Target Details
| UniProt AC | Q13233 |
|---|---|
| Gene Symbol | MAP3K1 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21040 (CEP104-like_TOG) PF00069 (Pkinase) PF04434 (SWIM) |
Summary
- Multi-target molecules 188
- Clinical molecules 4
- Avg pChEMBL 7.38
KEGG Pathways (9)
Associated Diseases (1)
Active Molecules (188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZXRMCWVMPXUCJH
|
6.7 | IC50 | 3 | — | |
JPOHYOWEEKRRJK
|
6.6 | IC50 | 3 | — | |
OZZKFBLHUBAGEQ
|
6.6 | IC50 | 3 | — | |
YVFAWXDKCQRMPA
|
6.6 | IC50 | 3 | — | |
BOUKILWEXWLSRJ
|
6.6 | IC50 | 3 | — | |
VOSBQMIZOZZEBZ
|
6.6 | IC50 | 3 | — | |
FJCQZSRKMFPCOW
|
6.6 | IC50 | 3 | — | |
NKWJABPDWZOARV
|
6.6 | IC50 | 3 | — | |
LTXXWWCTWJCQQL
|
6.6 | IC50 | 3 | — | |
BKWCDRNUXDVCQV
|
6.6 | IC50 | 3 | — | |
RXYXZBWUKQLVKR
|
6.6 | IC50 | 3 | — | |
IUEPNGJGSBBBHF
|
6.5 | IC50 | 3 | — | |
OXHGKUOZRLFONP
|
6.5 | IC50 | 3 | — | |
JGXHQMQPGIDNQB
|
6.5 | IC50 | 3 | — | |
RNRYJOIXVZVCNT
|
6.5 | IC50 | 3 | — | |
LMMJFBMMJUMSJS
|
6.5 | IC50 | 5 | — | |
AFPAJDOKDKWGGI
|
6.5 | IC50 | 3 | — | |
MTLRPYAACHUORY
|
6.5 | IC50 | 3 | — | |
COTQMNHTEKDUSB
|
6.5 | IC50 | 3 | — | |
DAHOKVXQXIXZEY
|
6.5 | IC50 | 3 | — | |
REOWJUIZCQXSQH
|
6.5 | IC50 | 3 | — | |
WLGLAXWJUWQYEQ
|
6.5 | IC50 | 3 | — | |
VOURFPDYANCOLP
|
6.4 | IC50 | 3 | — | |
XUMQXLFNDALQFY
|
6.4 | IC50 | 3 | — | |
GUGQTZDITULCAM
|
6.4 | IC50 | 3 | — | |
OGTULHQQFZVXGB
|
6.4 | IC50 | 3 | — | |
HKSZLNNOFSGOKW
|
6.4 | IC50 | 408 | — | |
YHATZJNTNYXLOB
|
6.3 | IC50 | 3 | — | |
FNHKPVJBJVTLMP
|
6.3 | Kd | 29 | — | |
JDBMWHCBKTXEIL
|
6.3 | IC50 | 3 | — | |
PHXJVRSECIGDHY
|
6.3 | Kd | 59 | — | |
TVOFCCIKXFMAKW
|
6.3 | IC50 | 3 | — | |
XKFTZKGMDDZMJI
|
6.3 | Kd | 64 | Yes | |
HQTKAIDPYRFHMI
|
6.2 | IC50 | 3 | — | |
QDXQGTXUKDYEBI
|
6.1 | IC50 | 3 | — | |
JEIJQBSAHGKSHC
|
6.1 | IC50 | 3 | — | |
QSDVZPULRUJSBC
|
6.1 | IC50 | 4 | — | |
KKORZXWRRHLIMN
|
6.1 | IC50 | 3 | — |