Target Details
| UniProt AC | Q13315 |
|---|---|
| Gene Symbol | ATM |
| Protein Name | Serine-protein kinase ATM |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02259 (FAT) PF02260 (FATC) PF00454 (PI3_PI4_kinase) PF11640 (TAN) |
Summary
- Multi-target molecules 170
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (14)
- Apoptosis
- Cell cycle
- Cellular senescence
- FoxO signaling pathway
- Homologous recombination
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- MicroRNAs in cancer
- NF-kappa B signaling pathway
- Platinum drug resistance
- Shigellosis
- Transcriptional misregulation in cancer
- p53 signaling pathway
Associated Diseases (3)
Active Molecules (170)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FPHLASQTEAWKKW
|
6.3 | IC50 | 2 | — | |
GQUJOOVYNSNQLU
|
6.3 | IC50 | 3 | — | |
GYWPMKOUCJEYNO
|
6.3 | IC50 | 3 | — | |
JQXHDOKWOABELF
|
6.3 | IC50 | 2 | — | |
KASNAMAOPPOPNR
|
6.3 | IC50 | 2 | — | |
OHERNBRGXOVCSR
|
6.3 | IC50 | 4 | — | |
PDYCTPQIULBADZ
|
6.3 | IC50 | 2 | — | |
PQQPUILDPHGQHI
|
6.3 | IC50 | 2 | — | |
SCJFBVYWHMWCLF
|
6.3 | IC50 | 2 | — | |
TXGXVGZVOFHZBI
|
6.3 | IC50 | 4 | — | |
UUAWGVGBYJWRND
|
6.3 | IC50 | 2 | — | |
VIGQGNDNBYWABF
|
6.3 | IC50 | 2 | — | |
VTNYVWSVPWEXFE
|
6.3 | IC50 | 4 | — | |
XMSRADCMDDJZDM
|
6.3 | IC50 | 3 | — | |
XYUHZXOGIAVMOX
|
6.3 | IC50 | 2 | — | |
ZXUAFMGZIYRRQO
|
6.3 | IC50 | 3 | — | |
WOXCVRPHALGLIX
|
6.1 | IC50 | 2 | — | |
XZOGJLXYXXEFHY
|
6.1 | IC50 | 2 | — | |
WRNCIFYXNUAFIH
|
6.0 | IC50 | 2 | — | |
LKHMVKNMSWRHJH
|
6.0 | IC50 | 7 | — |