Target Details
| UniProt AC | Q13233 |
|---|---|
| Gene Symbol | MAP3K1 |
| Protein Name | Mitogen-activated protein kinase kinase kinase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF21040 (CEP104-like_TOG) PF00069 (Pkinase) PF04434 (SWIM) |
Summary
- Multi-target molecules 188
- Clinical molecules 4
- Avg pChEMBL 7.38
KEGG Pathways (9)
Associated Diseases (1)
Active Molecules (188)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GSSSJMXLSDAINU
|
9.0 | IC50 | 3 | — | |
MRONWWYUJGYEFK
|
9.0 | IC50 | 3 | — | |
TXRDPXPHKUXGQL
|
9.0 | IC50 | 3 | — | |
GFOXCTULQRSDEP
|
8.7 | IC50 | 3 | — | |
MWLIRBVDTHSBRM
|
8.7 | IC50 | 2 | — | |
NJSXKZAXYUNSFP
|
8.7 | IC50 | 3 | — | |
OHRLRWVLPBHNJE
|
8.7 | IC50 | 3 | — | |
UTEIFOJYUWWJFJ
|
8.7 | IC50 | 3 | — | |
WHQSHUVXTQTMMK
|
8.7 | IC50 | 2 | — | |
XLXDRLLBZCUGME
|
8.7 | IC50 | 3 | — | |
KXEFWEJDWLGBJH
|
8.5 | IC50 | 3 | — | |
QNTGJAKMNSBSBC
|
8.5 | IC50 | 3 | — | |
MEMXIDIPZZGONE
|
8.4 | IC50 | 3 | — | |
MZRCKIBDAXSKTH
|
8.4 | IC50 | 3 | — | |
UAFZNGTVQDQROK
|
8.4 | IC50 | 3 | — | |
YLQUXDOVSUUPRE
|
8.4 | IC50 | 3 | — | |
ARPRCGHYASNNQS
|
8.3 | IC50 | 3 | — | |
CEANXZMNDMARKN
|
8.3 | IC50 | 3 | — | |
CIKANSHRRQAREB
|
8.3 | IC50 | 3 | — | |
FWQJRYBMLTWKKN
|
8.3 | IC50 | 3 | — | |
GLOUSHGJLYWNJY
|
8.3 | IC50 | 3 | — | |
GUAIRYVTDVHCNC
|
8.3 | IC50 | 3 | — | |
IVLPNLXFDCHLKA
|
8.3 | IC50 | 3 | — | |
IRCLZLJAEFQVQA
|
8.2 | IC50 | 2 | — | |
MLELTKLIDNFCOS
|
8.2 | IC50 | 3 | — | |
MQQWOJADUXWJBJ
|
8.2 | IC50 | 3 | — | |
RSMGUCWXMLOUPS
|
8.2 | IC50 | 2 | — | |
SELMBQSIGDYSEC
|
8.2 | IC50 | 3 | — | |
FRLQZRDDFJVTJS
|
8.2 | IC50 | 3 | — | |
NNHZDYBLENYVRI
|
8.2 | IC50 | 3 | — | |
SUDAHWBOROXANE
|
8.2 | IC50 | 6 | — | |
UYEYSWPYMREJSD
|
8.2 | IC50 | 3 | — | |
ANPIINUOZKZYFD
|
8.1 | IC50 | 3 | — | |
BCASZHPJDWDMSA
|
8.1 | IC50 | 3 | — | |
LNQFHCFBVWZBDV
|
8.1 | IC50 | 2 | — | |
NFDHPUYCJNANAA
|
8.1 | IC50 | 3 | — | |
QHNDLISOJCGFBM
|
8.1 | IC50 | 3 | — | |
QSENMPAGYMUVDE
|
8.1 | IC50 | 5 | — | |
YKYFNNNNXYBCDU
|
8.1 | IC50 | 3 | — | |
HEVHEWAKLRICCA
|
8.1 | IC50 | 3 | — | |
GRZCUOLWBQKOEY
|
8.0 | IC50 | 3 | — | |
GZEKNZXQCOKIPI
|
8.0 | IC50 | 3 | — | |
MAEIMZUQBHFKFG
|
8.0 | IC50 | 3 | — | |
DVSZEHUFBBJQKJ
|
8.0 | IC50 | 3 | — | |
SGCQOTWECLPFOA
|
8.0 | IC50 | 3 | — | |
CBVUTXWXSYHWDW
|
7.9 | IC50 | 3 | — | |
YRKLUPVSKKKSFY
|
7.9 | IC50 | 3 | — | |
DNFMTAJPYCSJJR
|
7.9 | IC50 | 3 | — | |
KVLZSRGASWOICS
|
7.9 | IC50 | 3 | — | |
OZMFPIJIZRXMPR
|
7.9 | IC50 | 3 | — |