Target Details
| UniProt AC | Q13188 |
|---|---|
| Gene Symbol | STK3 |
| Protein Name | Serine/threonine-protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11629 (Mst1_SARAH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 285
- Clinical molecules 27
- Avg pChEMBL 6.72
KEGG Pathways (4)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KTEIFNKAUNYNJU
|
6.1 | Ki | 48 | — | |
MADCXGNPDBWPLM
|
6.1 | Ki | 25 | — | |
MFMXAWQGPQXDRJ
|
6.1 | Ki | 27 | — | |
MMFBBQQGBVPLQQ
|
6.1 | Ki | 13 | — | |
NRZYTPAJGVTKIM
|
6.1 | Ki | 38 | — | |
ORUUEFDGYYTXAF
|
6.1 | Ki | 26 | — | |
PJSBFZAYJQMORO
|
6.1 | Ki | 11 | — | |
PTVPBWWDGZSEAF
|
6.1 | Ki | 63 | — | |
RIDCOBPCGROHQY
|
6.1 | Ki | 4 | — | |
SAOVTENLRUIQAM
|
6.1 | IC50 | 2 | — | |
SPMHGQZFMNZCBV
|
6.1 | Ki | 30 | Yes | |
ZGZVRPRSFXRGCF
|
6.1 | Ki | 76 | — | |
DTEKTGDVSARYDS
|
6.1 | IC50 | 11 | — | |
ODPGGGTTYSGTGO
|
6.1 | Kd | 153 | — | |
PDOQBOJDRPLBQU
|
6.1 | Kd | 21 | — | |
ZCBUQCWBWNUWSU
|
6.0 | Kd | 59 | — | |
XIVPVCPBGAFXJA
|
6.0 | IC50 | 2 | — | |
ACNCCUVYXQGPKZ
|
6.0 | Ki | 31 | — | |
GWMATETWMAQOFL
|
6.0 | Ki | 36 | — | |
HKZKELVPGXJIMW
|
6.0 | Ki | 41 | — | |
HSMUWLLZAZCLHF
|
6.0 | Ki | 25 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
KAKGFGCTONHQJW
|
6.0 | Ki | 25 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KTEIFNKAUNYNJU
|
6.0 | Kd | 114 | — | |
LJKJYKWDLJUZHA
|
6.0 | Ki | 24 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MASJMHFQMYAPJR
|
6.0 | Ki | 41 | — | |
NFKMFNBKEOQNPZ
|
6.0 | Ki | 43 | — | |
NRGYZNJPCGRCLV
|
6.0 | Ki | 52 | — | |
QJIVDCJIPGAKQZ
|
6.0 | Ki | 25 | — | |
RWKDVIAVTRRJIR
|
6.0 | Ki | 23 | — | |
ULVWJFBHQIXEPE
|
6.0 | Ki | 10 | — | |
XXSPHNFKLDJDAK
|
6.0 | Ki | 26 | — | |
ZAARMHXLYCHRAK
|
6.0 | Ki | 20 | — |