Target Details
| UniProt AC | Q13188 |
|---|---|
| Gene Symbol | STK3 |
| Protein Name | Serine/threonine-protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11629 (Mst1_SARAH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 285
- Clinical molecules 27
- Avg pChEMBL 6.72
KEGG Pathways (4)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NZVDDFRUBIEKLV
|
6.3 | Ki | 20 | — | |
OPLHMHMCXQXEQG
|
6.3 | Ki | 10 | — | |
SRONQUHCRFZABC
|
6.3 | Ki | 28 | — | |
UOOZSMNSBYVUGZ
|
6.3 | Ki | 32 | — | |
USHMNZBDAOGLMB
|
6.3 | Ki | 26 | — | |
VQPBIJGXSXEOCU
|
6.3 | Ki | 24 | — | |
WZISGNDZZPSYRP
|
6.3 | Ki | 20 | — | |
GCIKSSRWRFVXBI
|
6.3 | Kd | 109 | Yes | |
CVJJGKHSVZTCSY
|
6.3 | IC50 | 2 | — | |
DEUHRYNUMMEYHI
|
6.3 | IC50 | 2 | — | |
DIABFIQALHQONE
|
6.3 | IC50 | 2 | — | |
IBOVLFFYQWKZFN
|
6.3 | IC50 | 2 | — | |
LBWANVYGDFHTRC
|
6.3 | IC50 | 2 | — | |
LZVQWGYDMCTNJC
|
6.3 | IC50 | 2 | — | |
MIURWHKJMYMLCP
|
6.3 | IC50 | 2 | — | |
MPDAGVPGHCHPMC
|
6.3 | IC50 | 2 | — | |
MXEUNJLZLFMHOA
|
6.3 | IC50 | 2 | — | |
NEWMPWSBRISBBJ
|
6.3 | IC50 | 2 | — | |
PDUOASXHLKZWEN
|
6.3 | IC50 | 2 | — | |
PRZMXPRPGHYMHN
|
6.3 | IC50 | 2 | — | |
RIUCXIZLRCRCFO
|
6.3 | IC50 | 2 | — | |
UHKXLPHLKSGYPI
|
6.3 | IC50 | 2 | — | |
VNHDCNPUZFAZKU
|
6.3 | IC50 | 2 | — | |
VWNJEWMXAGIYCW
|
6.3 | IC50 | 2 | — | |
YLYXECAEEDEGIO
|
6.3 | IC50 | 2 | — | |
ZSBOVIKNCKVUHX
|
6.3 | IC50 | 2 | — | |
ZWDUUSQSMVRZHV
|
6.2 | IC50 | 3 | — | |
JPOSFPUHBHRUAX
|
6.2 | IC50 | 40 | Yes | |
AWDORCFLUJZUQS
|
6.2 | Ki | 22 | — | |
BPNUQXPIQBZCMR
|
6.2 | Ki | 60 | — | |
DJLORVJVWIBDME
|
6.2 | Ki | 24 | — | |
GQERVRMWWVZZDB
|
6.2 | IC50 | 2 | — | |
HEUSUIRCBWROMH
|
6.2 | Ki | 64 | — | |
LYNBNVBMAGDJRW
|
6.2 | Ki | 81 | — | |
MMMPFWNSQKXKDX
|
6.2 | Ki | 14 | — | |
MTCHQDWUHQADSY
|
6.2 | Ki | 29 | — | |
NHFDRBXTEDBWCZ
|
6.2 | Ki | 41 | — | |
PJUVRETYCLPAFV
|
6.2 | Ki | 20 | — | |
QQUXFYAWXPMDOE
|
6.2 | Ki | 31 | — | |
UXMNYFJHEBEDJS
|
6.2 | Ki | 19 | Yes | |
WUWDLXZGHZSWQZ
|
6.2 | Ki | 41 | — | |
FWEIAKDAIDQPRK
|
6.2 | IC50 | 2 | — | |
XKZQZMSAWVDRSP
|
6.2 | IC50 | 39 | Yes | |
NRSGWEVTVGZDFC
|
6.2 | IC50 | 50 | — | |
DYNHJHQFHQTFTP
|
6.1 | Kd | 38 | — | |
QZZMUIJVVAGHJA
|
6.1 | IC50 | 3 | — | |
TZWUTAYHWCWNFP
|
6.1 | IC50 | 3 | — | |
GLMWKEAUVZDGKE
|
6.1 | Ki | 23 | — | |
GWJHMRBQEUHFOC
|
6.1 | Ki | 42 | — | |
IFPPYSWJNWHOLQ
|
6.1 | Ki | 52 | Yes |