Target Details
| UniProt AC | Q13233 |
|---|---|
| Gene Symbol | MAP3K1 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21040 (CEP104-like_TOG) PF00069 (Pkinase) PF04434 (SWIM) |
Summary
- Multi-target molecules 188
- Clinical molecules 4
- Avg pChEMBL 7.38
KEGG Pathways (9)
Associated Diseases (1)
Active Molecules (188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QUBGEHFUYLWZSU
|
7.9 | IC50 | 3 | — | |
XJDANWRYPRBMQG
|
7.9 | IC50 | 3 | — | |
CAEVAIJWIJNLRN
|
7.8 | IC50 | 3 | — | |
LGBJHKOWLHCKDD
|
7.8 | IC50 | 3 | — | |
LTRIGNNYJQRLEJ
|
7.8 | IC50 | 3 | — | |
SGZHLFXKVNMWRZ
|
7.8 | IC50 | 3 | — | |
BGLWMTSHLFRIJS
|
7.8 | IC50 | 3 | — | |
HKCOWFAZOPDVRG
|
7.8 | IC50 | 3 | — | |
LOPFFGYJBIMBSE
|
7.8 | IC50 | 3 | — | |
AMURVXAYQGXAHX
|
7.7 | IC50 | 3 | — | |
VTFKWORYPCZIMJ
|
7.7 | IC50 | 3 | — | |
CHVGFSQLXGYINP
|
7.7 | IC50 | 3 | — | |
KDGGEXSGBVHGBQ
|
7.7 | IC50 | 3 | — | |
ODEYDNDAGZWGHG
|
7.7 | IC50 | 3 | — | |
OQPWKRIFJWBPSI
|
7.7 | IC50 | 3 | — | |
IHWHZUVPXIRKBX
|
7.7 | IC50 | 2 | — | |
SCRBPYXFLBEPGI
|
7.7 | IC50 | 3 | — | |
XSGBYNRBLKXGAM
|
7.7 | IC50 | 3 | — | |
KKCJMVOTVSOBJV
|
7.6 | IC50 | 3 | — | |
MUXRNPAKNHSLBA
|
7.6 | IC50 | 3 | — | |
DYPFTHVSPQWZLZ
|
7.6 | IC50 | 3 | — | |
SGSOHKXRUURWTO
|
7.6 | IC50 | 3 | — | |
ZGWQEJGAIHLJAW
|
7.6 | IC50 | 2 | — | |
BMPYEMYLYOLWFA
|
7.5 | IC50 | 3 | — | |
LMWLLHDHDDTUEP
|
7.5 | IC50 | 3 | — | |
MUWRTVLHQJDEDE
|
7.5 | IC50 | 3 | — | |
XUHYQVAQOGSJTJ
|
7.5 | IC50 | 3 | — | |
MWUFVYLAWAXDHQ
|
7.5 | IC50 | 2 | — | |
NWKVBUTWVCHMAL
|
7.5 | IC50 | 3 | — | |
TZSUJFHSWGXSAL
|
7.5 | IC50 | 3 | — | |
GWNDZYBUJRBHJC
|
7.5 | IC50 | 3 | — | |
XXYXZSAPTFLBKY
|
7.5 | IC50 | 3 | — | |
PLDLSGBXZGLUTQ
|
7.5 | IC50 | 3 | — | |
QKHAXMNYKRGEFU
|
7.5 | IC50 | 3 | — | |
ZTWYLYKACYNBBZ
|
7.5 | IC50 | 3 | — | |
FHOMOWNRVSMFRC
|
7.5 | IC50 | 3 | — | |
YUNJOJPTHYKRCY
|
7.4 | IC50 | 3 | — | |
ALLVOVRKMVXXDY
|
7.4 | IC50 | 3 | — | |
NYDBSTFAISDDAE
|
7.4 | IC50 | 3 | — | |
QUIWMANKWJDNGK
|
7.4 | IC50 | 2 | — | |
QUPOXIBOWFOVQM
|
7.4 | IC50 | 3 | — | |
ZDACFCFMMWTLTA
|
7.3 | IC50 | 9 | — | |
GPQZSOKVRXFLTO
|
7.3 | IC50 | 3 | — | |
XLNYFDGIIRQJMP
|
7.3 | IC50 | 3 | — | |
RUGZAGYYZGVWBZ
|
7.3 | IC50 | 3 | — | |
SZWMQRVECIKICL
|
7.3 | IC50 | 3 | — | |
MBLVLWZXURYDFW
|
7.3 | IC50 | 3 | — | |
UPUBHFBOYYXILS
|
7.3 | IC50 | 3 | — | |
OIEYGVGFYHDQFP
|
7.3 | IC50 | 3 | — | |
BKMQVXMXPSFWIB
|
7.3 | IC50 | 3 | — |