTRKRJIYZENAK
|
8.9 | IC50 | 2 | — | |
YIHRBRJTFIGRRV
|
8.9 | Ki | 2 | — | |
YIHRBRJTFIGRRV
|
8.9 | Ki | 2 | — | |
IQJNGBXKROFQRM
|
8.9 | IC50 | 2 | — | |
KFUIXDNQSMKKJQ
|
8.8 | IC50 | 2 | — | |
FUFHRWPFPLHLRL
|
8.6 | Ki | 2 | — | |
BIIOOWPFSOAZSO
|
8.4 | Ki | 2 | — | |
YZGWWUVHEOPLKF
|
8.3 | IC50 | 2 | — | |
CMZOBLKSINEYCW
|
8.3 | IC50 | 2 | — | |
HBBPLUNKEXJZQZ
|
8.3 | IC50 | 2 | — | |
PNMZQWKBJIQQJL
|
8.2 | IC50 | 2 | — | |
WBNJZEUGPLZJAS
|
8.2 | IC50 | 2 | — | |
GBONBLHJMVUBSJ
|
7.9 | Ki | 2 | — | |
GBONBLHJMVUBSJ
|
7.9 | Ki | 2 | — | |
BYXIIQICFOHBMN
|
7.3 | IC50 | 2 | — | |
QBKRBQAPESJEEH
|
7.2 | IC50 | 2 | — | |
QEEJLLNYQOBRRM
|
7.1 | Ki | 2 | — | |
QEEJLLNYQOBRRM
|
7.1 | Ki | 2 | — | |
FFMNQLRIMQJKNK
|
6.6 | IC50 | 2 | — | |
LSFVOPLRJHUUNQ
|
6.5 | IC50 | 2 | — | |
FTOXJSMDKHMORW
|
6.3 | IC50 | 2 | — | |
KZZNPWMYQJUTPP
|
6.2 | IC50 | 2 | — | |
BKABKOFLTNTFIF
|
6.1 | IC50 | 2 | — | |
DOEWJZPYNWPPDF
|
6.1 | IC50 | 2 | — | |
MRNRDFOQXNZICL
|
6.1 | IC50 | 2 | — | |
KGXVFKLVFKBFRR
|
6.1 | IC50 | 2 | — | |
IMAXYSCPKOIFBE
|
6.1 | IC50 | 2 | — | |
GALUEGSXWCYSQD
|
6.1 | IC50 | 2 | — | |
ZEGBRYNTIJDVHP
|
6.1 | IC50 | 2 | — | |
KCPHVCVRMSDLQN
|
6.0 | IC50 | 2 | — | |
ZUYRUNKZVZVHHE
|
6.0 | IC50 | 2 | — | |
AKHFOJODMTWXAB
|
6.0 | IC50 | 2 | — | |
KZXCSFVNVIGEKX
|
6.0 | IC50 | 2 | — |