Target Details
| UniProt AC | Q13233 |
|---|---|
| Gene Symbol | MAP3K1 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21040 (CEP104-like_TOG) PF00069 (Pkinase) PF04434 (SWIM) |
Summary
- Multi-target molecules 188
- Clinical molecules 4
- Avg pChEMBL 7.38
KEGG Pathways (9)
Associated Diseases (1)
Active Molecules (188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NEHSGKZSBWLRCZ
|
7.3 | IC50 | 3 | — | |
KWSIGBRAMTYPHR
|
7.3 | IC50 | 3 | — | |
OGFOENLUWIJPAQ
|
7.3 | IC50 | 3 | — | |
XKJZAXRHJJVTOB
|
7.3 | IC50 | 3 | — | |
IOYRVIKODRKVSN
|
7.2 | IC50 | 3 | — | |
PLWVNCSSFNLWHM
|
7.2 | IC50 | 3 | — | |
FYVWDSXUBVIRLZ
|
7.2 | IC50 | 3 | — | |
WFLXIWOCFBMJNU
|
7.2 | IC50 | 2 | — | |
OTUVOFAIBFSMKE
|
7.2 | IC50 | 3 | — | |
QJRCOIYPHTWFQW
|
7.2 | IC50 | 3 | — | |
IWUMUNQLJUUETN
|
7.2 | IC50 | 3 | — | |
MSWUJKZTIFJSKD
|
7.2 | IC50 | 3 | — | |
HDJNFIJEBGMBCW
|
7.1 | IC50 | 3 | — | |
YYNHOTVNSZCMHV
|
7.1 | IC50 | 3 | — | |
IOSBNDVPSNIAPM
|
7.1 | IC50 | 3 | — | |
KSKCPNLILMFPES
|
7.1 | IC50 | 3 | — | |
ODEYDNDAGZWGHG
|
7.1 | IC50 | 3 | — | |
KDVBIOIYBMCFJP
|
7.1 | IC50 | 3 | — | |
MEPYJUWXGSNWDU
|
7.1 | IC50 | 3 | — | |
SWHQVOZRMNFELZ
|
7.1 | IC50 | 3 | — | |
VHFTYKJUELSQJS
|
7.1 | IC50 | 3 | — | |
ODEYDNDAGZWGHG
|
7.0 | IC50 | 3 | — | |
FVFORBHNFLVKQY
|
7.0 | IC50 | 3 | — | |
YLFYLSDYLABJKV
|
7.0 | IC50 | 3 | — | |
HHCBMISMPSAZBF
|
7.0 | IC50 | 23 | — | |
UUICRMJNOIDISB
|
7.0 | IC50 | 3 | — | |
WVUNYSQLFKLYNI
|
7.0 | Kd | 46 | Yes | |
HXALSNAYPNDDSO
|
7.0 | IC50 | 3 | — | |
XHKSUXGHCHDDJK
|
7.0 | IC50 | 3 | — | |
GJFBRQSLUZVDGK
|
7.0 | IC50 | 3 | — | |
UBPYILGKFZZVDX
|
7.0 | Kd | 130 | Yes | |
ZHJGWYRLJUCMRT
|
7.0 | Kd | 18 | — | |
LXLMKDYNQSTBFW
|
6.9 | IC50 | 3 | — | |
OQADNYQXVWLBPF
|
6.9 | IC50 | 3 | — | |
NUSWWDDYQRQFHO
|
6.9 | IC50 | 3 | — | |
JKPCWAYLRAJUNU
|
6.9 | IC50 | 3 | — | |
RZQMSENSUWINNW
|
6.9 | IC50 | 3 | — | |
XCDDJSDCNNSGEH
|
6.9 | IC50 | 3 | — | |
CSAPGOSLBLMIPS
|
6.9 | IC50 | 3 | — | |
HXHAJRMTJXHJJZ
|
6.9 | Kd | 52 | Yes | |
KJPIZTFQJJVHTA
|
6.9 | IC50 | 3 | — | |
PCTIECVOHLCQSU
|
6.9 | IC50 | 3 | — | |
KPIKBRJPWVYBJZ
|
6.8 | IC50 | 3 | — | |
VTZVVDZIRWWZJR
|
6.8 | IC50 | 3 | — | |
OLLSPENBOWNTBY
|
6.7 | IC50 | 3 | — | |
SIBULRRGAQTCNA
|
6.7 | IC50 | 3 | — | |
JMFSLLJECHALSO
|
6.7 | IC50 | 3 | — | |
FPFBRLFCFHRESP
|
6.7 | IC50 | 3 | — | |
AIENEURRWLHMLD
|
6.7 | IC50 | 3 | — | |
YSOXURBNXLFBCL
|
6.7 | IC50 | 3 | — |