Target Details
| UniProt AC | Q13315 |
|---|---|
| Gene Symbol | ATM |
| Protein Name | Serine-protein kinase ATM |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02259 (FAT) PF02260 (FATC) PF00454 (PI3_PI4_kinase) PF11640 (TAN) |
Summary
- Multi-target molecules 170
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (14)
- Apoptosis
- Cell cycle
- Cellular senescence
- FoxO signaling pathway
- Homologous recombination
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- MicroRNAs in cancer
- NF-kappa B signaling pathway
- Platinum drug resistance
- Shigellosis
- Transcriptional misregulation in cancer
- p53 signaling pathway
Associated Diseases (3)
Active Molecules (170)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
TWIZQAVJLJJRIO
|
8.3 | IC50 | 2 | — | |
VFJHEBMKBXLCDG
|
8.3 | IC50 | 2 | — | |
XNQLBCLHQMLKIC
|
8.3 | IC50 | 3 | — | |
YVQDIBOPRZOYGI
|
8.3 | IC50 | 3 | — | |
FZLLSBHPQYLGLH
|
8.2 | Ki | 2 | — | |
SYYKNMAYZDJNLK
|
8.2 | IC50 | 2 | — | |
HRZBUHAVTBTHTM
|
8.2 | IC50 | 3 | — | |
FZLLSBHPQYLGLH
|
8.2 | IC50 | 2 | — | |
JOGKUKXHTYWRGZ
|
8.2 | IC50 | 28 | — | |
KGAAOKXUCALAPY
|
8.2 | IC50 | 8 | — | |
BWCDJBGHHAEAMF
|
8.1 | IC50 | 2 | — | |
PQUHOMYHDNTHRG
|
8.1 | IC50 | 2 | — | |
FZLLSBHPQYLGLH
|
8.0 | IC50 | 3 | — | |
CORFNGYLXZFTMD
|
8.0 | IC50 | 3 | — | |
KREZBWKMMRSYDH
|
8.0 | IC50 | 2 | — | |
NRCHETGDZOLUIQ
|
8.0 | IC50 | 4 | — | |
SCELLOWTHJGVIC
|
8.0 | IC50 | 4 | — | |
FPWSKINOJYCEJK
|
7.9 | IC50 | 3 | — | |
XRKYMMUGXMWDAO
|
7.9 | IC50 | 5 | Yes | |
SYVQAQHCFMTBNA
|
7.8 | IC50 | 3 | — | |
KZJLHYQNEJSYNN
|
7.8 | IC50 | 6 | — | |
NUUYFIBMHLLMSL
|
7.8 | IC50 | 2 | — | |
FNNGURVIOIZXRF
|
7.8 | IC50 | 3 | — | |
YWWWQQYKTOUASO
|
7.7 | IC50 | 3 | — | |
ZJXHODMMACVLQQ
|
7.7 | IC50 | 3 | — | |
ILBRKJBKDGCSCB
|
7.7 | IC50 | 2 | — | |
JJVQWARGSDQRCL
|
7.7 | IC50 | 2 | — | |
YBKLBECNVUXSJN
|
7.6 | Ki | 2 | — | |
GCKKBGHFJIZIAB
|
7.6 | IC50 | 3 | — | |
GWPIPOHZYJCBCD
|
7.6 | IC50 | 4 | — | |
NUUYFIBMHLLMSL
|
7.5 | Ki | 2 | — | |
XHNKFGYYGPLYPT
|
7.5 | IC50 | 3 | — | |
JEKDMEAMHWNRLL
|
7.4 | IC50 | 4 | — | |
IAQPXVJIBLLKDW
|
7.4 | IC50 | 2 | — | |
JZCWLJDSIRUGIN
|
7.4 | IC50 | 16 | — | |
DISRGUXSEDBDDN
|
7.3 | IC50 | 2 | — | |
ZVOIZFFFPDDJHJ
|
7.3 | Ki | 2 | — | |
CEUPOOINALBZRR
|
7.3 | IC50 | 6 | — | |
AGPLDYRKDIYXTM
|
7.3 | IC50 | 2 | — | |
CUVROQGPQACSNV
|
7.3 | IC50 | 3 | — | |
DVEUJBRMVAYSCW
|
7.3 | IC50 | 3 | — | |
FLODHIIWXLIRRR
|
7.3 | IC50 | 4 | — | |
GAXWSUSCGHPCKH
|
7.3 | IC50 | 3 | — | |
GKXFLUILDKFQAY
|
7.3 | IC50 | 3 | — | |
GRLIKHGGVMEHAA
|
7.3 | IC50 | 2 | — | |
HKDWNCUIOZJHCX
|
7.3 | IC50 | 2 | — | |
IJDLDJGJYHPWSI
|
7.3 | IC50 | 3 | — | |
JUGUPSCRPXAHBW
|
7.3 | IC50 | 2 | — | |
JVKKETWPNJSWSC
|
7.3 | IC50 | 2 | — | |
LCWHFJMGEPVAGK
|
7.3 | IC50 | 3 | — |