Target Details
| UniProt AC | Q13188 |
|---|---|
| Gene Symbol | STK3 |
| Protein Name | Serine/threonine-protein kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF11629 (Mst1_SARAH) PF00069 (Pkinase) |
Summary
- Multi-target molecules 285
- Clinical molecules 27
- Avg pChEMBL 6.72
KEGG Pathways (4)
Active Molecules (285)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XPHWIERLJBFPFV
|
6.6 | Ki | 69 | — | |
YMIJUBCSOKSFRU
|
6.6 | Ki | 87 | — | |
ZHRYDDVDLCQYQA
|
6.6 | Ki | 5 | — | |
AXVWXYOCYXZGCZ
|
6.6 | IC50 | 3 | — | |
XRCXPEPDTZGHNO
|
6.6 | IC50 | 2 | — | |
FZIPVCYYDYBQOZ
|
6.6 | IC50 | 2 | — | |
RCRFSYHNZNAAKZ
|
6.6 | IC50 | 2 | — | |
YDRMVAPJCHICGE
|
6.5 | IC50 | 2 | — | |
QQWUGDVOUVUTOY
|
6.5 | Kd | 231 | Yes | |
VXBAJLGYBMTJCY
|
6.5 | Kd | 34 | Yes | |
AYJBHLUSGLQYDG
|
6.5 | Ki | 16 | — | |
CHADTINFLWZSKR
|
6.5 | Ki | 26 | — | |
DPRGOXVMSNDADU
|
6.5 | Ki | 16 | — | |
KAKFXRYHYUPXSU
|
6.5 | Ki | 16 | — | |
KRIUNPBAQZGFQA
|
6.5 | Ki | 76 | — | |
LVECPYVAIBNSRV
|
6.5 | Ki | 33 | — | |
NXNQLECPAXXYTR
|
6.5 | Ki | 29 | — | |
QONPPIZSNSSCSK
|
6.5 | Ki | 45 | Yes | |
SKKRZILJUKYLJS
|
6.5 | Ki | 25 | — | |
UYGYYOIUVFMGKQ
|
6.5 | Ki | 30 | — | |
VUHZDNOPEVGHEO
|
6.5 | Ki | 29 | — | |
NMUOPBMRTBMZGB
|
6.5 | IC50 | 2 | — | |
QGACVLPEELTUQG
|
6.5 | IC50 | 2 | — | |
XZKDYHDTDSBKKV
|
6.5 | IC50 | 2 | — | |
UBPYILGKFZZVDX
|
6.4 | Kd | 130 | Yes | |
AIQDZMUPVYDVLB
|
6.4 | Ki | 48 | — | |
FQYLJBVSYHZWLT
|
6.4 | Ki | 35 | Yes | |
GCBJDOWIQHMCMR
|
6.4 | Ki | 84 | — | |
HNODKCFEFLQKBO
|
6.4 | Ki | 6 | — | |
KTWBYGUSEYSRND
|
6.4 | Ki | 28 | — | |
LGHBDVLAHHANMX
|
6.4 | Ki | 53 | — | |
QPORZABOFXPRHM
|
6.4 | Ki | 18 | — | |
RITAVMQDGBJQJZ
|
6.4 | Ki | 33 | — | |
UDFDIIVNIYWXDM
|
6.4 | Ki | 74 | — | |
XJSFDMGICAWQFS
|
6.4 | Ki | 60 | — | |
XKFTZKGMDDZMJI
|
6.4 | Ki | 56 | — | |
UJLAWZDWDVHWOW
|
6.3 | Kd | 4 | — | |
ALKJNCZNEOTEMP
|
6.3 | Kd | 55 | — | |
ZTSOUDMNSOYCTG
|
6.3 | IC50 | 10 | — | |
PIQCTGMSNWUMAF
|
6.3 | Kd | 137 | Yes | |
SJUNPBBKTNPXAO
|
6.3 | IC50 | 2 | — | |
ACSYKUPGCXYRRO
|
6.3 | Ki | 26 | — | |
CFIBXVQLBVNOHW
|
6.3 | Ki | 64 | — | |
DFMCXVONDDGQIY
|
6.3 | Ki | 66 | — | |
DZSUJUOJJJCWGG
|
6.3 | Ki | 55 | Yes | |
FUSGHFKTWQRWPV
|
6.3 | Ki | 4 | — | |
KEZAHTDTAWUZDU
|
6.3 | Ki | 8 | — | |
LRZYYIZFBXFSJB
|
6.3 | Ki | 69 | — | |
MQRDVGBWWVWMEN
|
6.3 | Ki | 47 | — | |
MZDKLVOWGIOKTN
|
6.3 | Ki | 80 | — |