Target Details
| UniProt AC | Q13255 |
|---|---|
| Gene Symbol | GRM1 |
| Protein Name | Metabotropic glutamate receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00003 (7tm_3) PF01094 (ANF_receptor) PF10606 (GluR_Homer-bdg) PF07562 (NCD3G) |
Summary
- Multi-target molecules 92
- Clinical molecules 0
- Avg pChEMBL 7.07
KEGG Pathways (15)
- Calcium signaling pathway
- Estrogen signaling pathway
- FoxO signaling pathway
- Gap junction
- Glutamatergic synapse
- Long-term depression
- Long-term potentiation
- Neuroactive ligand signaling
- Neuroactive ligand-receptor interaction
- Pathways of neurodegeneration - multiple diseases
- Phospholipase D signaling pathway
- Prostate cancer
- Retrograde endocannabinoid signaling
- Spinocerebellar ataxia
- Taste transduction
Associated Diseases (2)
Active Molecules (92)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WOADNNTWYZOWNV
|
9.0 | IC50 | 2 | — | |
FIYKKDYTSVKXEL
|
8.7 | IC50 | 2 | — | |
ATPSAOLGMWJQNL
|
8.7 | IC50 | 2 | — | |
VCUKKMIXURRDKL
|
8.5 | IC50 | 2 | — | |
TUKBLRJBXIQJPU
|
8.3 | IC50 | 2 | — | |
UKYYPMIATFNGSH
|
8.3 | IC50 | 2 | — | |
GFWSBYBQNHQKCS
|
8.2 | IC50 | 2 | — | |
DWPQODZAOSWNHB
|
8.2 | Ki | 3 | — | |
XSGFZVPHOUBKKN
|
8.2 | Ki | 2 | — | |
DUHWKHAOHAPCIH
|
8.2 | IC50 | 2 | — | |
INXYUZGZBZNQGF
|
8.2 | IC50 | 2 | — | |
OVLFPONZEJZITI
|
8.2 | IC50 | 2 | — | |
ZSBBASZUYKREPU
|
8.2 | IC50 | 2 | — | |
OVURPMRKVYGKGC
|
8.1 | IC50 | 2 | — | |
QVMIPZSIWADRIE
|
8.1 | IC50 | 2 | — | |
QQYIWENGMXJJRT
|
8.1 | IC50 | 2 | — | |
ASVIRPJBVKLRRZ
|
8.0 | IC50 | 2 | — | |
GYWGXEGOXODOQU
|
8.0 | IC50 | 2 | — | |
JMIBSVABGHKOBI
|
8.0 | IC50 | 2 | — | |
YSSBTWFASLVAGY
|
8.0 | IC50 | 5 | — | |
FVEOBLKOMQNQJN
|
7.9 | IC50 | 2 | — | |
WBNYTWXVORUJBL
|
7.8 | IC50 | 2 | — | |
ZCPJZMIIRATEAI
|
7.8 | IC50 | 2 | — | |
VWOMTTIMBHBPBI
|
7.8 | IC50 | 3 | — | |
HSEURPKENJFQMI
|
7.8 | IC50 | 2 | — | |
FHPVPCRSNMYQFP
|
7.7 | IC50 | 2 | — | |
UIRMNVOEQMAKFM
|
7.7 | IC50 | 7 | — | |
JAIOFGJWUSFJQH
|
7.7 | IC50 | 2 | — | |
DTWANULJDRVTFI
|
7.6 | IC50 | 5 | — | |
ZDHUMLUZTXYHOB
|
7.6 | IC50 | 2 | — | |
ASNFTDCKZKHJSW
|
7.5 | Ki | 5 | — | |
SWPVFHZSTTYORI
|
7.5 | IC50 | 5 | — | |
GGNUBGHBZKNFOS
|
7.5 | IC50 | 2 | — | |
QXXCGFFXNAYIRR
|
7.5 | IC50 | 2 | — | |
NEWKHUASLBMWRE
|
7.4 | Ki | 4 | — | |
BKXZRLFPGYWHTM
|
7.4 | IC50 | 7 | — | |
ZCUSHDLLJXLSPP
|
7.4 | IC50 | 2 | — | |
GRTPVLUWVUWRRC
|
7.4 | IC50 | 2 | — | |
XGWUUIBWCCASNG
|
7.3 | IC50 | 2 | — | |
AKQCXZGTHURUGU
|
7.1 | IC50 | 2 | — | |
OYLCIUHGUBNPFB
|
7.1 | IC50 | 2 | — | |
YRTJBUGCGGXTRV
|
7.1 | IC50 | 5 | — | |
MSOYXZGDANCFCO
|
7.0 | IC50 | 2 | — | |
NZPDJEQFQMMJCR
|
7.0 | IC50 | 2 | — | |
VYUFFNORDHWOJK
|
7.0 | IC50 | 2 | — | |
BSXAXDHXYFYFPY
|
7.0 | IC50 | 3 | — | |
YYVZSQMPPRXPRD
|
6.8 | IC50 | 2 | — | |
MDTAHECBRZZGJE
|
6.8 | IC50 | 2 | — | |
RCCMXKJGURLWPB
|
6.8 | Ki | 4 | — | |
CVIRWLJKDBYYOG
|
6.8 | IC50 | 2 | — |