Target Details
| UniProt AC | Q13255 |
|---|---|
| Gene Symbol | GRM1 |
| Protein Name | Metabotropic glutamate receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00003 (7tm_3) PF01094 (ANF_receptor) PF10606 (GluR_Homer-bdg) PF07562 (NCD3G) |
Summary
- Multi-target molecules 92
- Clinical molecules 0
- Avg pChEMBL 7.07
KEGG Pathways (15)
- Calcium signaling pathway
- Estrogen signaling pathway
- FoxO signaling pathway
- Gap junction
- Glutamatergic synapse
- Long-term depression
- Long-term potentiation
- Neuroactive ligand signaling
- Neuroactive ligand-receptor interaction
- Pathways of neurodegeneration - multiple diseases
- Phospholipase D signaling pathway
- Prostate cancer
- Retrograde endocannabinoid signaling
- Spinocerebellar ataxia
- Taste transduction
Associated Diseases (2)
Active Molecules (92)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VZYVQEMZRNNEBB
|
6.8 | IC50 | 2 | — | |
MRIYQDALPQSCHI
|
6.7 | IC50 | 2 | — | |
JTMQTEDUASKITJ
|
6.7 | IC50 | 2 | — | |
XMXWQEOSRWRHAD
|
6.7 | IC50 | 2 | — | |
XMBSSAPUXAATEP
|
6.7 | IC50 | 2 | — | |
TXNDLRUNCXZKOT
|
6.6 | IC50 | 2 | — | |
BWXIPDFABPPPPW
|
6.5 | IC50 | 2 | — | |
KHTQVNOASPZXBZ
|
6.5 | IC50 | 2 | — | |
WHUUTDBJXJRKMK
|
6.5 | Ki | 4 | — | |
KXEPELZEWQYLKO
|
6.5 | Ki | 2 | — | |
WHUUTDBJXJRKMK
|
6.4 | Ki | 20 | — | |
HACWSZJCCKJLHH
|
6.4 | IC50 | 2 | — | |
KWHZAURFDIUNMU
|
6.4 | IC50 | 2 | — | |
DMJNZMXZSQWBRT
|
6.4 | IC50 | 2 | — | |
VPQOPIIMLMRDJT
|
6.3 | IC50 | 2 | — | |
DNCAVIPSMHFJEK
|
6.3 | IC50 | 2 | — | |
URKBBETZPSNPJV
|
6.3 | IC50 | 2 | — | |
ZQLNLYNPYFHOMH
|
6.3 | IC50 | 2 | — | |
MBZUZSSPUFLUTF
|
6.3 | IC50 | 2 | — | |
CQQUHBDYEUOOMX
|
6.2 | IC50 | 2 | — | |
OKPWMAWSGHTGOX
|
6.2 | IC50 | 2 | — | |
VWVNXKONKNIJFU
|
6.2 | IC50 | 2 | — | |
CXTMBWBHTXAOFX
|
6.2 | IC50 | 2 | — | |
FYGXJVFGWUEFMS
|
6.2 | IC50 | 2 | — | |
KVUODOBLFAHUOE
|
6.2 | IC50 | 2 | — | |
ZDULCLFYDBDVDF
|
6.2 | IC50 | 2 | — | |
VPOBZVBTTIDGGK
|
6.2 | IC50 | 2 | — | |
KXLYHSSJUUTFEL
|
6.2 | IC50 | 2 | — | |
LGUFTKSMTYDGRD
|
6.2 | IC50 | 2 | — | |
MHCSEEMETVIDGF
|
6.2 | IC50 | 2 | — | |
NKPUWTADMNLUBA
|
6.2 | IC50 | 2 | — | |
VTJXVUYJMWDVSF
|
6.2 | IC50 | 2 | — | |
DBSRCEYBLWCRLN
|
6.2 | IC50 | 2 | — | |
FJMUBIPCGBRIPD
|
6.2 | IC50 | 2 | — | |
PTMMCLBXSOCORB
|
6.2 | IC50 | 2 | — | |
REEMCNVFTXZLSO
|
6.1 | IC50 | 2 | — | |
DOLMPPAKPUQJRP
|
6.1 | IC50 | 2 | — | |
RCNPMPFRYJOVFT
|
6.1 | IC50 | 2 | — | |
FYMJCZZKTSYDNR
|
6.1 | IC50 | 2 | — | |
GANCFFDZYNZRLX
|
6.0 | IC50 | 2 | — | |
QQBUKBJTUTUJSQ
|
6.0 | IC50 | 2 | — | |
SUZNBZLSOXCXCA
|
6.0 | IC50 | 2 | — |