Target Details
| UniProt AC | Q13315 |
|---|---|
| Gene Symbol | ATM |
| Protein Name | Serine-protein kinase ATM |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02259 (FAT) PF02260 (FATC) PF00454 (PI3_PI4_kinase) PF11640 (TAN) |
Summary
- Multi-target molecules 170
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (14)
- Apoptosis
- Cell cycle
- Cellular senescence
- FoxO signaling pathway
- Homologous recombination
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- MicroRNAs in cancer
- NF-kappa B signaling pathway
- Platinum drug resistance
- Shigellosis
- Transcriptional misregulation in cancer
- p53 signaling pathway
Associated Diseases (3)
Active Molecules (170)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LUBFLYDYTPVXHF
|
7.3 | IC50 | 2 | — | |
LUGPTJMETIONMP
|
7.3 | IC50 | 3 | — | |
LUMCFRRSGMTLBH
|
7.3 | IC50 | 3 | — | |
NDYPMEATJRJEHM
|
7.3 | IC50 | 3 | — | |
OOGWCQBQPOULGK
|
7.3 | IC50 | 3 | — | |
PEKHSWOOLJTLAP
|
7.3 | IC50 | 3 | — | |
PUWSVGWDZWYMHD
|
7.3 | IC50 | 3 | — | |
QIUXGKIHBYLVDG
|
7.3 | IC50 | 3 | — | |
SUSHENREWKQEFA
|
7.3 | IC50 | 3 | — | |
WLGXNSHVQAUMAT
|
7.3 | IC50 | 3 | — | |
WTOVLONEHSCFLI
|
7.3 | IC50 | 3 | — | |
ZITCKJQNZLGXNI
|
7.3 | IC50 | 2 | — | |
OEWUSAJPHBVLOD
|
7.2 | IC50 | 2 | — | |
VYPJIEHUDAVBLF
|
7.2 | IC50 | 2 | — | |
PQEIMHBVHXTVNA
|
7.2 | IC50 | 5 | — | |
KHOSFSGTKQFGDP
|
7.1 | IC50 | 2 | — | |
DYJRBYYBKYZZGT
|
7.1 | IC50 | 4 | — | |
DPKWEPQBVKHUQT
|
7.1 | IC50 | 4 | — | |
BRGUQOISTYVOBM
|
7.1 | Ki | 3 | — | |
BZDFDZUZTQDDOL
|
7.1 | Ki | 2 | — | |
WLGXNSHVQAUMAT
|
7.1 | IC50 | 4 | — | |
WLVBJQUVPORFNZ
|
7.0 | Ki | 2 | — | |
BRGUQOISTYVOBM
|
7.0 | Ki | 2 | — | |
BLHDWFGAYUVFER
|
6.9 | Ki | 2 | — | |
MQWCGLLYOBFYNX
|
6.9 | IC50 | 2 | — | |
KCBCGZCZHKEUPT
|
6.9 | IC50 | 2 | — | |
KQZZSMVSVVANOL
|
6.9 | IC50 | 4 | — | |
UFZMEAYSFGBIBJ
|
6.9 | IC50 | 4 | — | |
NGJICJQCRNGWDQ
|
6.9 | IC50 | 4 | — | |
UBFGOBLWCVBCBP
|
6.9 | IC50 | 2 | — | |
HAFHNTJKCXCNQK
|
6.7 | Ki | 2 | — | |
WEOFJQBDUVLXHQ
|
6.7 | Ki | 2 | — | |
HLCDNLNLQNYZTK
|
6.7 | IC50 | 2 | — | |
UMGDCJDMYOKAJW
|
6.7 | IC50 | 2 | — | |
HZYTVQKACFDSMV
|
6.7 | IC50 | 4 | — | |
YFHBYQHMVTVHDA
|
6.5 | IC50 | 3 | — | |
OKNNPZZFEHDVHC
|
6.5 | IC50 | 2 | — | |
QPTLAOOZWOLYLB
|
6.4 | IC50 | 2 | — | |
NVZFTEWCKUYXCM
|
6.4 | IC50 | 2 | — | |
ZFQAKLNTCBPIMT
|
6.4 | Ki | 2 | — | |
HBYVDORXKRHBBS
|
6.4 | IC50 | 3 | — | |
YSOQBYOYIBXQGO
|
6.4 | IC50 | 6 | — | |
JKADCYKTYYGDKT
|
6.3 | IC50 | 2 | — | |
YMLAOBUVHWUIQH
|
6.3 | IC50 | 4 | — | |
MFZAHAAVYSHLCP
|
6.3 | IC50 | 7 | — | |
BBNGXFSLGHDPJG
|
6.3 | IC50 | 3 | — | |
BSGBCKRSUJYENI
|
6.3 | IC50 | 2 | — | |
CIZCIUKZKXFSME
|
6.3 | IC50 | 2 | — | |
DFUFAVMVCOEDLG
|
6.3 | IC50 | 2 | — | |
DPLMXAYKJZOTKO
|
6.3 | IC50 | 5 | — |