Target Details
| UniProt AC | Q13315 |
|---|---|
| Gene Symbol | ATM |
| Protein Name | Serine-protein kinase ATM |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02259 (FAT) PF02260 (FATC) PF00454 (PI3_PI4_kinase) PF11640 (TAN) |
Summary
- Multi-target molecules 170
- Clinical molecules 1
- Avg pChEMBL 7.64
KEGG Pathways (14)
- Apoptosis
- Cell cycle
- Cellular senescence
- FoxO signaling pathway
- Homologous recombination
- Human T-cell leukemia virus 1 infection
- Human immunodeficiency virus 1 infection
- Human papillomavirus infection
- MicroRNAs in cancer
- NF-kappa B signaling pathway
- Platinum drug resistance
- Shigellosis
- Transcriptional misregulation in cancer
- p53 signaling pathway
Associated Diseases (3)
Active Molecules (170)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZPOCWOPPQUMNCW
|
9.8 | IC50 | 3 | — | |
QNJITDREARMZMY
|
9.7 | IC50 | 2 | — | |
YXJGKECEJNCEIH
|
9.6 | IC50 | 3 | — | |
YXJGKECEJNCEIH
|
9.6 | IC50 | 2 | — | |
NLDJVYUQOPIMNA
|
9.6 | IC50 | 3 | — | |
HVCFZONVQJFMNR
|
9.5 | IC50 | 2 | — | |
NDSGFLSESAHGIW
|
9.5 | IC50 | 3 | — | |
ABKGTFFKSJEJIQ
|
9.5 | IC50 | 2 | — | |
SBWOIJRPFUUCGS
|
9.4 | IC50 | 2 | — | |
OVFIHIWNXSZYOH
|
9.4 | Ki | 2 | — | |
QIUHOMNRLMPPFS
|
9.3 | IC50 | 2 | — | |
ARZGDKFYXFLWNZ
|
9.3 | IC50 | 3 | — | |
SBWOIJRPFUUCGS
|
9.3 | IC50 | 2 | — | |
BHZJNQALHTWTBX
|
9.2 | IC50 | 3 | — | |
AOTRIQLYUAFVSC
|
9.2 | IC50 | 5 | — | |
ARZGDKFYXFLWNZ
|
9.2 | IC50 | 3 | — | |
OPVXIIKFNBQKCN
|
9.2 | IC50 | 2 | — | |
VCKBRXFQRMSHFD
|
9.1 | IC50 | 2 | — | |
DCYIRFHUZMQEJE
|
9.1 | IC50 | 3 | — | |
ABKGTFFKSJEJIQ
|
9.0 | IC50 | 3 | — | |
SIKMYPMDQGCEPL
|
9.0 | IC50 | 3 | — | |
FNNGURVIOIZXRF
|
9.0 | Ki | 2 | — | |
KAHMZYOZNYFPKN
|
9.0 | IC50 | 3 | — | |
OVFIHIWNXSZYOH
|
9.0 | IC50 | 3 | — | |
UNETUVMFOUXHNZ
|
9.0 | IC50 | 2 | — | |
WEEIJHAKEWVFES
|
9.0 | IC50 | 2 | — | |
WMHJLJSPDADNGQ
|
9.0 | IC50 | 2 | — | |
JDAPKZUDSPQCGU
|
9.0 | IC50 | 3 | — | |
PIGDKCHEKYYPIG
|
9.0 | IC50 | 2 | — | |
NJZBNLVCEXZHPD
|
9.0 | IC50 | 2 | — | |
KVVLNFCQHKOZRL
|
9.0 | IC50 | 2 | — | |
MZBVEJCJSWMSLU
|
8.9 | IC50 | 2 | — | |
QEJSKPORGMNWPI
|
8.9 | IC50 | 2 | — | |
SJOFSBIUJPEXTG
|
8.8 | IC50 | 2 | — | |
CIZOSCVUGRBXEZ
|
8.8 | IC50 | 4 | — | |
FZLLSBHPQYLGLH
|
8.7 | Ki | 2 | — | |
IIBZKDYAYJSSGB
|
8.5 | IC50 | 2 | — | |
QKORYAJYXMUUGT
|
8.5 | IC50 | 2 | — | |
GHXGFAYAOFHWSA
|
8.5 | IC50 | 2 | — | |
KVVLNFCQHKOZRL
|
8.4 | IC50 | 2 | — | |
NZIMJPCYKSLDOJ
|
8.4 | IC50 | 2 | — | |
VMAXCDSINZOJPZ
|
8.3 | IC50 | 2 | — | |
DWYVTGLLPDRAAD
|
8.3 | IC50 | 3 | — | |
FIWFFXNIBNYLPJ
|
8.3 | IC50 | 3 | — | |
HBJSIJQBVFRMSX
|
8.3 | IC50 | 2 | — | |
HTFDMWIUEKMNHH
|
8.3 | IC50 | 4 | — | |
JAKMNRHMGLQOEF
|
8.3 | IC50 | 3 | — | |
JYCHMDIHDKDPNS
|
8.3 | IC50 | 3 | — | |
QJZCPMKZUHZQIV
|
8.3 | IC50 | 3 | — | |
QXILYQTXHFZFST
|
8.3 | IC50 | 3 | — |